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Results for "

hypoxia/reoxygenation (H/R)-treated brain

" in MedChemExpress (MCE) Product Catalog:

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7306

Inhibitors & Agonists

Screening Libraries

Fluorescent Dye

243

Biochemical Assay Reagents

845

Peptides

MCE Kits

129

Inhibitory Antibodies

833

Natural
Products

982

Recombinant Proteins

646

Isotope-Labeled Compounds

337

Antibodies

Click Chemistry

334

Oligonucleotides

Targets Recommended: HIF/HIF Prolyl-Hydroxylase

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-157088

C105SR	Caspase Apoptosis Cyclophilin	Others
C105SR is a cyclophilin D (CypD) inhibitor targeting to peptidyl-prolylcis-trans isomerase (PPIase). C105SR inhibits mitochondrial permeability transition opening (mPTP) with an IC ₅₀ of 5 nM. C105SR inhibits hypoxia and reoxygenation inudced hepatocyte apoptosis and increases the level of calcium retention capacity (CRC). C105SR exhibits hepaprotective effect in ischaemia-reperfusion injury (IRI) mouse model .

HY-N2506

Ginsenoside Ra1	Others	Cardiovascular Disease
Ginsenoside Ra1 is a component from ginseng, inhibits protein tyrosine kinase (PTK) activation induced by hypoxia/reoxygenation .

HY-N0272

Eleutheroside E 2 Publications Verification	Apoptosis NF-κB	Neurological Disease Inflammation/Immunology
Eleutheroside E is an important component of ginseng that can be taken orally. Eleutheroside E has anti-inflammatory and antioxidant properties, and it helps reduce apoptosis in heart cells caused by hypoxia-reoxygenation (H/R) damage. Eleutheroside E can improve type 2 diabetes, enhance cognitive function, and has neuroprotective effects .

HY-P4439

H-Met-Val-OH	Amino Acid Derivatives	Neurological Disease
H-Met-Val-OH is a dipeptide containing free N-terminal methionine. H-Met-Val-OH exhibits activity against cDNA expressing Flavin-containing monooxygenase (FMO) 1 and FMO3. H-Met-Val-OH has potential applications in the growth of neuritis .

HY-170774

Hypoxia inducer-1	Apoptosis Reactive Oxygen Species (ROS)	Cardiovascular Disease
Hypoxia inducer-1 (Compound N6) is an orally active hypoxia activated nitric oxide (NO) donor compound. Hypoxia inducer-1 exhibits highly selective NO release under hypoxic conditions and inhibits hypoxia-induced apoptosis, necrosis, and the increase in ROS levels. Hypoxia inducer-1 regulates vascular dilation and has a protective effect in a mouse model of myocardial hypoxia injury. Hypoxia inducer-1 can be used in the research of coronary heart disease .

HY-127022

Anisodine Daturamine; α-Hydroxyscopolamine	mAChR Calcium Channel Reactive Oxygen Species (ROS)	Neurological Disease
Anisodine (Daturamine) is a neuroprotective compound that reduces exacerbated M1, M2, M4, and M5 receptor expression in brain tissues under hypoxia/reoxygenation conditions. Anisodine inhibits calcium ion influx and *reactive oxygen* species (ROS)*levels. Anisodine leads to decreased aspartate levels during hypoxia* .

HY-127022A

Anisodine hydrobromide Daturamine hydrobromide; α-Hydroxyscopolamine hydrobromide	mAChR Calcium Channel Reactive Oxygen Species (ROS)	Neurological Disease
Anisodine (Daturamine) hydrobromide is a neuroprotective compound that reduces exacerbated M1, M2, M4, and M5 receptor expression in brain tissues under hypoxia/reoxygenation conditions. Anisodine hydrobromide inhibits calcium ion influx and *reactive oxygen* species (ROS)*levels. Anisodine hydrobromide leads to decreased aspartate levels during hypoxia* .

HY-106110

OP-2507	Prostaglandin Receptor	Metabolic Disease
OP-2507 is a prostacyclin analog. OP-2507 can increase brain glucose levels in mice, suppress the breakdown of energy metabolism under hypoxic conditions, and has a protective effect against changes in cyclic nucleotides in hypoxic brain tissue (specifically, an increase in cyclic AMP and a decrease in cyclic GMP). OP-2507 provides protective effects against brain hypoxia and edema .

HY-134571

Brain Extract Total	Biochemical Assay Reagents	Neurological Disease
Brain Extract Total is a natural brain total lipid extract that can be used to prepare neuronal membranes. Brain Extract Total can be used for the study of Alzheimer's disease .

HY-P4658

H-Val-Ala-pNA	Dipeptidyl Peptidase	Others
H-Val-Ala-pNA is a substrate for the dipeptide aminopeptidase (DPAPase) of Streptococcus bovis. H-Val-Ala-pNA can be used to measure the activity of the protease .

HY-P4554

H-Phe-Arg-OH	Endogenous Metabolite	Metabolic Disease
H-Phe-Arg-OH is a dipeptide containing phenylalanine and arginine. H-Phe-Arg-OH can be separated from Bradykinin (HY-P0206) through Angiotensin-converting enzyme (ACE, HY-P2983). H-Phe-Arg-OH can be used for metabolic research .

HY-P4553

H-Met-Pro-OH	Amino Acid Derivatives	Others
H-Met-Pro-OH is a dipeptide containing methionine and proline. H-Met-Pro-OH is a substrate for aminopeptidase P (APP) and skin fibroblast prolidase .

HY-P4531

H-Ser-Tyr-OH	Opioid Receptor	Neurological Disease
H-Ser-Tyr-OH is a dipeptide consisting of glutamic acid, glycine and histidine. H-Ser-Tyr-OH can form a copper(II) complex with copper ions to form a strong free radical scavenging activity. H-Ser-Tyr-OH also increases the intracellular uptake of the delta opioid receptor ligand deltorphin .

HY-P4648

H-Trp-Trp-Trp-OH	Bacterial	Infection
H-Trp-Trp-Trp-OH is a tripeptide consisting of tryptophan. H-Trp-Trp-Trp-OH has antibacterial activity .

HY-P4654

H-Tyr-Lys-OH	Angiotensin-converting Enzyme (ACE)	Others
H-Tyr-Lys-OH is a dipeptide that can be used as a biomarker for AJH-1. H-Tyr-Lys-OH has a good binding affinity to angiotensin converting enzyme (ACE) .

HY-P4296

H-Gly-Sar-Sar-OH	Amino Acid Derivatives	Others
H-Gly-Sar-Sar-OH is an orally active tripeptide. H-Gly-Sar-Sar-OH is transported through PepT1 within Caco-2 cells. H-Gly Sar Sar OH has potential applications in material transportation .

