2. Neuronal Signaling Immunology/Inflammation GPCR/G Protein
  3. Sigma Receptor Histamine Receptor
  4. KSK94

KSK94 is a high-affinity histamine H3 receptor antagonist, with Kis of 7.9, 2958, 75.2 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK94 can be used for research of nociceptive and neuropathic pain.

For research use only. We do not sell to patients.

KSK94

KSK94 Chemical Structure

CAS No. : 2566716-07-0

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25 mg Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks
50 mg Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks
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Based on 1 publication(s) in Google Scholar

KSK94 Related Antibodies

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Sigma 1 Receptor Sigma 2 Receptor

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H1 Receptor H2 Receptor H3 Receptor H4 Receptor Histamine Receptor

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Description

KSK94 is a high-affinity histamine H3 receptor antagonist, with Kis of 7.9, 2958, 75.2 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK94 can be used for research of nociceptive and neuropathic pain[1].

IC50 & Target

7.9, 2958, 75.2 nM (H3 receptor, sigma-1, sigma-2 receptor)[1]
Molecular Weight

398.50

Formula

C25H26N4O
CAS No.
SMILES

N#CC(C=C1)=CC=C1C2=CC=C(OCCCN3CCN(C4=CC=NC=C4)CC3)C=C2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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KSK94 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

KSK942566716-07-0KSK 94KSK-94Sigma ReceptorHistamine ReceptornociceptiveneuropathicpainhistamineInhibitorinhibitorinhibit

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