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α-Hydroxy Metoprolol-d<sub>5</sub> (Mixture of Diastereomers)

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Click Chemistry:	Labeling and Fluorescence Imaging (1) Azide (3) Alkynes (19)
Oligonucleotides:	Solvents (1) A (3) Nucleosides and their Analogs (3) Rat Pre-designed siRNA Sets (1) Phospholipids (1) Solubilizing Agents (1) Antisense Oligonucleotides (1) siRNAs (4) Nucleotides and their Analogs (2) U (1) Aptamers (1) Emulsifiers (2) Mouse Pre-designed siRNA Sets (1) Cationic Lipids (4) Human Pre-designed siRNA Sets (1)

5018

Inhibitors & Agonists

Screening Libraries

Fluorescent Dye

Biochemical Assay Reagents

Peptides

MCE Kits

Inhibitory Antibodies

144

Natural
Products

192

Recombinant Proteins

4260

Isotope-Labeled Compounds

265

Antibodies

Click Chemistry

Oligonucleotides

Targets Recommended: Nuclear Factor of activated T Cells (NFAT) P-glycoprotein

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-131396

α-Hydroxy Montelukast	Drug Metabolite	Inflammation/Immunology
α-Hydroxy Montelukast (M7) is a metabolite of Montelukast (HY-13315A) .

HY-W653769

*Deltamethrin-d5 (Mixture* of Diastereomers)**	Isotope-Labeled Compounds	Others
Deltamethrin-d5 (Mixture of Diastereomers) is the deuterium labeled Deltamethrin (Mixture of Diastereomers) .

HY-134670S

α-Hydroxy Metoprolol-d5 (Mixture of Diastereomers)	Isotope-Labeled Compounds	Others
α-Hydroxy Metoprolol-d₅ (Mixture of Diastereomers) is the deuterium labeled α-Hydroxy Metoprolol Mixture of Diastereomers .

HY-118714S

α-Hydroxy alprazolam-d5 U 40125-d<sub>5sub>; alpha-Hydroxyalprazolam-d<sub>5sub>	Isotope-Labeled Compounds	Others
α-Hydroxy alprazolam-d₅ (U 40125-d₅; alpha-Hydroxyalprazolam-d₅) is the deuterium labled α-hydroxy alprazolam (HY-118714).

HY-172744

α-Hydroxy bromazolam	Drug Metabolite	Metabolic Disease
α-Hydroxy bromazolam is a metabolite of Bromazolam catalyzed by CYP enzymes and can be found in plasma and urine. α-Hydroxy bromazolam is an important biomarker for Bromazolam intake .

HY-139367

α-Hydroxy flubromazolam	Drug Derivative	Neurological Disease
α-Hydroxy flubromazolam is a benzodiazepine.

HY-W753325

α-Hydroxy flualprazolam	Drug Metabolite	Neurological Disease
α-Hydroxy flualprazolam is a benzodiazepine.

HY-W705371

α-Hydroxy etizolam	Drug Metabolite GABA Receptor	Others
α-Hydroxy etizolam is the primary metabolite of Etizolam, possessing nearly identical pharmacological potency and high affinity for benzodiazepine receptors as Etizolam .

HY-132676S

*Ramiprilat-d5 (Mixture* of Diastereomers)**	Isotope-Labeled Compounds	Others
Ramiprilat-d₅ (Mixture of Diastereomers) is the deuterium labeled Ramiprilat (Mixture of Diastereomers) .

HY-A0115S

*Ramiprilat-d3 (Mixture* of Diastereomers)**	Isotope-Labeled Compounds Angiotensin-converting Enzyme (ACE) Endogenous Metabolite	Others
Ramiprilat-d₃ (Mixture of Diastereomers) is the deuterium labeled Ramiprilat (Mixture of Diastereomers) .

HY-W777700

*Cuscohygrine-d6 (mixture* of diastereomers)**	Isotope-Labeled Compounds	Others
Cuscohygrine-d₆ (mixture of diastereomers) is the deuterium labeled Cuscohygrine (Mixture of Diastereomers) (HY-N9904).

HY-W654395

*Methyl jasmonate-d5 (mixture* of diastereomers)** Methyl jasmonate-d<sub>5sub> (2,4,4-d3; acetyl-2,2-d2)(Mixture of Diastereomers)	Isotope-Labeled Compounds	Others
Methyl jasmonate-d₅ (mixture of diastereomers) is deuterium labeled Methyl (Z)-2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate .

HY-132706S

*N-Deformyl Formoterol-d6 Fumarate (Mixture* of Diastereomers)**	Isotope-Labeled Compounds	Others
N-Deformyl Formoterol-d₆ Fumarate (Mixture of Diastereomers) is the deuterium labeled N-Deformyl Formoterol Fumarate (Mixture of Diastereomers) .

HY-W742256

*N-Nitroso nebivolol (mixture* of diastereomers)**	Adrenergic Receptor	Cancer
N-Nitroso nebivolol (mixture of diastereomers) is a nitrosamine and mutagenic .

HY-W766409

*Ciclesonide-d11 (Mixture* of Diastereomers)**	Isotope-Labeled Compounds	Others
Ciclesonide-d₁₁ (Mixture of Diastereomers) is the deuterium labeled Ciclesonide.

HY-W768541

*Idarubicinol-d4 (Mixture* of Diastereomers)**	Isotope-Labeled Compounds	Others
Idarubicinol-d₄ (Mixture of Diastereomers) is the deuterium labeled Idarubicinol.

HY-128942

*MAC glucuronide α-hydroxy* lactone-linked SN-38**	Drug-Linker Conjugates for ADC	Cancer
MAC glucuronide α-hydroxy lactone-linked SN-38 (Topoisomerase I inhibitor) is a stabilized lactone MAC glucuronide α-hydroxy lactone-linked SN-38 agent linker. MAC glucuronide α-hydroxy lactone-linked SN-38 is cytotoxic across L540cy cells and Ramos cells with IC₅₀ values of 99 and 105 ng/mL, respectively .

HY-118714

α-Hydroxy alprazolam U 40125; alpha-Hydroxyalprazolam	Drug Metabolite	Neurological Disease
α-Hydroxy alprazolam (U 40125) is a main metabolite of Alprazolam. α-Hydroxy alprazolam is pharmacologically active accounting for 60% of the activity of Alprazolam .

HY-W744273

*Pravastatin-d9 Sodium (mixture* of 2 diastereomers)**	Isotope-Labeled Compounds	Others
Pravastatin-d₉ Sodium (mixture of 2 diastereomers) is the deuterium labeled Pravastatin Sodium.

HY-12650S

*Mirogabalin-13C2,d1 (Mixture* of Diastereomers)** DS5565-¹³C<sub>2sub>,d<sub>1sub> (Mixture of Diastereomers)	Isotope-Labeled Compounds	Others
Mirogabalin-13C2,d1 (Mixture of Diastereomers) is a C13 and deuterium labeled Mirogabalin. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS .

HY-132379S

Hydroxy Pioglitazone-d5 (M-IV) (Mixture of-diastereomers)	Isotope-Labeled Compounds	Others
Hydroxy Pioglitazone-d₅ (M-IV) (Mixture of-diastereomers) is the deuterium labeled Hydroxy Pioglitazone (M-IV) (Mixture of-diastereomers) .

HY-W711709

*Terameprocol-d12 (Mixture* of Diastereomers)**	Isotope-Labeled Compounds	Others
Terameprocol-d₁₂ (Mixture of Diastereomers) is the deuterium labeled 4,4'-(2,3-Dimethylbutane-1,4-diyl)bis(1,2-dimethoxybenzene) (HY-W422348).