HY-P4287

H-Gly-Lys-Gly-OH	Amino Acid Derivatives	Others
H-Gly-Lys-Gly-OH is a tripeptide containing glycine and lysine. H-Gly-Lys-Gly-OH can be used for the synthesis of casein and soybean protein .

HY-P4486

H-Pro-Gly-Pro-OH	Drug Derivative	Others
H-Pro-Gly-Pro-OH is a collagen-derived matrikine that has classically been described as a neutrophil chemoattractant. H-Pro-Gly-Pro-OH is perfectly positioned to focus neutrophils on the site required and direct a localized repair response. H-Pro-Gly-Pro-OH activates the transcription of neurotrophins and their receptor genes after cerebral ischemia .

HY-P4294

H-Gly-Pro-Gly-OH	Amino Acid Derivatives	Others
H-Gly-Pro-Gly-OH is a tripeptide containing glycine and proline. H-Gly-Pro-Gly-OH can be used for the synthesis of other polypeptides, such as (Pro Gly Gly)_n .

HY-P4641

H-Trp-Phe-OH	Angiotensin-converting Enzyme (ACE)	Cardiovascular Disease
H-Trp-Phe-OH is a dipeptide consisting of tryptophan and phenylalanine (Trp-Phe). H-Trp-Phe-OH is also an antihypertensive peptide with inhibitory activity on angiotensin-converting enzyme (ACE), dose-dependently increases NO levels, and decreases endothelin-1 (ET-1) levels. H-Trp-Phe-OH (2 mg/kg; subcutaneous injection; 6 injections over 3 days) causes an increase in ovarian weight in female mice .

HY-P4393

H-Leu-Trp-Met-Arg-OH	Aminopeptidase	Others
H-Leu-Trp-Met-Arg-OH is a tetrapeptide. H-Leu-Trp-Met-Arg-OH can be used as a substrate for aminopeptidase-mediated hydrolysis studies .

HY-P4437

H-Met-Phe-OH	Amino Acid Derivatives	Others
H-Met-Phe-OH is a methionine derivative containing methionine and phenylalanine .

HY-N2941

Bisandrographolide C	TRP Channel	Metabolic Disease Inflammation/Immunology
Bisandrographolide C is an unusual dimer of ent-labdane diterpenoid isolated and identified from Andrographis paniculata. Bisandrographolide C activates TRPV1 and TRPV3 channels with K_d values of 289 and 341 μM respectively, and protects cardiomyocytes from hypoxia-reoxygenation injury .

HY-P4420

H-Lys-Trp-OH	Angiotensin-converting Enzyme (ACE)	Cardiovascular Disease
H-Lys-Trp-OH (KW) is an ACE inhibitory peptide with an IC₅₀ of 7.8 μM .

HY-P4292

H-Gly-Pro-Gly-NH2	HIV Amino Acid Derivatives	Infection
H-Gly-Pro-Gly-NH2 is a tripeptide that inhibits HIV-1 replication. H-Gly-Pro-Gly-NH2 inhibits the activity of HIV-1 III_B and HIV-2 ROD with EC₅₀ values of 35 µM and 30 µM, respectively. H-Gly Pro Gly NH2 inhibits HIV-1 replication in vitro by interfering with capsid formation. H-Gly Pro Gly NH2 has antiviral activity and can be used for virus research .

HY-P4487

H-Pro-Pro-Asp-NH2	Biochemical Assay Reagents	Others
H-Pro-Pro-Asp-NH2 is a potent and selective catalyst for asymmetric aldol reactions. H-Pro-Pro-Asp-NH2 catalyzes aldol reactions between acetone and several aldehydes .

HY-P4431

H-Met-Asp-OH	Amino Acid Derivatives	Others
H-Met-Asp-OH is a dipeptide containing methionine and aspartic acid, which can be used for the synthesis of polypeptides .

HY-119306

MCC-134	Potassium Channel	Cardiovascular Disease
MCC-134, a blocker of mitochondrial and opener of surface ATP-sensitive K+ (K_ATP) channels, abrogates cardioprotective effects of chronic hypoxia. MCC-134 is a vasorelaxing agent .

HY-P4488

H-Pro-Pro-Gln-OH	Dipeptidyl Peptidase	Others
H-Pro-Pro-Gln-OH is a oligopeptide with excellent dipeptidyl peptidase-IV (DPP-IV) inhibitory activity .

HY-P4254

H-Gly-Glu-pNA	PAI-1 Ser/Thr Protease	Others
H-Gly-Glu-pNA is a chromogenic peptide substrate that can be widely used in enzymatic analysis, including trypsin and urokinase-type plasminogen activator (uPA) .

HY-169164

Antiproliferative agent-58	Others	Cancer
Antiproliferative agent-58 (compound 8nj) is a potent antiproliferative agent. Antiproliferative agent-58 shows antiproliferative activity in normoxia and hypoxia .

HY-134458A

H-Lys-Tyr-OH TFA Lysyltyrosine TFA	P2X Receptor	Neurological Disease
H-Lys-Tyr-OH TFA (Lysyltyrosine TFA) is a dipeptide composed of lysine and tyrosine. H-Lys-Tyr-OH TFA prevents neurological diseases or improves brain function by promoting the release of noradrenaline and tyrosine into the brain .

HY-P4322

H-Ile-Lys-Val-Ala-Val-OH 1 Publications Verification	ERK Akt	Neurological Disease Cancer
H-Ile-Lys-Val-Ala-Val-OH is one of the most potent active sites of laminin-1. H-Ile-Lys-Val-Ala-Val-OH promotes cell adhesion, neurite outgrowth, and tumor growth. H-Ile-Lys-Val-Ala-Val-OH stimulates BMMSC population growth and proliferation by activating MAPK/ERK1/2 and PI3K/Akt signalling pathways .

HY-W250118

Cephalin form bovine brain	Liposome Autophagy	Neurological Disease Metabolic Disease
Cephalin form bovine brain is an orally active phospholipid widely present in organisms.Cephalin form bovine brain participates in the formation of autophagosome membrane as a lipid anchor of autophagy-related protein Atg8/LC3. Cephalin form bovine brain enhances Autophagic flux, promotes cell differentiation, regulates lipid droplet fusion, delays aging, and also affects lipid metabolism and membrane integrity .

HY-P4651

H-Tyr-Ile-Gly-Ser-Arg-NH2	TGF-β Receptor	Others
H-Tyr-Ile-Gly-Ser-Arg-NH2 is a hexapeptide that is an essential fragment of laminin responsible for efficient cell adhesion and receptor binding. H-Tyr-Ile-Gly-Ser-Arg-NH2 promotes various epithelial cell adhesion activities .

HY-P1350

H-Lys-Trp-Lys-OH	Bacterial	Infection
H-Lys-Trp-Lys-OH is a small molecule peptide which displays antibacterial and antiviral activities extracted from patent CN 104072579 A, Compound AMP12.

