2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. H3R antagonist 7

H3R antagonist 7 (compounds 4) is a histamine subtype 3 receptor (H3R) antagonist with a Ki of 3.15 nM. H3R antagonist 7 is a potential PET radioligand for the study of central nervous system (CNS) diseases.

For research use only. We do not sell to patients.

H3R antagonist 7

H3R antagonist 7 Chemical Structure

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H3R antagonist 7 Related Antibodies

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Description

H3R antagonist 7 (compounds 4) is a histamine subtype 3 receptor (H3R) antagonist with a Ki of 3.15 nM. H3R antagonist 7 is a potential PET radioligand for the study of central nervous system (CNS) diseases[1].

IC50 & Target

H3 receptor

3.15 nM (Ki)

Molecular Weight

330.44

Formula

C20H27FN2O
SMILES

O=C(N1CCN(C2CCCCC2)CC1)[C@@H]3[C@@H](C4=CC=C(F)C=C4)C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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H3R antagonist 7 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

H3R antagonist 7Histamine Receptorcentral nervous system (CNS)histamine subtype 3 receptorAntagonistPETInhibitorinhibitorinhibit

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