HY-W777284

*Zeranol-d5 (mixture* of diastereomers)**	Isotope-Labeled Compounds Estrogen Receptor/ERR	Endocrinology
Zeranol-d₅ (mixture of diastereomers) is the deuterium labeled Zeranol (HY-N6709). Zeranol, a metabolite of the mycoestrogen zearalenone, is an estrogen receptor agonist. Zeranol is used as a growth promoter of livestock due to its strong estrogenic activity .

HY-W654209

*Glycopyrrolate iodide-d3 (mixture* of diastereomers)**	Isotope-Labeled Compounds	Others
Glycopyrrolate iodide-d₃ (mixture of diastereomers) is deuterium labeled 3-(2-Cyclopentyl-2-hydroxy-2-phenylacetoxy)-1,1-dimethylpyrrolidin-1-ium iodide .

HY-113026S

*(2RS,4R,8R)-δ-Tocopherol-d4 (Mixture* of Diastereomers)**	Endogenous Metabolite Isotope-Labeled Compounds	Others
(2RS,4R,8R)-δ-Tocopherol-d₄ (Mixture of Diastereomers) is the deuterium labeled (2RS,4R,8R)-δ-Tocopherol (Mixture of Diastereomers) .

HY-W100026S

*Galaxolide-d6 (mixture* of diastereomers) (>80%)**	Isotope-Labeled Compounds Glutathione S-transferase Estrogen Receptor/ERR	Endocrinology
Galaxolide-d₆ (mixture of diastereomers) (>80%) is the deuterium labeled Galaxolide (HY-W100026). Galaxolide can induce estrogenic activity (Estrogen Receptor/ERR), trigger oxidative stress and genotoxicity, and induce EROD and GST (Glutathione S-transferase) enzyme activity .

HY-152040S

*Tenuazonic acid-(acetyl-13C2) (mixture* of diastereomers) in methanol** 3-(Acetyl-¹³C<sub>2sub>)-5-((S)-sec-butyl)-4-Hydroxy-1,5-dihydro-2H-pyrrol-2-one	Isotope-Labeled Compounds	Others
Tenuazonic acid-(acetyl- ¹³C₂) (mixture of diastereomers) in methanol (3-(Acetyl- ¹³C₂)-5-((S)-sec-butyl)-4-hydroxy-1,5-dihydro-2H-pyrrol-2-one) is ¹³C labeled Tenuazonic acid-(acetyl) (mixture of diastereomers) in methanol .

HY-150857S

*Thymine-α,α,α,6-d4 Glycol (mixture* of diastereomers)-d4**	Isotope-Labeled Compounds	Others
Thymine-α,α,α,6-d₄ Glycol (mixture of diastereomers)-d₄ is the deuterium labeled Thymine-α,α,α,6-d4 Glycol (mixture of diastereomers) .

HY-172743

α-Hydroxy phenazolam	Drug Metabolite	Metabolic Disease
α-Hydroxyphenazolam is a metabolite of Phenazolam .

HY-17503S

Metoprolol-d7	Isotope-Labeled Compounds Adrenergic Receptor	Cardiovascular Disease Endocrinology
Metoprolol-d₇ is the deuterium labeled Metoprolol. Metoprolol (Toprol) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension[1][2].

HY-17503S3

Metoprolol-d5	Apoptosis Adrenergic Receptor	Cancer
Metoprolol-d₅ is the deuterium labeled Metoprolol . Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-17503AS

Metoprolol-d7 hydrochloride	Isotope-Labeled Compounds Adrenergic Receptor	Infection Cardiovascular Disease Endocrinology Cancer
Metoprolol-d₇ (hydrochloride) is the deuterium labeled Metoprolol. Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-132382S

*β-Sitosterol-d7 (mixture* of diasteromers)**	Isotope-Labeled Compounds	Others
β-Sitosterol-d₇ (Mixture of Diastereomers) is the deuterium labeled β-Sitosterol (mixture of diasteromers) .

HY-170045

(±)-9α-Hydroxy hexahydrocannabinol (±)-9α-Hydroxy HHC; (±)-9α-OH-HHC	Cannabinoid Receptor	Neurological Disease
(±)-9α-Hydroxy hexahydrocannabinol ((±)-9α-Hydroxy HHC) is structurally similar to known phytocannabinoids .

HY-17503BS

Metoprolol-d6 tartrate	Isotope-Labeled Compounds Adrenergic Receptor	Infection Cardiovascular Disease Endocrinology Cancer
Metoprolol-d₆ (tartrate) is the deuterium labeled Metoprolol tartrate. Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-17503AS1

Metoprolol-d6 succinate	Isotope-Labeled Compounds Adrenergic Receptor Apoptosis	Cardiovascular Disease Endocrinology Cancer
Metoprolol-d₆ (succinate) is deuterium labeled Metoprolol (succinate). Metoprolol succinate is an orally active, selective β1-adrenoceptor antagonist. Metoprolol succinate shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-W740664

20α-Hydroxy Cholesterol-d7	Isotope-Labeled Compounds	Others
20α-Hydroxy Cholesterol-d₇ is the deuterium labeled 20α-Hydroxy Cholesterol.

HY-W740771

6α-Hydroxy cortisol-d4	Isotope-Labeled Compounds	Others
6α-Hydroxy cortisol-d₄ is the deuterium labeled 6α-Hydroxy cortisol.

HY-136347R

3α-Hydroxy pravastatin sodium (Standard)	Reference Standards HMG-CoA Reductase (HMGCR) Drug Metabolite	Cardiovascular Disease
3α-Hydroxy pravastatin (sodium) (Standard) is the analytical standard of 3α-Hydroxy pravastatin (sodium). This product is intended for research and analytical applications. 3α-Hydroxy pravastatin sodium is the major metabolite of Pravastatin. Pravastatin is a competitive HMG-CoA reductase inhibitor .

HY-131654

16α-Hydroxy progesterone	Biochemical Assay Reagents	Others
16α-Hydroxy progesterone is a biochemical reagent.

HY-125348S

6α-Hydroxy Paclitaxel-d5	Isotope-Labeled Compounds	Cancer
6α-Hydroxy Paclitaxel-d₅ is the deuterium labeled 6α-Hydroxy paclitaxel. 6α-Hydroxy paclitaxel is a primary metabolite of Paclitaxel. 6α-Hydroxy paclitaxel retains a time-dependent effect on organic anion-transporting polypeptides 1B1/SLCO1B1 (OATP1B1) with similar inhibition potency to Paclitaxel, whereas it no longer showed time-dependent inhibition of OATP1B3. 6α-Hydroxy paclitaxel can be used for the research of cancer .

HY-W400424

(-)-6α-Hydroxy cannabidiol	Cannabinoid Receptor	Neurological Disease
(-)-6α-Hydroxy cannabidiol is a metabolite of Cannabidiol .

HY-133966S

6α-Hydroxy-5α-cholestane-d7	Isotope-Labeled Compounds	Others
6α-Hydroxy-5α-cholestane-d₇ is deuterium labeled 6α-Hydroxy-5α-cholestane.

HY-114744

6α-Hydroxy metandienone	Androgen Receptor	Endocrinology
6α-Hydroxy metandienone is an androgenic anabolic steroid metabolite of Metandienone.