HY-157375

Brain Heart Infusion Agar	Biochemical Assay Reagents	Infection Inflammation/Immunology
Brain Heart Infusion Agar is growth medium for the cultivation of a wide variety of microorganisms .

HY-N0712

Typhaneoside 2 Publications Verification	Autophagy	Cardiovascular Disease Inflammation/Immunology
Typhaneoside, extracted from Typha angustifolia L., Typhaneoside can inhibit the excessive autophagy of hypoxia/reoxygenation cells and increase the phosphorylation of Akt and mTOR. Typhaneoside has certain effects on the cardiovascular system, including lowering blood lipid levels, promoting antiatherosclerosis activities, as well as improving immune and coagulation function .

HY-P4232

H-Gly-Arg-Ala-Asp-Ser-Pro-OH	Amino Acid Derivatives	Others
H-Gly-Arg-Ala-Asp-Ser-Pro-OH (GRADSP) is a negative control peptide of GRGDSPK .

HY-N2638

Ilexsaponin A	Apoptosis	Cardiovascular Disease
Ilexsaponin A, isolated from the root of Ilex pubescens, attenuates ischemia-reperfusion-induced myocardial injury through anti-apoptotic pathway. Ilexsaponin A can reduce myocardial infarct size, lower the serum levels of LDH, AST and CK-MB, increase cellular viability and inhibit apoptosis in hypoxia/reoxygenation cardiomyocytes .

HY-106809

BMY-21502 BMS-181168	Drug Derivative	Neurological Disease
BMY-21502 (BMS-181168) is a pyrrolidinone derivative with memory- and cognition-enhancing activities. BMS-181168 attenuates hypoxia-induced deterioration in brain function, as delta/theta decreases, alpha activity increases and the centroid of the combined delta/theta waves is accelerated .

HY-129067

Brain natriuretic peptide BNP (1-32), human	Angiotensin Receptor	Cardiovascular Disease
Brain natriuretic peptide inhibits angiotensin II-induced blood pressure. Brain natriuretic peptide can be used in the control of blood pressure .

HY-157355

Brain Heart Infusion Broth BHI	Biochemical Assay Reagents	Others
Brain Heart Infusion Broth (BHI) is suitable for microbiological culture (For example: Anopheles arabiensis).

HY-E70228

Cathepsin H, human liver	Ser/Thr Protease	Cancer
Cathepsin H, human liver is an aminopeptidase and an endopeptidase. Involved in the catabolism of proteins in the lysosomal system. Cathepsin H, human liver has a key role in the regulation of the biological behavior of tumor cells and the pathological processes of brain diseases .

HY-P4556

H-Phe-Gly-His-p-nitro-Phe-Phe-Ala-Phe-OMe	Biochemical Assay Reagents	Others
H-Phe-Gly-His-p-nitro-Phe-Phe-Ala-Phe-OMe is a polypeptide that can be hydrolyzed by Rennin (HY-P2810). H-Phe-Gly-His-p-nitro-Phe-Phe-Ala-Phe-OMe is commonly used as a biochemical reaction reagent .

HY-161838

ICT10336	ATM/ATR	Cancer
ICT10336 is a hypoxia-responsive prodrug of ATR inhibitor, AZD6738 (HY-19323). ICT10336 is hypoxia-activated and specifically releases AZD6738 only in hypoxic conditions in vitro. This can inhibit ATR activation (T1989 and S428 phosphorylation) and subsequently abrogate HIF1a-mediated adaptation of hypoxic cancers cells, thus selectively inducing cell death in 2D and 3D cancer models. ICT10336 is a metabolic substrate of CYPOR activity.

HY-103227

Desidustat 2 Publications Verification ZYAN1	HIF/HIF Prolyl-Hydroxylase	Cardiovascular Disease
Desidustat is an orally active HIF hydroxylase inhibitor. Desidustat can be used for the research of various disorders including anemia of different types and conditions associated with ischemia/hypoxia .

HY-136748

HIF-2α-IN-4 1 Publications Verification	HIF/HIF Prolyl-Hydroxylase	Cancer
HIF-2α-IN-4 is a potent inhibitor of hypoxia inducible factor-2α (HIF-2α) translation, with an IC₅₀ of 5 μM. HIF-2α-IN-4 decreases both constitutive and hypoxia-induced HIF-2α protein expression. HIF-2α-IN-4 links its 5'UTR iron-responsive element to oxygen sensing .

HY-P1573

Brain Natriuretic Peptide-45, rat BNP-45, rat	Natriuretic Peptide Receptor (NPR)	Cardiovascular Disease
Brain Natriuretic Peptide-45, rat (BNP-45, rat) is a circulating form of rat brain natriuretic peptide isolated from rat heart with potent hypotensive and natriuretic potency .

HY-172371

Hypoxystat	Reactive Oxygen Species (ROS)	Others
Hypoxystat increases the affinity of hemoglobin for oxygen and reduces the release of oxygen to tissues, thereby inducing the tissue hypoxia. Hypoxystat alleviates the mitochondrial disease Leigh syndrome in Ndufs4 knockout mouse models. Hypoxystat exhibits orally activity .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-N2506

Ginsenoside Ra1	Cardiovascular Disease Panax ginseng C. A. Meyer Triterpenes Structural Classification Classification of Application Fields Terpenoids Source classification Plants Disease Research Fields Araliaceae	Others
Ginsenoside Ra1 is a component from ginseng, inhibits protein tyrosine kinase (PTK) activation induced by hypoxia/reoxygenation .

HY-N0272

Eleutheroside E 2 Publications Verification	Structural Classification Classification of Application Fields Source classification Lignans Phenylpropanoids Acanthopanax senticosus (Rupr. et Maxim.) Harms Plants Inflammation/Immunology Disease Research Fields Araliaceae	Apoptosis NF-κB
Eleutheroside E is an important component of ginseng that can be taken orally. Eleutheroside E has anti-inflammatory and antioxidant properties, and it helps reduce apoptosis in heart cells caused by hypoxia-reoxygenation (H/R) damage. Eleutheroside E can improve type 2 diabetes, enhance cognitive function, and has neuroprotective effects .

HY-N0712

Typhaneoside 2 Publications Verification	Cardiovascular Disease Flavonols Structural Classification Flavonoids Typhaceae Classification of Application Fields Typha angustifolia L. Source classification Phenols Polyphenols Plants Disease Research Fields	Autophagy
Typhaneoside, extracted from Typha angustifolia L., Typhaneoside can inhibit the excessive autophagy of hypoxia/reoxygenation cells and increase the phosphorylation of Akt and mTOR. Typhaneoside has certain effects on the cardiovascular system, including lowering blood lipid levels, promoting antiatherosclerosis activities, as well as improving immune and coagulation function .

