2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. SB 242084 dihydrochloride (Standard)

SB 242084 (dihydrochloride) (Standard) is the analytical standard of SB 242084 (dihydrochloride). This product is intended for research and analytical applications. SB 242084 dihydrochloride is a selective, competitive and high-affinity (pKi=9.0) 5-HT2C receptor antagonist (crosses the blood-brain barrier). SB 242084 dihydrochloride increases basal activity of dopaminergic neurons in the ventral tegmental area (VTA) of the midbrain and dopamine release in the vomeronasal nucleus. SB 242084 dihydrochloride also increases mitochondrial gene expression and oxidative metabolism via 5-HT2A receptor. SB 242084 dihydrochloride has good research potential in the negative symptoms of anxiety, depression and schizophrenia, as well as in acute organ damage.

For research use only. We do not sell to patients.

SB 242084 dihydrochloride (Standard)

SB 242084 dihydrochloride (Standard) Chemical Structure

CAS No. : 1049747-87-6

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SMILES

O=C(N1CCC2=C1C=C(Cl)C(C)=C2)NC3=CC=C(OC4=CC=CN=C4C)N=C3.[H]Cl.[H]Cl
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SB 242084 dihydrochloride (Standard) Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SB 242084 dihydrochloride (Standard)1049747-87-65-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptoracute organ damageanxietydepressionschizophreniaSH-SY5YRPTC cellsInhibitorinhibitorinhibit

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