HY-125348

6α-Hydroxy paclitaxel	Drug Metabolite	Cancer
6α-Hydroxy paclitaxel is a primary metabolite of Paclitaxel. 6α-Hydroxy paclitaxel retains a time-dependent effect on *organic anion–transporting polypeptides 1B1/SLCO1B1* (OATP1B1) with similar inhibition potency to Paclitaxel, whereas it no longer showed time-dependent inhibition of OATP1B3**. 6α-Hydroxy paclitaxel can be used for the research of cancer .

HY-113031S1

16α-Hydroxydehydroepiandrosterone-d5 16α-Hydroxy-DHEA-d<sub>5sub>; 16α-OH-DHEA-d<sub>5sub>	Isotope-Labeled Compounds Endogenous Metabolite	Metabolic Disease
16α-Hydroxydehydroepiandrosterone-d₅ (16α-Hydroxy-DHEA-d₅) is the deuterium labeled 16α-Hydroxydehydroepiandrosterone (HY-113031) .

HY-W683681

16α-Hydroxy etiocholanolone	Cytochrome P450	Endocrinology
16α-Hydroxy etiocholanolone is a metabolite of 16a-Hydroxydehydroisoandrosterone (HY-113031) .

HY-123519

14α-Hydroxy Paspalinine	Insecticide	Infection
14α-Hydroxy Paspalinine is a paspalinine derivative with antiinsectan activity from the sclerotia of Aspergillus nomius .

HY-136347

3α-Hydroxy pravastatin sodium	HMG-CoA Reductase (HMGCR) Drug Metabolite	Cardiovascular Disease
3α-Hydroxy pravastatin sodium is the major metabolite of Pravastatin. Pravastatin is a competitive HMG-CoA reductase inhibitor .

HY-128041

alpha-Hydroxy farnesyl phosphonic acid Hydroxyfarnesyl phosphate	Farnesyl Transferase	Others
α-hydroxy Farnesyl phosphonic acid is a nonhydrolyzable analog of farnesyl pyrophosphate which acts as a competitive inhibitor of farnesyl transferase (FTase). At concentrations greater than 1 μM, α-hydroxy farnesyl phosphonic acid inhibits the processing of Ras in Ha-ras-transformed NIH3T3 cells.

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-113259

7α-Hydroxy-4-cholesten-3-one	Structural Classification Microorganisms Classification of Application Fields Source classification Metabolic Disease Endogenous metabolite Disease Research Fields Steroids	Endogenous Metabolite
7α-Hydroxy-4-cholesten-3-one is an intermediate in synthesis of bile acids from cholesterol. 7α-Hydroxy-4-cholesten-3-one is a pregnane X receptor (PXR) agonist. 7α-Hydroxy-cholest-4-en-3-one is a biomarker for bile acid loss, irritable bowel syndrome, and other diseases associated with defective bile acid biosynthesis. 7α-Hydroxy-cholest-4-en-3-one is the physiological substrate for CYP8B1 .

HY-N6013

*Aloin(mixture* of A&B)**	Infection Liliaceae Classification of Application Fields Ketones, Aldehydes, Acids Source classification Phenols Polyphenols Aloe vera (L.) Burm. f. Plants Inflammation/Immunology Disease Research Fields	MMP Bacterial Fungal
Aloin (mixture of A&B) is anthraquinone derivative isolated from Aloe vera. Aloin (mixture of A&B) has diverse biological activities such as anti-inflammatory, immunity, antidiabetic, antioxidant, antibacterial, antifungal, and antitumor activities. Aloin (mixture of A&B) also an effective inhibitor of stimulated granulocyte matrix metalloproteinases (MMPs) .

HY-123519

14α-Hydroxy Paspalinine	Infection Alkaloids Structural Classification Microorganisms Classification of Application Fields Source classification Disease Research Fields Indole Alkaloids	Insecticide
14α-Hydroxy Paspalinine is a paspalinine derivative with antiinsectan activity from the sclerotia of Aspergillus nomius .

HY-113259R

7α-Hydroxy-4-cholesten-3-one (Standard)	Structural Classification Classification of Application Fields Source classification Metabolic Disease Endogenous metabolite Disease Research Fields Steroids	Reference Standards Endogenous Metabolite
7α-Hydroxy-4-cholesten-3-one (Standard) is the analytical standard of 7α-Hydroxy-4-cholesten-3-one. This product is intended for research and analytical applications. 7α-Hydroxy-4-cholesten-3-one is an intermediate in synthesis of bile acids from cholesterol. 7α-Hydroxy-4-cholesten-3-one is a pregnane X receptor (PXR) agonist. 7α-Hydroxy-cholest-4-en-3-one is a biomarker for bile acid loss, irritable bowel syndrome, and other diseases associated with defective bile acid biosynthesis. 7α-Hydroxy-cholest-4-en-3-one is the physiological substrate for CYP8B1 .

HY-N1729

2α-Hydroxy-1,8-cineole	Structural Classification Natural Products Classification of Application Fields Source classification Metabolic Disease Endogenous metabolite Disease Research Fields	Endogenous Metabolite
2α-Hydroxy-1,8-cineole is a metabolite of 1,8-cineole (HY-N0066) .

HY-N12136

1α-Hydroxy-3-deoxypseudoanisatin	Structural Classification Terpenoids Sesquiterpenes Source classification Plants Illicium merrillianum A. C. Smith Schisandraceae	Others
1α-Hydroxy-3-deoxypseudoanisatin (Iso-γ-fagarine) is a sesquiterpenoid obtained from star anise (Illicium merrillianum) isolated from the peel .

HY-N9137

2α-Hydroxy-8β-(2-methylbutyryloxy)costunolide	Structural Classification Terpenoids Sesquiterpenes Artemisia myriantha Wall. ex Besser Source classification Asteraceae Plants	Others
2α-Hydroxy-8β-(2-methylbutyryloxy)costunolide is a Sesquiterpenoids product that can be isolated from the aerial parts of Artemisia myriantha .

HY-131152

*Leucinostatin (mixture* of A&B)**	Structural Classification Microorganisms Antifungal Classification of Application Fields Antibiotics Source classification Antibacterial Disease Research Anticancer Inflammation/Immunology Disease Research Fields Other Antibiotics	Antibiotic
Leucinostatin (mixture of A&B), the major components of an atypical nonapeptide complex produced by Paecilomyces lilacinus, are antibiotics .

HY-N11644

Lanosta-7,9(11),24-trien-3α-hydroxy-26-oic acid	Triterpenes Structural Classification Microorganisms Terpenoids Source classification	Others
Lanosta-7,9(11),24-trien-3α-hydroxy-26-oic acid, also known as ganoderic acid 24. Lanosta-7,9(11),24-trien-3α-hydroxy-26-oic acid shows high cytotoxicity against cancer cells, such as human lung cancer cells CH27, melanoma cells M21, and oral cancer cells HSC-3 .

HY-N3810

ent-11α-Hydroxy-15-oxokaur-16-en-19-oic acid	Structural Classification Terpenoids Source classification Pteridaceae Diterpenoids Plants Pteris semipinnata L. Sp.	Tyrosinase
ent-11α-Hydroxy-15-oxokaur-16-en-19-oic acid is an anti-melanin synthesis tyrosinase inhibitor, which can be isolated from Pteris fern. ent-11α-Hydroxy-15-oxokaur-16-en-19-oic acid regulates the melanogenesis transcription factor microphthalmia-associated transcription factor (MITF). The 11α-OH, 15-oxo and 16-en moieties of ent-11α-Hydroxy-15-oxokaur-16-en-19-oic acid are key fragments that inhibit melanin synthesis. The 19-COOH moiety has been implicated in the inhibition of cytotoxicity associated with 11α-OH KA and related compounds .