HY-N2638

Ilexsaponin A	Cardiovascular Disease Aquifoliaceae Triterpenes Classification of Application Fields Terpenoids Source classification Ilex pubescens Hook. et Arn. Plants Disease Research Fields	Apoptosis
Ilexsaponin A, isolated from the root of Ilex pubescens, attenuates ischemia-reperfusion-induced myocardial injury through anti-apoptotic pathway. Ilexsaponin A can reduce myocardial infarct size, lower the serum levels of LDH, AST and CK-MB, increase cellular viability and inhibit apoptosis in hypoxia/reoxygenation cardiomyocytes .

HY-127022

Anisodine Daturamine; α-Hydroxyscopolamine	Structural Classification Alkaloids Other Alkaloids Anisodus tanguticus (Maxinowicz) Pascher Source classification Solanaceae Plants	mAChR Calcium Channel Reactive Oxygen Species (ROS)
Anisodine (Daturamine) is a neuroprotective compound that reduces exacerbated M1, M2, M4, and M5 receptor expression in brain tissues under hypoxia/reoxygenation conditions. Anisodine inhibits calcium ion influx and *reactive oxygen* species (ROS)*levels. Anisodine leads to decreased aspartate levels during hypoxia* .

HY-134571

Brain Extract Total	Structural Classification Lipid	Biochemical Assay Reagents
Brain Extract Total is a natural brain total lipid extract that can be used to prepare neuronal membranes. Brain Extract Total can be used for the study of Alzheimer's disease .

HY-N0712R

Typhaneoside (Standard)	Flavonols Structural Classification Flavonoids Typhaceae Typha angustifolia L. Source classification Phenols Polyphenols Plants	Reference Standards Autophagy
Typhaneoside (Standard) is the analytical standard of Typhaneoside. This product is intended for research and analytical applications. Typhaneoside, extracted from Typha angustifolia L., Typhaneoside can inhibit the excessive autophagy of hypoxia/reoxygenation cells and increase the phosphorylation of Akt and mTOR. Typhaneoside has certain effects on the cardiovascular system, including lowering blood lipid levels, promoting antiatherosclerosis activities, as well as improving immune and coagulation function .

HY-N2638R

Ilexsaponin A (Standard)	Aquifoliaceae Triterpenes Structural Classification Terpenoids Source classification Ilex pubescens Hook. et Arn. Plants	Reference Standards Apoptosis
Ilexsaponin A (Standard) is the analytical standard of Ilexsaponin A. This product is intended for research and analytical applications. Ilexsaponin A, isolated from the root of Ilex pubescens, attenuates ischemia-reperfusion-induced myocardial injury through anti-apoptotic pathway. Ilexsaponin A can reduce myocardial infarct size, lower the serum levels of LDH, AST and CK-MB, increase cellular viability and inhibit apoptosis in hypoxia/reoxygenation cardiomyocytes .

HY-N12908

Roridin H Verrucarin H	Structural Classification Microorganisms Macrolide Antibiotics Antibiotics Source classification	Antibiotic
Roridin H (Verrucarin H) is an antibiotic and can be isolated from Myrothecium verrucaria .

HY-N10643

Lushanrubescensin H Rabdoternin H	Labiatae Plants Cyrtocymura cincta var. cincta	Others
Lushanrubescensin H (Rabdoternin H) is an ent-Kaurane diterpenoid from Isodon ternifolius aboveground part .

HY-W037619

Pteridine-2,4(1H,3H)-dione	Natural Products Classification of Application Fields Source classification Metabolic Disease Endogenous metabolite Disease Research Fields	Endogenous Metabolite
Pteridine-2,4(1H,3H)-dione is an endogenous metabolite.

HY-N7582

Cimicifugoside H-2	Structural Classification Terpenoids Source classification Ranunculaceae Diterpenoids Plants Cimicifuga foetida Linn.	Others
Cimicifugoside H-2 is a cyclolanostanol xyloside. Cimicifugoside H-2 can be isolated from Cimicifuga Rhizome .

HY-129325

Cytochalasin H	Structural Classification Antibiotics Gramineae Source classification Plants Paspalum scrobiculatum L.	Antibiotic Bacterial Apoptosis Bcl-2 Family Caspase
Cytochalasin H is a nature product that could be isolated from fungus Phomopsis sp. Cytochalasin H inhibits cell growth and induces apoptosis. Cytochalasin H has anti-angiogenic activity. Cytochalasin H is an antibiotic and has antibacterial activity .

HY-16940

24(S)-Hydroxycholesterol 24S-OHC; 24S-HC; Cerebrosterol	Structural Classification Classification of Application Fields Source classification Disease markers Metabolic Disease Nervous System Disorder Endogenous metabolite Disease Research Fields Steroids	LXR iGluR Endogenous Metabolite
24(S)-Hydroxycholesterol (24S-OHC), the major brain cholesterol metabolite, plays an important role to maintain homeostasis of cholesterol in the brain. 24(S)-Hydroxycholesterol (24S-OHC) is one of the most efficient endogenous LXR agonist known and is present in the brain and in the circulation at relatively high levels. 24(S)-Hydroxycholesterol (24S-OHC) is a very potent, direct, and selective positive allosteric modulator of NMDARs with a mechanism that does not overlapthat of other allosteric modulators .

HY-N2607

Sanggenone H Sanggenon H	Flavonoids Classification of Application Fields Flavonones Source classification Other Diseases Phenols Polyphenols Plants Moraceae Disease Research Fields Morus alba Linn.	Others
Sanggenone H is found in Morus alba L .

HY-137566

Cucumarioside H	Triterpenes Structural Classification Animals Terpenoids Source classification	Mitochondrial Metabolism
Cucumarioside H is a novel triterpene glycoside isolated from the Far Eastern sea cucumber Eupentacta fraudatrix, including H2, H3 and H4. These glycosides have a branched pentasyl structure with a rare 3-O-methyl-D-xylose as the terminal monosaccharide. H2 contains 23,24,25,26,27-pentanolone sterols and has an 18(16)-lactone, which is not common in sea cucumbers. The glycoside portion of H3 contains an extremely rare ethoxyl radical at the 25 position, which may be an artifact formed during the long ethanol extraction process. Studies have shown that H1-3 are cytotoxic to mouse spleen lymphocytes, hemolytic to mouse erythrocytes, and cytotoxic to Ehrlich carcinoma cells. The presence of a 25-hydroxyl group in the glycoside portion significantly reduces these activities.

HY-N12877

Ophiobolin H	Structural Classification Natural Products Microorganisms Source classification	Bacterial
Ophiobolin H is a fungal metabolite that can be isolated from Aspergillus ustus. Ophiobolin H inhibits growth of Bacillus subtilis cultures. Ophiobolin H induces hyperacusia in day-old chicks at rates up to 375 mg/kg .