HY-W018512

7-Ketolithocholic acid 4 Publications Verification 3α-Hydroxy-7-oxo-5β-cholanic acid	Structural Classification Microorganisms Classification of Application Fields Source classification Metabolic Disease Endogenous metabolite Disease Research Fields Steroids	Endogenous Metabolite
7-Ketolithocholic acid (3α-Hydroxy-7-oxo-5β-cholanic acid), a bile acid, can be absorbed and suppresses endogenous bile acid production and biliary cholesterol secretion .

HY-W018772R

*D-Ribose(mixture* of isomers) (Standard)**	Structural Classification Microorganisms Source classification Endogenous metabolite Saccharides	Reference Standards Endogenous Metabolite
D-Ribose(mixture of isomers) (Standard) is the analytical standard of D-Ribose(mixture of isomers). This product is intended for research and analytical applications. D-Ribose(mixture of isomers) is an energy enhancer, and acts as a sugar moiety of ATP, and widely used as a metabolic therapy supplement for chronic fatigue syndrome or cardiac energy metabolism. D-Ribose(mixture of isomers) is active in protein glycation, induces NF-κB inflammation in a RAGE-dependent manner .

HY-W018772

*D-Ribose(mixture* of isomers)** 3 Publications Verification	Structural Classification Microorganisms Classification of Application Fields Source classification Endogenous metabolite Disease Research Fields Saccharides Cancer	Endogenous Metabolite
D-Ribose(mixture of isomers) is an energy enhancer, and acts as a sugar moiety of ATP, and widely used as a metabolic therapy supplement for chronic fatigue syndrome or cardiac energy metabolism. D-Ribose(mixture of isomers) is active in protein glycation, induces NF-κB inflammation in a RAGE-dependent manner .

HY-150356MR1

Mixture of Aflatoxins in Acetonitrile (Standard)	Structural Classification Microorganisms Source classification Phenylpropanoids Endogenous metabolite	Reference Standards
Mixture of Aflatoxins in Acetonitrile (Standard) is mainly used for the detection of aflatoxins in grain, oils, foods and traditional Chinese medicines

HY-W018512R

7-Ketolithocholic acid (Standard) 3α-Hydroxy-7-oxo-5β-cholanic acid (Standard)	Structural Classification Microorganisms Source classification Endogenous metabolite Steroids	Reference Standards Endogenous Metabolite
7-Ketolithocholic acid (Standard) is the analytical standard of 7-Ketolithocholic acid. This product is intended for research and analytical applications. 7-Ketolithocholic acid (3α-Hydroxy-7-oxo-5β-cholanic acid), a bile acid, can be absorbed and suppresses endogenous bile acid production and biliary cholesterol secretion .

HY-N2766

8alpha-Hydroxy-alpha-gurjunene	Structural Classification Terpenoids Sesquiterpenes Source classification Sarcandra glabra (Thunb.) Nakai Chloranthaceae Plants	Others
8alpha-Hydroxy-alpha-gurjunene is a Sesquiterpenoids product that can be isolated from the herbs of Sarcandra glabra .

HY-N9083

8α-Hydroxy-α-gurjunene	Structural Classification Flavonoids Leguminosae Source classification Plants Sophora tomentosa L.	Others
8α-Hydroxy-α-gurjunene is a Flavonoids product that can be isolated from the aerial parts of Sophora tomentosa L. .

HY-N12135

15α-Hydroxy-20-oxo-6,7-seco-ent-kaur-16-en-1,7α(6,11α)-diolide	Structural Classification Terpenoids Labiatae Source classification Diterpenoids Plants Cyrtocymura cincta var. cincta	Others
15α-Hydroxy-20-oxo-6,7-seco-ent-kaur-16-en-1,7α(6,11α)-diolide (compound 2) is an enantio-kaurene diterpenoid (ent -kaurene diterpenoid), which can be isolated from Rubescens rubescens. 15α-Hydroxy-20-oxo-6,7-seco-ent-kaur-16-en-1,7α(6,11α)-diolide has cellular activity against EC-1, U87, A549, MCF-7 and HeLa cell lines Toxicity, IC₅₀s are 37.69 μM, 79.362 μM, 80.07 μM, 197.35 μM, 462.13 μM, and 180.09 μM respectively .

HY-125833

Alpha-Naphthoflavone 5+ Cited Publications	Flavonoids Flavones Source classification Indigofera heterantha Wall. ex Brand. Plants Compositae Disease Research Fields Cancer	Cytochrome P450 Aryl Hydrocarbon Receptor Apoptosis
Alpha-Naphthoflavone is an orally active flavonoid that is a potent, competitive inhibitor of aromatase< b>aromatase. < b > IC < sub > 50 < / sub > < / b > and < b > K < sub > I < / sub > < / b > value were 0.5 and 0.2 microns. Alpha-Naphthoflavone can inhibit cell proliferation and induce apoptosis .

HY-125833R

Alpha-Naphthoflavone (Standard)	Flavonoids Flavones Source classification Indigofera heterantha Wall. ex Brand. Plants Compositae	Cytochrome P450 Aryl Hydrocarbon Receptor Apoptosis
Alpha-Naphthoflavone (Standard) is the analytical standard of Alpha-Naphthoflavone. This product is intended for research and analytical applications. Alpha-Naphthoflavone is an orally active flavonoid that is a potent, competitive inhibitor of aromatase< b>aromatase. < b > IC < sub > 50 < / sub > < / b > and < b > K < sub > I < / sub > < / b > value were 0.5 and 0.2 microns. Alpha-Naphthoflavone can inhibit cell proliferation and induce apoptosis .

HY-N11799

Neochilenin 3-O-Methylquercetin 4′-O-glucoside	Structural Classification Flavonoids Source classification Plants Compositae Other Flavonoids	Others
Neochilenin (3-O-Methylquercetin 4 '-O-glucoside) is a glycoside of 3-O-methylquercetin, which can be isolated from the sub-family Cereoideae (Cactaceae). .

HY-139637

(±)-Silybin Silibinin (Mixture of Silybin A and Silybin B)	Structural Classification Flavanonols Flavonoids Source classification Cyamopsis tetragonoloba (L.) Taub. Plants Compositae	Apoptosis
(±)-Silybin is the racemate of Silybin (HY-N0779A). Silybin induces apoptosis and exhibits hepatoprotective, antioxidant, anti-inflammatory, anti-cancer activity .

HY-145751

7α-Hydroxy-DHEA 7α-Hydroxydehydroepiandrosterone; 3β,7α-DiHydroxy-Δ5-androsten-17-one	Structural Classification Source classification Endogenous metabolite Steroids	Cytochrome P450 Mitochondrial Metabolism
7α-Hydroxy-DHEA (7α-Hydroxydehydroepiandrosterone) is a 7α-hydroxylated metabolite of DHEA (HY-14650), catalyzed by intracellular steroid 7α-hydroxylases such as P450 2A1. 7α-Hydroxy-DHEA exhibits biological activity comparable to DHEA but does not convert into compounds with androgenic or estrogenic activity. It induces the activity of thermogenic enzymes such as mitochondrial sn-glycerol-3-phosphate dehydrogenase and cytosolic malic enzyme, enhancing heat production and reducing food utilization efficiency. As a more efficient and safer metabolite compared to DHEA, 7α-Hydroxy-DHEA holds potential for studies in the fields of obesity, metabolic diseases, and adrenal carcinoma .

HY-113038B

α-Hydroxyglutaric acid 2-Hydroxyglutarate; 2-Hydroxyglutaric acid; 2-Hydroxypentanedioic acid	Structural Classification Immune System Disorder Microorganisms Classification of Application Fields Ketones, Aldehydes, Acids Source classification Disease markers Endocrine diseases Nervous System Disorder Endogenous metabolite Disease Research Fields Cancer	Histone Demethylase Endogenous Metabolite
α-Hydroxyglutaric acid (2-Hydroxyglutarate) is an α-hydroxy acid form of glutaric acid. α-Hydroxyglutaric acid is a competitive inhibitor of multiple α-ketoglutarate-dependent dioxygenases, including histone demethylases and the TET family of 5-methlycytosine (5mC) hydroxylases .

HY-W011474

Geranylgeraniol	Structural Classification Natural Products Microorganisms	NF-κB
Geranylgeraniol is an orally acitve vitamin K₂ sub-type, an intermediate of the mevalonate pathway. Geranylgeraniol targets NF-kB signaling pathway and could alleviate LPS-induced microglial inflammation in animal model .

HY-113038A

α-Hydroxyglutaric acid disodium 2-Hydroxyglutarate disodium; 2-Hydroxyglutaric acid disodium; 2-Hydroxypentanedioic acid disodium	Structural Classification Classification of Application Fields Ketones, Aldehydes, Acids Source classification Endogenous metabolite Disease Research Fields Cancer	Histone Demethylase Endogenous Metabolite
α-Hydroxyglutaric acid (2-Hydroxyglutarate) disodium is an α-hydroxy acid form of glutaric acid. α-Hydroxyglutaric acid disodium is a competitive inhibitor of multiple α-ketoglutarate-dependent dioxygenases, including histone demethylases and the TET family of 5-methlycytosine (5mC) hydroxylases .

HY-N15356

9-Oxooctadecanedioic acid	Structural Classification Ketones, Aldehydes, Acids Source classification Plants Quercus suber L. Fagaceae	Bacterial
9-Oxooctadecanedioic acid is an α,ω-dicarboxylic fatty acid monomer found in the cork suberin of Quercus suber. It contributes to the formation of the hydrophobic barrier structure in plant cell walls and may play an important role in functions such as water resistance and protection against microbial penetration .

HY-P2274

Argifin	Infection Structural Classification Natural Products Microorganisms Classification of Application Fields Source classification Disease Research Fields	Parasite
Argifin is a sub-nanomolar chitinase inhibitor produced by soil microorganisms, with IC₅₀s of 0.025 μM, 6.4 μM , 1.1 μM and 4.5 μM for SmChiA (Serratia marcescens chitinaese A), SmChiB, Aspergillus fumigatus chitinase B1 and human chitotriosidase, respectively .

HY-W011474R

Geranylgeraniol (Standard)	Structural Classification Natural Products Microorganisms	Reference Standards NF-κB
Geranylgeraniol (Standard) is the analytical standard of Geranylgeraniol. This product is intended for research and analytical applications. Geranylgeraniol is an orally acitve vitamin K2 sub-type, an intermediate of the mevalonate pathway. Geranylgeraniol targets NF-kB signaling pathway and could alleviate LPS-induced microglial inflammation in animal model [4].

HY-N10192

Aculene D	Infection Microorganisms Classification of Application Fields Terpenoids Sesquiterpenes Source classification Disease Research Fields	Endogenous Metabolite Bacterial
Aculene D, a fungal metabolite, shows quorum sensing (QS) inhibitory activity against Chromobacterium violaceum CV026, and could significantly reduce violacein production in N-hexanoyl-l-homoserine lactone (C6-HSL) induced C. violaceum CV026 cultures at sub-inhibitory concentrations .

HY-N0662

Amentoflavone 5+ Cited Publications Didemethyl-ginkgetin	Structural Classification Flavonoids Classification of Application Fields Source classification Phenols Polyphenols Selaginellaceae Plants Biflavones Selaginella tamariscina (P. Beauv.) Spring Disease Research Fields Cancer	Reactive Oxygen Species (ROS) Apoptosis Bacterial Fungal RSV GABA Receptor
Amentoflavone (Didemethyl-ginkgetin) is a potent and orally active GABA(A) negative modulator. Amentoflavone also shows anti-inflammatory, antioxidative, anti-viral, anti-tumor, anti-radiation, anti-fungal, antibacterial activity. Amentoflavone induces apoptosis and cell cycle arrest at sub-G1 phase .

HY-N15496

Fusaproliferin FUS	Structural Classification Microorganisms Terpenoids Sesquiterpenes Source classification	Reactive Oxygen Species (ROS) NO Synthase Interleukin Related TNF Receptor p38 MAPK ERK IKK NF-κB
Fusaproliferin is a sesterterpene mycotoxin isolated from Fusarium solani. Fusaproliferin reverse Lipopolysaccharides (HY-D1056) stimulation and the NF-κB and MAPKs signaling pathways contribute to the anti-inflammatory process. Fusaproliferin exhibits affinity for the TLR4 protein with K_D values of 28.6 μM. Fusaproliferin shows cytotoxicity against pancreatic cancer cell with rapid and sub-micromolar IC₅₀ .

HY-W011370

Pelargonidin chloride 1 Publications Verification	Structural Classification Anthocyans Flavonoids Classification of Application Fields Leguminosae Source classification Other Diseases Phenols Polyphenols Plants Phaseolus vulgaris Linn. Disease Research Fields	Quinone Reductase Reactive Oxygen Species (ROS)
Pelargonidin chloride is an anthocyanidin and also is a scavenger of nitric oxide radical and has antioxidant activities. Pelargonidin inhibits cell viability and induces cell cycle arrest at sub-G1 phase. Pelargonidin chloride increases the mRNA and protein expression of HO-1, NQO1, Nrf2. Pelargonidin chloride improves Aβ-induced memory and learning impairment .

HY-P2274R

Argifin (Standard)	Structural Classification Natural Products Microorganisms Source classification	Reference Standards Parasite
Argifin (Standard) is the analytical standard of Argifin. This product is intended for research and analytical applications. Argifin is a sub-nanomolar chitinase inhibitor produced by soil microorganisms, with IC50s of 0.025 μM, 6.4 μM , 1.1 μM and 4.5 μM for SmChiA (Serratia marcescens chitinaese A), SmChiB, Aspergillus fumigatus chitinase B1 and human chitotriosidase, respectively[1].

HY-N8549A

5-Dihydrocortisone	Structural Classification Classification of Application Fields Cardiacglycosides Source classification Metabolic Disease Endogenous metabolite Disease Research Fields Steroids	Endogenous Metabolite
5-Dihydrocortisone is a 5-Dihydrocortisone with mixture of isomers. 5β-Dihydrocortisone is a sterol metabolite of cortisone by 5β-reductase (AKR1D1) in liver

HY-N0662R

Amentoflavone (Standard) Didemethyl-ginkgetin (Standard)	Structural Classification Flavonoids Source classification Phenols Polyphenols Selaginellaceae Plants Biflavones Selaginella tamariscina (P. Beauv.) Spring	Reference Standards Reactive Oxygen Species (ROS) Apoptosis Bacterial Fungal RSV GABA Receptor
Amentoflavone (Standard) is the analytical standard of Amentoflavone. This product is intended for research and analytical applications. Amentoflavone (Didemethyl-ginkgetin) is a potent and orally active GABA(A) negative modulator. Amentoflavone also shows anti-inflammatory, antioxidative, anti-viral, anti-tumor, anti-radiation, anti-fungal, antibacterial activity. Amentoflavone induces apoptosis and cell cycle arrest at sub-G1 phase .