HY-N10397

Maceneolignan H	Structural Classification Natural Products Classification of Application Fields Source classification Myristicaceae Plants Myristica fragrans Houtt. Inflammation/Immunology Disease Research Fields	CCR
Maceneolignan H (Compound 8) is a neolignane compound isolated from the arils of Myristica fragrans. Maceneolignan H is a selective CCR3 antagonist (EC₅₀ = 1.4 μM). Maceneolignan H has the potential for the research of allergic diseases .

HY-N8141

Regaloside H	Monophenols other families Classification of Application Fields Simple Phenylpropanols Source classification Phenols Metabolic Disease Phenylpropanoids Plants Disease Research Fields	Others
Regaloside H, a phenylpropanoid glycerol glucoside, is a gluconeogenesis inhibitor. Regaloside H can reduce glucose production in Hepatocytes .

HY-N9321

Cathayanon H	Flavanonols Flavonoids Classification of Application Fields Source classification Phenols Polyphenols Plants Moraceae Morus cathayana Hemsl. Disease Research Fields Cancer	Others
Cathayanon H is isolated from the paper mulberry tree. Cathayanon H is cytotoxic against human ovariancarcinoma cells .

HY-123647

Satratoxin H	Structural Classification Natural Products Microorganisms Source classification	Apoptosis p38 MAPK
Satratoxin H is a trichothecene with cytotoxic activity. Satratoxin H can be used for cytotoxicological studies on lymphoid cell lines .

HY-N13317

Otophylloside H	Structural Classification Polysaccharides Source classification Asclepiadaceae Cynanchum otophyllum Schneid． Plants Saccharides	Others
Otophylloside H is a pregnane glycosides isolated from the roots of Cynanchum otophyllum. Otophylloside H can be used in epilepsy research .

HY-N10955

Dichotomine H	Structural Classification Alkaloids Pyrrole Alkaloids Source classification Psammosilene tunicoides W. C. Wu et C. Y. Wu Pyridine Alkaloids Plants Caryophyllaceae	Others
Dichotomine H is a P-carboline alkaloid that can be extracted from Stellaria dichotoma L. Dichotomine H has good antiallergic activity .

HY-N16144

Osmanthuside H	Structural Classification Monophenols Ipomoea nil (Linnaeus) Roth Source classification Phenols Plants Convolvulaceae	Aldehyde Dehydrogenase (ALDH)
Osmanthuside H (Compound 1), a phenylethanoid glycoside (PhG), is a alcohol dehydrogenase (ADH) inhibitor with an IC₅₀ of 175.4 μg/mL. Osmanthuside H can be isolated from the leaves of persimmon Diospyros kaki. Osmanthuside H has anti-inflammatory and neuroprotective activities .

HY-N13928

Arisugacin H	Structural Classification Natural Products Microorganisms Source classification	Cholinesterase (ChE)
Arisugacin H, a microbial metabolite, is a structural analog of Arisugacin A (HY-N13901). Arisugacin H shows no activity against AChE .

HY-N8270

Physalin H	Structural Classification Cardiacglycosides Source classification Solanum nigrum Linn. Plants Solanaceae Steroids	Hedgehog Endogenous Metabolite
Physalin H is a natural product that can be isolated from Solanum nigrum. Physalin H is an inhibitor of Hedgehog (Hh) signaling and it disrupts GLI1-DNA-complex formation. Physalin H inhibits GLI1 transcription with an IC₅₀ value of 0.7 μM. Physalin H shows cytotoxicity to PANC1 and DU145 cells with IC₅₀ values of 5.7 and 6.8 μM, respectively .

HY-N2600R

Kuwanon H (Standard)	Structural Classification Flavonoids Flavones Source classification Phenols Polyphenols Plants Moraceae Morus alba Linn.	Reference Standards Bombesin Receptor
Kuwanon H (Standard) is the analytical standard of Kuwanon H. This product is intended for research and analytical applications. Kuwanon H is a flavonoid isolated from Morus alba, which acts as a potent non-peptide bombesin receptor antagonist. Kuwanon H selectively inhibits binding of gastrin releasing peptide CRP to GRP-preferring recepotr, with a Ki value of 290 nM in cells .

HY-N11943

Kadsulignan H	Structural Classification Source classification Lignans Phenylpropanoids Plants Kadsura coccinea (Lem.) A. C. Smith Schisandraceae	NO Synthase
Kadsulignan H (compound 13) is a lignan with inhibitory activity on NO production. Kadsulignan H inhibits NO production in BV-2 cells with an IC₅₀ of 14.1 μM .

HY-N7051

Tubulysin H	Structural Classification Microorganisms Classification of Application Fields Ketones, Aldehydes, Acids Source classification Disease Research Fields Cancer	ADC Payload Microtubule/Tubulin
Tubulysin H is a highly cytotoxic anti-microtubule toxin (anti-microtubule toxins) that is synthesized as an ADC cytotoxin (ADC Cytotoxin). Tubulysin H can be isolated from the myxobacteria Archangium geophyra and Angiococcus disciformis. Tubulysin H displays extremely potent cytotoxic activity in mammalian cells, including multidrug-resistant cell lines, with IC₅₀ values in the low nanomolar range. Tubulysin H inhibits microtubule/tubulin polymerization and leads to cell cycle arrest and apoptosis .

HY-N14082

Monamycin H1	Structural Classification Microorganisms Macrolide Antibiotics Antibiotics Source classification	Antibiotic Bacterial
Monamycin H1 is an ester peptide antibiotic. Monamycin H1 has activity against Gram-positive bacteria .

HY-N14083

Monamycin H2	Structural Classification Microorganisms Macrolide Antibiotics Antibiotics Source classification	Antibiotic Bacterial
Monamycin H2 is an ester peptide antibiotic. Monamycin H2 has activity against Gram-positive bacteria .

HY-N11656

Poricoic acid H	Structural Classification Microorganisms Ketones, Aldehydes, Acids Source classification	Others
Poricoic acid H is a triterpene .

HY-135211

Rubomycin H	Structural Classification Microorganisms Antibiotics Source classification	Others
Rubomycin H is an active compound.

HY-N11434

Anisocoumarin H	Structural Classification Adenocarpus cincinnatus (Ball) Maire Source classification Coumarins Phenylpropanoids Plants Compositae	Fungal
Anisocoumarin H is a coumarin that exhibits antifungal activity. Anisocoumarin H shows the activities against Microsporum gypseum, Trichophyton rubrum and Trichophyton mentagrophytes with MICs of 62.5 µg/mL .

HY-76228R

1H-pyrazole (Standard)	Alkaloids Structural Classification Other Alkaloids Source classification Endogenous metabolite	Drug Intermediate Biochemical Assay Reagents
1H-pyrazole (Standard) is the analytical standard of 1H-pyrazole. This product is intended for research and analytical applications. 1H-pyrazole is a nitrogen-containing heterocyclic compound composed of a five-membered ring and two nitrogen atoms. 1H-pyrazole is an intermediate in organic synthesis. 1H-pyrazole coordinates with metal ions. 1H-pyrazole derivatives have antibacterial, anti-inflammatory, anti-malarial, and anti-leishmanial activities .