HY-W008150

*2-Hydroxy-3-methylbutanoic acid* 1 Publications Verification α-Hydroxyisovaleric acid	Structural Classification Ketones, Aldehydes, Acids Source classification Disease markers Endocrine diseases Nervous System Disorder Endogenous metabolite	Endogenous Metabolite
2-Hydroxy-3-methylbutanoic acid is an α-hydroxy analogue of valine and a valine precursor that reduces urea excretion. 2-Hydroxy-3-methylbutanoic acid can promote the growth of chickens and rats, and is converted into valine in the body, participating in protein synthesis and maintaining nitrogen balance, thereby supporting animal growth and development. 2-Hydroxy-3-methylbutanoic acid has a more significant effect on the valine-deficient dietary model. 2-Hydroxy-3-methylbutanoic acid is mainly used in animal nutrition research to evaluate its potential application as a nitrogen source substitute in feed .

HY-B0504S

Creatinine-d3 5 Publications Verification NSC13123-d<sub>3sub>	Classification of Application Fields Metabolic Disease Disease Research Fields	Isotope-Labeled Compounds Endogenous Metabolite
Creatinine-d₃ is a deuterium labeled Creatinine. Creatinine is a break-down product of creatine phosphate in muscle .

HY-113434B

5-HETE (±)-5-HETE	Structural Classification Classification of Application Fields Ketones, Aldehydes, Acids Source classification Endogenous metabolite Inflammation/Immunology Disease Research Fields	Endogenous Metabolite
5-HETE ((±)-5-HETE), a fatty acid, is a oxidative derivative of Arachidonic acid. 5-HETE is a mixture of 5(S)-HETE and 5(R)-HETE. 5-HETE is a potent aggregating agent that induces the aggregation of neutrophils with an IC₅₀ value of 200 nM .

HY-B0172R

Lithocholic acid (Standard) 10+ Cited Publications 3α-Hydroxy-5β-cholanic acid (Standard)	Structural Classification Human Gut Microbiota Metabolites Microorganisms Classification of Application Fields Anti-aging Source classification Metabolic Disease Endogenous metabolite Disease Research Fields Steroids	Reference Standards Autophagy Endogenous Metabolite Apoptosis FXR
Lithocholic acid (Standard) is the analytical standard of Lithocholic acid. This product is intended for research and analytical applications. Lithocholic acid is a toxic secondary bile acid that can promote intrahepatic cholestasis and promote tumorigenesis. Lithocholic acid is also a FXR antagonist and a PXR/SXR agonist ^[5].

HY-113319R

β-D-Fructose,98%(mixtures) (Standard)	Structural Classification Source classification Endogenous metabolite Saccharides Monosaccharides	Endogenous Metabolite
β-D-Fructose,98%(mixtures) (Standard) is the analytical standard of β-D-Fructose,98%(mixtures). This product is intended for research and analytical applications. β-D-Fructose is a β-fruit sugar that can be produced by the hydrolysis of sucrose. β-D-Fructose can be used as a sweetness potentiator. β-D-Fructose can be designed as a units of antiproliferative agents against breast (MCF-7) and colon (MDST8) cancer cell lines .

HY-N7265

Epi-galantamine	Alkaloids other families Source classification Plants	Cholinesterase (ChE)
Epi-galantamine is a diastereomer of Galantamine. Epi-galantamine is an alkaloid isolated from the bulbs and flowers of Caucasian snowdrop (Galanthus woronowii). Epi-galantamine inhibits AChE with an EC₅₀ of 45.7 μM .

HY-N2353

Arabinose (±)-Arabinose; DL-Arabinose; dl-Arabinose	Structural Classification Classification of Application Fields Source classification Metabolic Disease Endogenous metabolite Disease Research Fields Saccharides	Endogenous Metabolite
Arabinose is a 5-carbon sugar often found in plants. Arabinose is chiral diastereomer that exhibits specific crystallization behavior. Arabinose can be used as excipients or cocrystallization agents in pharmaceutical formulations. Arabinose is an intermediate for drug synthesis .

HY-133185

Megastigmatrienone (mixed isomers)	Microorganisms Source classification	Drug Derivative
Megastigmatrienone (mixed isomers) is a mixture of isomers of Megastigmatrienone, a compound that has the aroma of tobacco.

HY-N2078

Yamogenin Neodiosgenin	Structural Classification other families Classification of Application Fields Source classification Metabolic Disease Plants Disease Research Fields Steroids	LXR
Yamogenin (Neodiosgenin) is a diastereomer of diosgenin. Yamogenin (Neodiosgenin) antagonizes the activation of the liver X receptor (LXR) in luciferase ligand assay. Yamogenin (Neodiosgenin) inhibits triacylglyceride (TG) accumulation through the suppression of gene expression of fatty acid synthesis in HepG2 hepatocytes .

HY-W794998

Cedarwood terpenes	Structural Classification Other Monoterpenes Cedrus deodara (Roxburgh) G. Don Pinaceae Terpenoids Source classification Plants	Others
Cedarwood terpenes is a natural terpene mixture that can be extracted from cedar wood .

HY-N9761

Murrayanine	Structural Classification Alkaloids Pyrrole Alkaloids Source classification Rutaceae Murraya koenigii (L.) Spreng Plants	Others
Murrayanine is a dimeric pyranoquinoline alkaloid, a mixture of two enantiomers with a predominant configuration on the chiral axis .

HY-N7084

Methyl dihydrojasmonate	Structural Classification Oleaceae Classification of Application Fields Ketones, Aldehydes, Acids Source classification Other Diseases Jasminum grandiflorum Plants Disease Research Fields	Others
Methyl dihydrojasmonate is a fragrance ingredient with a jasmine-like odor, used in many fragrance mixtures .

HY-125932A

9β-Debilon	Structural Classification Terpenoids Sesquiterpenes Source classification Nardostachys jatamansi (D. Don) DC. Plants Valerianaceae	Serotonin Transporter
9β-Debilon is a sesquiterpenoid compound found in Nardostachys chinensis and may possess SERT regulatory activity. Structurally, 9β-Debilon is a diastereomer of Debilon (HY-125932). 9β-Debilon holds potential for research into neurological disorders .

HY-N0683A

rel-α-Vitamin E rel-D-α-Tocopherol	Structural Classification Natural Products Monophenols other families Classification of Application Fields Source classification Phenols Plants Inflammation/Immunology Disease Research Fields	Bacterial Influenza Virus Reactive Oxygen Species (ROS) Endogenous Metabolite
rel-α-Vitamin E (rel-D-α-Tocopherol) is a vitamin with antioxidant properties and also a mixture .

Cat. No.	Product Name	Chemical Structure

HY-W653769

*Deltamethrin-d5 (Mixture* of Diastereomers)**
Deltamethrin-d5 (Mixture of Diastereomers) is the deuterium labeled Deltamethrin (Mixture of Diastereomers) .

HY-134670S

α-Hydroxy Metoprolol-d5 (Mixture of Diastereomers)
α-Hydroxy Metoprolol-d₅ (Mixture of Diastereomers) is the deuterium labeled α-Hydroxy Metoprolol Mixture of Diastereomers .

HY-118714S

α-Hydroxy alprazolam-d5
α-Hydroxy alprazolam-d₅ (U 40125-d₅; alpha-Hydroxyalprazolam-d₅) is the deuterium labled α-hydroxy alprazolam (HY-118714).

HY-132676S

*Ramiprilat-d5 (Mixture* of Diastereomers)**
Ramiprilat-d₅ (Mixture of Diastereomers) is the deuterium labeled Ramiprilat (Mixture of Diastereomers) .

HY-A0115S

*Ramiprilat-d3 (Mixture* of Diastereomers)**
Ramiprilat-d₃ (Mixture of Diastereomers) is the deuterium labeled Ramiprilat (Mixture of Diastereomers) .

HY-W777700

*Cuscohygrine-d6 (mixture* of diastereomers)**
Cuscohygrine-d₆ (mixture of diastereomers) is the deuterium labeled Cuscohygrine (Mixture of Diastereomers) (HY-N9904).

HY-W654395

*Methyl jasmonate-d5 (mixture* of diastereomers)**
Methyl jasmonate-d₅ (mixture of diastereomers) is deuterium labeled Methyl (Z)-2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate .

HY-132706S

*N-Deformyl Formoterol-d6 Fumarate (Mixture* of Diastereomers)**
N-Deformyl Formoterol-d₆ Fumarate (Mixture of Diastereomers) is the deuterium labeled N-Deformyl Formoterol Fumarate (Mixture of Diastereomers) .

HY-W766409

*Ciclesonide-d11 (Mixture* of Diastereomers)**
Ciclesonide-d₁₁ (Mixture of Diastereomers) is the deuterium labeled Ciclesonide.

HY-W768541

*Idarubicinol-d4 (Mixture* of Diastereomers)**
Idarubicinol-d₄ (Mixture of Diastereomers) is the deuterium labeled Idarubicinol.

HY-W744273

*Pravastatin-d9 Sodium (mixture* of 2 diastereomers)**
Pravastatin-d₉ Sodium (mixture of 2 diastereomers) is the deuterium labeled Pravastatin Sodium.

HY-12650S

*Mirogabalin-13C2,d1 (Mixture* of Diastereomers)**
Mirogabalin-13C2,d1 (Mixture of Diastereomers) is a C13 and deuterium labeled Mirogabalin. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS .

HY-132379S

Hydroxy Pioglitazone-d5 (M-IV) (Mixture of-diastereomers)
Hydroxy Pioglitazone-d₅ (M-IV) (Mixture of-diastereomers) is the deuterium labeled Hydroxy Pioglitazone (M-IV) (Mixture of-diastereomers) .

HY-W711709

*Terameprocol-d12 (Mixture* of Diastereomers)**
Terameprocol-d₁₂ (Mixture of Diastereomers) is the deuterium labeled 4,4'-(2,3-Dimethylbutane-1,4-diyl)bis(1,2-dimethoxybenzene) (HY-W422348).

HY-W777284

*Zeranol-d5 (mixture* of diastereomers)**
Zeranol-d₅ (mixture of diastereomers) is the deuterium labeled Zeranol (HY-N6709). Zeranol, a metabolite of the mycoestrogen zearalenone, is an estrogen receptor agonist. Zeranol is used as a growth promoter of livestock due to its strong estrogenic activity .

HY-W654209

*Glycopyrrolate iodide-d3 (mixture* of diastereomers)**
Glycopyrrolate iodide-d₃ (mixture of diastereomers) is deuterium labeled 3-(2-Cyclopentyl-2-hydroxy-2-phenylacetoxy)-1,1-dimethylpyrrolidin-1-ium iodide .

HY-113026S

*(2RS,4R,8R)-δ-Tocopherol-d4 (Mixture* of Diastereomers)**
(2RS,4R,8R)-δ-Tocopherol-d₄ (Mixture of Diastereomers) is the deuterium labeled (2RS,4R,8R)-δ-Tocopherol (Mixture of Diastereomers) .

HY-W100026S

*Galaxolide-d6 (mixture* of diastereomers) (>80%)**
Galaxolide-d₆ (mixture of diastereomers) (>80%) is the deuterium labeled Galaxolide (HY-W100026). Galaxolide can induce estrogenic activity (Estrogen Receptor/ERR), trigger oxidative stress and genotoxicity, and induce EROD and GST (Glutathione S-transferase) enzyme activity .

HY-152040S

*Tenuazonic acid-(acetyl-13C2) (mixture* of diastereomers) in methanol**
Tenuazonic acid-(acetyl- ¹³C₂) (mixture of diastereomers) in methanol (3-(Acetyl- ¹³C₂)-5-((S)-sec-butyl)-4-hydroxy-1,5-dihydro-2H-pyrrol-2-one) is ¹³C labeled Tenuazonic acid-(acetyl) (mixture of diastereomers) in methanol .

HY-150857S

*Thymine-α,α,α,6-d4 Glycol (mixture* of diastereomers)-d4**
Thymine-α,α,α,6-d₄ Glycol (mixture of diastereomers)-d₄ is the deuterium labeled Thymine-α,α,α,6-d4 Glycol (mixture of diastereomers) .

HY-17503S

Metoprolol-d7
Metoprolol-d₇ is the deuterium labeled Metoprolol. Metoprolol (Toprol) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension[1][2].

HY-17503S3

Metoprolol-d5
Metoprolol-d₅ is the deuterium labeled Metoprolol . Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-17503AS

Metoprolol-d7 hydrochloride
Metoprolol-d₇ (hydrochloride) is the deuterium labeled Metoprolol. Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-132382S

*β-Sitosterol-d7 (mixture* of diasteromers)**
β-Sitosterol-d₇ (Mixture of Diastereomers) is the deuterium labeled β-Sitosterol (mixture of diasteromers) .

HY-17503BS

Metoprolol-d6 tartrate
Metoprolol-d₆ (tartrate) is the deuterium labeled Metoprolol tartrate. Metoprolol is an orally active, selective β1-adrenoceptor antagonist. Metoprolol shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-17503AS1

Metoprolol-d6 succinate
Metoprolol-d₆ (succinate) is deuterium labeled Metoprolol (succinate). Metoprolol succinate is an orally active, selective β1-adrenoceptor antagonist. Metoprolol succinate shows anti-inflammation, antitumor and anti-angiogenic properties .

HY-W740664

20α-Hydroxy Cholesterol-d7
20α-Hydroxy Cholesterol-d₇ is the deuterium labeled 20α-Hydroxy Cholesterol.

HY-W740771

6α-Hydroxy cortisol-d4
6α-Hydroxy cortisol-d₄ is the deuterium labeled 6α-Hydroxy cortisol.

HY-125348S

6α-Hydroxy Paclitaxel-d5

6α-Hydroxy Paclitaxel-d₅ is the deuterium labeled 6α-Hydroxy paclitaxel. 6α-Hydroxy paclitaxel is a primary metabolite of Paclitaxel. 6α-Hydroxy paclitaxel retains a time-dependent effect on organic anion-transporting polypeptides 1B1/SLCO1B1 (OATP1B1) with similar inhibition potency to Paclitaxel, whereas it no longer showed time-dependent inhibition of OATP1B3. 6α-Hydroxy paclitaxel can be used for the research of cancer .

HY-133966S

6α-Hydroxy-5α-cholestane-d7
6α-Hydroxy-5α-cholestane-d₇ is deuterium labeled 6α-Hydroxy-5α-cholestane.