HY-N7296

Derrisisoflavone H	Structural Classification Flavonoids Leguminosae Source classification Derris trifoliata Lour. Plants Other Flavonoids	Others
Derrisisoflavone H is a natural product .

HY-N13544

Lespedezaflavanone H	Structural Classification Flavonoids Leguminosae Flavonones Source classification Sophora tonkinensis Gagnep. Plants	Others
Lespedezaflavanone H is a natural product .

HY-N13685

Buxifoliadine H	Structural Classification Alkaloids Piperidine Alkaloids Source classification Atalantia buxifolia (Poir.) Oliv. Rutaceae Plants	Others
Buxifoliadine H is a natural product .

HY-N13661

Shanciol H	Structural Classification Orchidaceae Source classification Pleione yunnanensis (Rolfe) Rolfe Phenols Polyphenols Plants	Others
Shanciol H is a natural product .

HY-N13451

Cannabisin H	Structural Classification Monophenols Cannabis sativa L Source classification Phenols Plants Moraceae	Others
Cannabisin H is a natural product .

HY-N14499

Saframycin H	Structural Classification Natural Products Microorganisms Source classification	Bacterial
Saframycin H has the effect of anti-Gram-positive bacteria. Saframycin H has the effect of inhibiting mouse lymphocyte L-1210 with an ID₅₀ of 0.033 μM .

HY-137323

Leucinostatin H	Structural Classification Microorganisms Antibiotics Source classification Other Antibiotics	Antibiotic Bacterial
Leucinostatin H is a polypeptide antibiotic discovered in Paecilomyces marquandii, characterized by a tertiary amine-oxide terminal group. Leucinostatin H exhibits inhibitory activity against Gram-positive bacteria, such as Bacillus subtilis, B. cereus, and Staphylococcus aureus (MIC 10-100 μg/mL). Leucinostatin H holds potential for research in anti-infective and plant disease control applications .

HY-130347

H2S Donor 5a	Structural Classification Natural Products Classification of Application Fields Source classification Other Diseases Endogenous metabolite Disease Research Fields	Endogenous Metabolite
H2S Donor 5a is a cysteine-activated H2S donor. H₂S plays important roles in biological systems. H2S Donor 5a is a useful tool in H₂S research .

HY-101412

2-(Methylamino)-1H-purin-6(7H)-one 1 Publications Verification N2-methylguanine	Structural Classification Natural Products Classification of Application Fields Source classification Other Diseases Endogenous metabolite Disease Research Fields	Bacterial DNA/RNA Synthesis Endogenous Metabolite
2-(Methylamino)-1H-purin-6(7H)-one (N2-Methylguanine) is a modified nucleoside. 2-(Methylamino)-1H-purin-6(7H)-one is an endogenous methylated nucleoside found in human fluids.

HY-N14394

Fusicoccin H	Structural Classification Natural Products Microorganisms Source classification	Others
Fusicoccin H is a metabolite of Fusicoccum amygdali .

HY-121430

Lamellarin H	Structural Classification Alkaloids Animals Other Alkaloids Source classification	Drug Derivative
Lamellarin H is a benzo-isoquinoline-coumarin .

HY-N1682

2,7-Dihydroxy-2H-1,4-benzoxazin-3(4H)-one	Structural Classification Alkaloids Other Alkaloids Source classification Scrophulariaceae Scoparia dulcis L Plants	Others
2,7-Dihydroxy-2H-1,4-benzoxazin-3(4H)-one is a Alkaloids product that can be isolated from the roots of Scoparia dulcis .

HY-N3237

Mulberrofuran H	Source classification Phenols Polyphenols Plants Moraceae Morus alba Linn.	Dopamine Receptor
Mulberrofuran H is a 2-arylbenzofuran derivative from the cultivated mulberry tree (Morus lhou (ser.) Koidz.). Mulberrofuran H demonstrates potent inhibition against substrates L-tyrosine (IC₅₀=4.45 µM) and L-DOPA (IC₅₀=19.70 µM). Mulberrofuran H also shows potent anti-inflammatory and antioxidative activities .

HY-123075

Odoroside H	Digitalis purpurea Linn. Structural Classification Cardiacglycosides Source classification Scrophulariaceae Plants Steroids	Others
Odoroside H is a natural cardenolide with anticancer activities .

HY-W782096

Salvianolic acid H	Structural Classification Labiatae Source classification Samanea saman (Jacq.) Merr. Phenols Polyphenols Plants	Cholinesterase (ChE)
Salvianolic acid H is a potent acetylcholinesterase (AChE) inhibitor .

Cat. No.	Product Name	Chemical Structure

HY-W008385S

H-HoArg-OH-d4
H-HoArg-OH-d₄ is a deuterium labeled H-HoArg-OH (HY-W008385). H-HoArg-OH, a homologue arginine, is a strong inhibitor of human bone and liver alkaline phosphatase.

HY-W010589S2

H-Abu-OH-d6
H-Abu-OH-d₆ is the deuterium labeled H-Abu-OH. H-Abu-OH, one of the three isomers of aminobutyric acid, is elevated in the plasma of children with with Reye's syndrome, tyrosinemia, homocystinuria, nonketotic hyperglycinemia, and ornithine transcarbamylase deficiency.

HY-B0113S5

Omeprazole-d6

Omeprazole-d₆ (H 16868-d₆) is deuterium labeled Omeprazole. Omeprazole (H 16868), a proton pump inhibitor (PPI), is available for treatment of acid-related gastrointestinal disorders. Omeprazole shows competitive inhibition of CYP2C19 activity with a K_i of 2 to 6 μM . Omeprazole also inhibits growth of Gram-positive and Gram-negative bacteria .Omeprazole is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor) .

HY-W738325

H-Phe-OMe.hydrochloride-d5
H-Phe-OMe.hydrochloride-d₅ is the deuterium labeled H-Phe-OMe.hydrochloride (HY-Y1394). H-Phe-OMe.hydrochloride is a phenylalanine derivative .

HY-154741S

6-β-D-Ribofuranosyl-2,4(1H,3H)-pyrimidinedione-15N2
6-β-D-Ribofuranosyl-2,4(1H,3H)-pyrimidinedione- ¹⁵N₂ is ¹⁵N labeled (HY-154741).

HY-132732S

2H-2-Ethyl-d5 candesartan
2H-2-Ethyl-d₅ Candesartan is the deuterium labeled 2H-2-Ethyl Candesartan .

HY-132733S

1H-1-Ethyl-d5 candesartan
1H-1-Ethyl-d₅ Candesartan is the deuterium labeled 1H-1-Ethyl Candesartan .

HY-150678S

Adenosine:H20-13c
Adenosine:H20- ¹³C is the ¹³C labeled Adenosine:H20 .

HY-W010589S

H-Abu-OH-d3
H-Abu-OH-d₃ is the deuterium labeled H-Abu-OH. H-Abu-OH, one of the three isomers of aminobutyric acid, is elevated in the plasma of children with with Reye's syndrome, tyrosinemia, homocystinuria, nonketotic hyperglycinemia, and ornithine transcarbamylase deficiency.

HY-W010589S1

H-Abu-OH-d2
H-Abu-OH-d₂ is the deuterium labeled H-Abu-OH. H-Abu-OH, one of the three isomers of aminobutyric acid, is elevated in the plasma of children with with Reye's syndrome, tyrosinemia, homocystinuria, nonketotic hyperglycinemia, and ornithine transcarbamylase deficiency.

HY-135180S

1H-1-Ethyl Candesartan Cilexetil-d5
1H-1-Ethyl Candesartan Cilexetil-d₅ is the deuterium labeled 1H-1-Ethyl Candesartan Cilexetil .

HY-W007750S

H-Lys(Z)-OH-d3
H-Lys(Z)-OH-d₃ is the deuterium labeled H-Lys(Z)-OH.

HY-W010590S1

H-DL-Abu-OH-d6
H-DL-Abu-OH-d₆ is the deuterium labeled H-DL-Abu-OH .

HY-143907S

Atorvastatin EP impurity H-d5
Atorvastatin EP impurity H-d₅ is the deuterium labeled Atorvastatin EP impurity H .

HY-W095672AS4

((2S,7aR)-2-Fluorotetrahydro-1H-pyrrolizin-7a(5H)-yl)methanol-d2
((2S,7aR)-2-Fluorotetrahydro-1H-pyrrolizin-7a(5H)-yl)methanol-d₂ ((2S,7aR)-2-Fluorotetrahydro-1H-pyrrolizine-7a(5H)-methanol-d₂) is the deuterium labeled ((2S,7aR)-2-Fluorotetrahydro-1H-pyrrolizin-7a(5H)-yl)methanol.

HY-W703411

Dibenzo[a,h]acridine-d6
Dibenzo[a,h]acridine-d₆ is the deuterium labeled Dibenz[a,h]acridine (HY-W762000).

HY-B0113S4

Omeprazole-d3 sodium

Omeprazole-d₃ sodium is deuterated labeled Omeprazole (HY-B0113). Omeprazole (H 16868), a proton pump inhibitor (PPI), is available for treatment of acid-related gastrointestinal disorders. Omeprazole shows competitive inhibition of CYP2C19 activity with a K_i of 2 to 6 μM . Omeprazole also inhibits growth of Gram-positive and Gram-negative bacteria .Omeprazole is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor) .

HY-W018710S

2(3H)-Benzothiazolone-d4
2(3H)-Benzothiazolone-d₄ is the deuterium labeled 2(3H)-Benzothiazolone .

HY-B0113S1

Omeprazole-d3-1

Omeprazole-d₃-1 is the deuterium labeled Omeprazole. Omeprazole (H 16868), a proton pump inhibitor (PPI), is available for treatment of acid-related gastrointestinal disorders. Omeprazole shows competitive inhibition of CYP2C19 activity with a K_i of 2 to 6 μM . Omeprazole also inhibits growth of Gram-positive and Gram-negative bacteria .Omeprazole is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor) .

HY-W701580

6-Amino-3-methylpyrimidine-2,4(1H,3H)-dione-d3
6-Amino-3-methylpyrimidine-2,4(1H,3H)-dione-d₃ (6-Amino-3-methyluracil-d₃) is the deuterium labeled 6-Amino-3-methylpyrimidine-2,4(1H,3H)-dione (HY-W038777).

HY-W007497S

H-β-Ala-NH2.-d4HCl
H-β-Ala-NH2.-d₄ HCl is the deuterium labeled H-β-Ala-NH2.HCl .

HY-W779244

1H-Pyrazole-3,4,5-d3
1H-Pyrazole-3,4,5-d₃ is the deuterium labeled 1H-pyrazole (HY-76228). 1H-pyrazole is a nitrogen-containing heterocyclic compound composed of a five-membered ring and two nitrogen atoms. 1H-pyrazole is an intermediate in organic synthesis. 1H-pyrazole coordinates with metal ions. 1H-pyrazole derivatives have antibacterial, anti-inflammatory, anti-malarial, and anti-leishmanial activities .

HY-148233S

JNJ-6204
JNJ-6204 is a dual inhibitor for CSNK1D (Casein Kinase 1 Delta) and CSNK1E (Casein Kinase 1 Epsilon) (CSNK1D IC₅₀=2.3 nM; CSNK1E IC₅₀=137 nM). JNJ-6204 shows good brain exposure .

HY-W029450S

Tetrahydropyrimidine-2(1H)-thione-d6
Tetrahydropyrimidine-2(1H)-thione-d₆ is the deuterium labeled Tetrahydropyrimidine-2(1H)-thione .

HY-W014340S

2-Nitro-9H-fluorene-d9
2-Nitro-9H-fluorene-d₉ is the deuterium labeled 2-Nitro-9H-fluorene .

HY-W008452S

H-Tyr(3-I)-OH-13C6
H-Tyr(3-I)-OH- ¹³C₆ is the ¹³C-labeled H-Tyr(3-I)-OH. H-Tyr(3-I)-OH is a potent and effective tyrosine hydroxylase inhibitor. H-Tyr(3-I)-OH is an intermediate in the production of thyroid hormones and has a role as a human or mouse metabolite .

HY-105129AS

Pimonidazole-d10

Pimonidazole-d₁₀ is the deuterium labeled Pimonidazole. Pimonidazole is a novel hypoxia marker for complementary study of tumor hypoxia and cell proliferation in tumor . Pimonidazole accumulates in hypoxic cells via covalent binding with macromolecules or by forming reductive metabolites after reduction of its nitro group, it can be used for qualitative and quantitative assessment of tumor hypoxia .

HY-W101495S3

Boc-Leu-OH·H2O-d7
Boc-Leu-OH·H2O-d₇ is the deuterium labeled Boc-Leu-OH·H2O.

HY-W012997S

Tetrahydro-2H-pyran-2-one-d4
Tetrahydro-2H-pyran-2-one-d₄ is the deuterium labeled Tetrahydro-2H-pyran-2-one. Tetrahydro-2H-pyran-2-one is an endogenous metabolite with antioxidant capacity. Tetrahydro-2H-pyran-2-one is the small active molecule and can be used as drug intermediate .

HY-W101495S2

Boc-Leu-OH·H2O-d10
Boc-Leu-OH·H2O-d₁₀ is the deuterium labeled Boc-Leu-OH·H2O .