HY-113031S1

16α-Hydroxydehydroepiandrosterone-d5
16α-Hydroxydehydroepiandrosterone-d₅ (16α-Hydroxy-DHEA-d₅) is the deuterium labeled 16α-Hydroxydehydroepiandrosterone (HY-113031) .

HY-146773S

7α-Hydroxy-3-oxocholest-4-enoic acid-d3
7α-Hydroxy-3-oxocholest-4-enoic acid-d₃ is deuterium labeled 7α-Hydroxy-3-oxocholest-4-enoic acid.

HY-10844S1

Pretomanid-d5
Pretomanid-d₅ is deuterated labeled Pretomanid (HY-10844). Pretomanid (PA-824) is an antibiotic used for the research of multi-drug-resistant tuberculosis affecting the lungs. Pretomanid exhibits a sub-micromolar MIC against M. tuberculosis (MTB). The MIC values of PA-824 against a panel of MTB pan-sensitive and Rifampin mono-resistant clinical isolates range from 0.015 to 0.25 μg/mL.

HY-113259S

7α-Hydroxy-4-cholesten-3-one-d7

7α-Hydroxy-4-cholesten-3-one-d₇ is the deuterium labeled 7α-Hydroxy-4-cholesten-3-one. 7α-Hydroxy-4-cholesten-3-one is an intermediate in synthesis of bile acids from cholesterol. 7α-Hydroxy-4-cholesten-3-one is a pregnane X receptor (PXR) agonist. 7α-Hydroxy-cholest-4-en-3-one is a biomarker for bile acid loss, irritable bowel syndrome, and other diseases associated with defective bile acid biosynthesis. 7α-Hydroxy-cholest-4-en-3-one is the physiological substrate for CYP8B1 .

HY-113038AS

α-Hydroxyglutaric acid-13C5 disodium
α-Hydroxyglutaric acid- ¹³C₅ (sodium) is the ¹³C labeled α-Hydroxyglutaric acid sodium . α-Hydroxyglutaric acid (2-Hydroxyglutarate) sodium is an α-hydroxy acid form of glutaric acid. α-Hydroxyglutaric acid sodium is a competitive inhibitor of multiple α-ketoglutarate-dependent dioxygenases, including histone demethylases and the TET family of 5-methlycytosine (5mC) hydroxylases .

HY-17503S2

*(S)-Metoprolol-d7*
(S)-Metoprolol-d₇ is the deuterium labeled Metoprolol. Metoprolol (Toprol) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension[1][2].

HY-17503S1

*(R)-Metoprolol-d7*
(R)-Metoprolol-d₇ is the deuterium labeled Metoprolol. Metoprolol (Toprol) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension[1][2].

HY-113031S

16α-Hydroxydehydroepiandrosterone-d6
16α-Hydroxydehydroepiandrosterone-d₆ (16α-Hydroxy-DHEA-d₆) is the deuterium labeled 16α-Hydroxydehydroepiandrosterone .

HY-132485S

*N-Methyl Pantoprazole-d3 (Mixture* of 1 and 3 isomers)**
N-Methyl Pantoprazole-d₃ (Mixture of 1 and 3 isomers) is the deuterium labeled N-Methyl Pantoprazole (Mixture of 1 and 3 isomers) .

HY-132637S

*Chlorfenvinphos-d10(Mixture* of cis-trans isomers)**
Chlorfenvinphos-d₁₀(Mixture of cis-trans isomers) is the deuterium labeled Chlorfenvinphos (Mixture of cis-trans isomers) .

HY-113038AS1

α-Hydroxyglutaric acid-d4 disodium

α-Hydroxyglutaric acid-d₄ (disodium) is the deuterium labeled α-Hydroxyglutaric acid disodium . α-Hydroxyglutaric acid (2-Hydroxyglutarate) disodium is an α-hydroxy acid form of glutaric acid. α-Hydroxyglutaric acid disodium is a competitive inhibitor of multiple α-ketoglutarate-dependent dioxygenases, including histone demethylases and the TET family of 5-methlycytosine (5mC) hydroxylases .

HY-W018772S15

D-Ribose(mixture of isomers)-13C5

D-Ribose(mixture of isomers)- ¹³C₅ isomers)- ¹³C₅ is the ¹³C labeled D-Ribose(mixture of isomers) . D-Ribose(mixture of isomers) is an energy enhancer, and acts as a sugar moiety of ATP, and widely used as a metabolic therapy supplement for chronic fatigue syndrome or cardiac energy metabolism. D-Ribose(mixture of isomers) is active in protein glycation, induces NF-κB inflammation in a RAGE-dependent manner .

HY-W758414

*Phoxim-d5 (phenyl-d5) (mixture* of isomers)**
Phoxim-d₅ (phenyl-d₅) (mixture of isomers) is the deuterium labeled Phoxim (HY-B0819). Phoxim is an organic phosphorus pesticide and widely applies worldwide for agricultural purposes .

HY-W744215

*3-Hydroxy* tibolone-d5 (mixture of 3a & 3b isomers)**
3-Hydroxy tibolone-d₅ (mixture of 3a & 3b isomers) is the deuterium labeled 3-Hydroxy tibolone.

HY-B0172S1

Lithocholic acid-d5
Lithocholic acid-d₅ is deuterium labeled Lithocholic acid.

HY-W767484

Nicotinamide riboside-d4 (triflate)
Nicotinamide riboside-d₄ (triflate) (Nicotinamide riboside-d₄ triflate (d3-major)a/b mixture) is deuterium labeled Nicotinamide riboside (triflate) .

HY-W012481S

Nirvanol-d5
Nirvanol-d₅ (Ethylphenylhydantoin-d₅) is deuterium labeled Nirvanol (HY-W012481) . Nirvanol (Ethylphenylhydantoin) is a metabolite of Mephenytoin (HY-B1184) that exerts anticonvulsant effects in the maximal electroshock (M.E.S.) seizure model in mice. Nirvanol shows potential for research in epilepsy-related neurological disorders .

HY-141901S1

DHEA-d5

DHEA-d₅ (Prasterone-d₅; Dehydroisoandrosterone-d₅; Dehydroepiandrosterone-d₅) is the deuterium labeled DHEA (HY-14650). DHEA (Prasterone) is one of the most abundant steroid hormones. DHEA (Prasterone) mediates its action via multiple signaling pathways involving specific membrane receptors and via transformation into androgen and estrogen derivatives (e.g., androgens, estrogens, 7α and 7β DHEA, and 7α and 7β epiandrosterone derivatives) acting through their specific receptors.

HY-14198S

Selegiline-d5
Selegiline-d₅ (Deprenyl-d₅) is deuterium labeled Selegiline. Selegiline (Deprenyl) is a potent, selective and irreversible inhibitor of MAO-B, with an IC₅₀ of 51 nM. Selegiline exhibits 450-flod selectivity for MAO-B over MAO-A (IC₅₀=23 μM). Selegiline can be used for the research of Parkinson's disease, Alzheimer's disease and major depressive disorder .

HY-14199S

Selegiline-d5 hydrochloride

Selegiline-d₅ (hydrochloride) (Deprenyl-d₅ (hydrochloride)) is deuterium labeled Selegiline (hydrochloride). Selegiline (Deprenyl) hydrochloride is a potent, selective and irreversible inhibitor of MAO-B, with an IC₅₀ of 51 nM. Selegiline hydrochloride exhibits 450-flod selectivity for MAO-B over MAO-A (IC₅₀=23 μM). Selegiline hydrochloride can be used for the research of Parkinson's disease, Alzheimer's disease and major depressive disorder .

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