HY-W101495S1

Boc-Leu-OH·H2O-d3
Boc-Leu-OH·H2O-d₃ is the deuterium labeled Boc-Leu-OH·H2O .

HY-W779904

H-Gly-OBzl.TosOH-13C2,15N
H-Gly-OBzl.TosOH- ¹³C₂, ¹⁵N is the ¹³C- and ¹⁵N-labeled H-Gly-OBzl.TosOH (HY-W011200). H-Gly-OBzl.TosOH is a Glycine (HY-Y0966) derivative .

HY-W015224S

Methyl 2-(1H-indol-3-yl)acetate-d5
Methyl 2-(1H-indol-3-yl)acetate-d₅ is the deuterium labeled Methyl 2-(1H-indol-3-yl)acetate. Methyl 2-(1H-indol-3-yl)acetate is an endogenous metabolite.

HY-B0113S3

Omeprazole-13C,d3

Omeprazole- ¹³C,d₃ is a ¹³C-labeled and deuterium labeled Omeprazole. Omeprazole (H 16868), a proton pump inhibitor (PPI), is available for treatment of acid-related gastrointestinal disorders. Omeprazole shows competitive inhibition of CYP2C19 activity with a K_i of 2 to 6 μM . Omeprazole also inhibits growth of Gram-positive and Gram-negative bacteria .Omeprazole is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor) .

HY-69188S

3,4-Dihydro-2H-benzo[b][1,4]thiazine-d2
3,4-Dihydro-2H-benzo[b][1,4]thiazine-d₂ (3,4-Dihydro-2H-1,4-benzothiazine-d₂) is the deuterium labeled 3,4-Dihydro-2H-benzo[b][1,4]thiazine.

HY-W004264S

Tetrahydro-2H-pyran-4-ol-d5
Tetrahydro-2H-pyran-4-ol-d₅ is the deuterium labeled Tetrahydro-2H-pyran-4-ol .

HY-W705408

1H-Imidazole-5-carboxaldehyde-15N2
1H-Imidazole-5-carboxaldehyde- ¹⁵N₂ is the ¹⁵N-labeled 1H-Imidazole-5-carboxaldehyde (HY-59303). 1H-Imidazole-5-carboxaldehyde is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-W005435S

2,3,4,5-Tetrahydro-1H-benzo[b]azepine-d2
2,3,4,5-Tetrahydro-1H-benzo[b]azepine-d₂ (2,3,4,5-Tetrahydro-1H-1-benzazepine-d₂) is the deuterium labeled 2,3,4,5-Tetrahydro-1H-benzo[b]azepine.

HY-W002116S

Methyl syringate-d6

Methyl syringate-d₆ is the deuterium labeled Methyl syringate. Methyl syringate is a selective TRPA1 agonist. Methyl syringate regulates food intake and gastric emptying through a TRPA1-mediated pathway. Methyl syringate is an efficient phenolic mediator for bacterial and fungal laccases. Methyl syringate is a chemical marker of Asphodel monofloral honey. Methyl syringate contributes to the antibacterial activity of honey. Methyl syringate inhibits aflatoxin production. Methyl syringate can contribute to weight suppression. Methyl syringate can be studies for cancer prevention (e.g. lung cancer), suppression of hypoxia-induced inflammatory response and tumorigenesis .

HY-W014389S

9,9-Dimethyl-9H-xanthene-d2
9,9-Dimethyl-9H-xanthene-d2 is the deuterium labeled 9,9-Dimethyl-9H-xanthene (HY-W014389) .

HY-23805S

3,6-Dichloro-9H-carbazole-13C12
3,6-Dichloro-9H-carbazole- ¹³C₁₂ is ¹³C labeled 3,6-Dichloro-9H-carbazole .

HY-W751834

6-Amino-5-nitropyrimidine-2,4(1H,3H)-dione-13C3
6-Amino-5-nitropyrimidine-2,4(1H,3H)-dione- ¹³C₃ (NSC 99321- ¹³C₃) is the ¹³C-labeled 6-Amino-5-nitropyrimidine-2,4(1H,3H)-dione (HY-W016913).

HY-44302S

4'-Ethyl-4'-hydroxy-7',8'-dihydrospiro[[1,3]dioxolane-2,6'-pyrano[3,4-f]indolizine]-3',10'(1'H,4'H)-dione-d5
4'-Ethyl-4'-hydroxy-7',8'-dihydrospiro[[1,3]dioxolane-2,6'-pyrano[3,4-f]indolizine]-3',10'(1'H,4'H)-dione-d₅ is the deuterium labeled 4'-Ethyl-4'-hydroxy-7',8'-dihydrospiro[[1,3]dioxolane-2,6'-pyrano[3,4-f]indolizine]-3',10'(1'H,4'H)-dione .

HY-W010269S

5-Methoxy-1H-benzo[d]imidazole-d3
5-Methoxy-1H-benzo[d]imidazole-d₃ is the deuterium labeled 5-Methoxy-1H-benzo[d]imidazole .

HY-44745S

4-Ethyl-1,4,7,8-tetrahydro-3H,10H-spiro[pyrano[3,4-f]indolizine-6,2'-[1,3]dioxolane]-3,10-dione-d5
4-Ethyl-1,4,7,8-tetrahydro-3H,10H-spiro[pyrano[3,4-f]indolizine-6,2'-[1,3]dioxolane]-3,10-dione-d5 is the deuterium labeled 4-Ethyl-1,4,7,8-tetrahydro-3H,10H-spiro[pyrano[3,4-f]indolizine-6,2'-[1,3]dioxolane]-3,10-dione .

HY-Y0688S

1H-Benzotriazole-4,5,6,7-d4
1H-Benzotriazole-4,5,6,7-d₄ is the deuterium labeled 1H-Benzo[d][1,2,3]triazole .

HY-B0303AS1

Diphenhydramine-d5 hydrochloride
Diphenhydramine-d₅ (hydrochloride) is the deuterium labeled Diphenhydramine hydrochloride. Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB) .

HY-B0303AS

Diphenhydramine-d6 hydrochloride
Diphenhydramine-d₆ (hydrochloride) is the deuterium labeled Diphenhydramine hydrochloride. Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB) .

HY-W015597S

rel-3a,4,7,7a-Tetrahydro-1H-isoindole-1,3(2H)-dione-d6
rel-3a,4,7,7a-Tetrahydro-1H-isoindole-1,3(2H)-dione-d₆ is the deuterium labeled rel-3a,4,7,7a-Tetrahydro-1H-isoindole-1,3(2H)-dione .

HY-W090625S

5H-Benzofuro[3,2-c]carbazole-d10
5H-Benzofuro[3,2-c]carbazole-d₁₀ is the deuterium labeled 5H-Benzofuro[3,2-c]carbazole (HY-W090625) .

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