1. Signaling Pathways
  2. JAK/STAT Signaling
    Stem Cell/Wnt
  3. STAT
  4. STAT Inhibitors

STAT Inhibitors

STAT3

STAT5

STAT6

STAT1

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STAT Inducers, Degraders, Inhibitors, Agonists, Activators & Modulators
Product Name STAT3 STAT5 STAT6 STAT1 Purity
Stattic
STAT3
      99.58%
Cilengitide
STAT3 ([3])
      99.80%
Homoharringtonine
STAT3
      99.96%
AS1517499    
STAT6, IC50: 21 nM
  99.17%
Fulipiftide
STAT3
     
AG490
Stat-3
      99.86%
Artesunate
Stat-3
      99.89%
GYY4137
Stat-3
      98.08%
Niclosamide
STAT3, IC50: 0.25 μM (in HeLa cells)
      99.96%
Colivelin
STAT3
      99.92%
C188-9
STAT3, Kd: 4.7 nM
      99.84%
NSC 74859
STAT3, IC50: 86 μM
      98.35%
Ritlecitinib
STAT3
STAT5
STAT6
  99.80%
TPCA-1
STAT3
      99.66%
Astaxanthin
STAT3
      98.0%
Cryptotanshinone
STAT3, IC50: 4.6 μM
      98.80%
WP1066
STAT3
      99.77%
Scutellarin
STAT3
      99.04%
Napabucasin
STAT3
      99.94%
Butyzamide
STAT3
STAT5
    99.83%
STAT5-IN-1  
STAT5β, IC50: 47 μM
    98.35%
Pimozide
STAT3
STAT5
    99.91%
SD-36
STAT3, Kd: 50 nM
      99.73%
Diosgenin
STAT3
      99.92%
Colivelin TFA
STAT3
      99.52%
AC-4-130  
STAT5
    99.93%
Saikosaponin D
STAT3
      99.78%
AK-1690    
STAT6, DC50: 1 nM
  99.91%
AS2863619  
STAT5
    99.94%
Morusin
STAT3
      99.94%
Cucurbitacin I
STAT3
      99.56%
SH-4-54
STAT3, Kd: 300 nM
STAT5, Kd: 464 nM
    99.80%
AK-2292  
STAT5, DC50: 0.10 μM
    99.73%
SC-43
p-STAT3
      99.01%
SI-109
STAT3, Ki: 9 nM
      99.91%
BP-1-102
STAT3, IC50: 6.8 μM
      99.52%
Alantolactone
STAT3
      99.94%
Nifuroxazide
STAT3
      99.90%
YM-341619    
STAT6, IC50: 0.70 nM
  98.01%
Erasin
STAT3, IC50: 9.7 μM
   
STAT1, IC50: 24 μM
AS1810722    
STAT6, IC50: 1.9 nM
  98.10%
1-Stearoyl-sn-glycero-3-phosphocholine
p-STAT3
      99.53%
ML115
Stat-3, EC50: 2 nM
      99.89%
STAT3-IN-1
Stat-3, IC50: 1.82 μM (in HT29 cells)
Stat-3, IC50: 2.14 μM (in MDA-MB 231 cells)
     
STAT6-IN-4    
STAT6, IC50: 0.34 μM
  99.77%
Brevilin A
STAT3, IC50: 10.6 μM
      99.86%
Atractylenolide II
p-STAT3
      99.94%
NSC-370284
STAT3
STAT5
    99.27%
Peramivir
STAT3
      99.94%
KT-333
STAT3
     
STAT6-IN-5    
STAT6, IC50: 0.24 μM
  99.88%
Flubendazole
STAT3
      99.05%
BD750  
STAT5
    99.02%
Stapokibart    
STAT6
  99.37%
HJC0152
STAT3
      99.75%
LLL12
p-STAT3
      99.45%
CAY10594
p-STAT3
      98.64%
Radotinib
STAT3
      99.19%
STAT3-IN-3
STAT3
      98.40%
Perindopril
STAT3
      99.56%
HO-3867
STAT3
      99.67%
JMS-053
STAT3
      98.0%
Broussonin E
STAT3
      98.11%
Stafib-1  
STAT5b, IC50: 154 nM
    ≥98.0%
Stafia-1  
STAT5a, Ki: 10.9 μM
STAT5a, IC50: 22.2 μM
    99.39%
STAT3-IN-25
STAT3
      99.36%
Anti-Mouse IL-6 Antibody (MP5-20F3)
STAT3
      99.20%
OSM-SMI-10B
p-STAT3
      99.70%
Garcinone D
p-STAT3
      99.88%
Picroside I    
STAT6
  99.48%
GMB-475  
STAT5
    98.69%
STX-0119
STAT3, IC50: 74 μM (STAT3 transcription)
      98.40%
Perindopril erbumine
STAT3
      99.98%
Ginkgolic acid C17:1
STAT3
      99.80%
IST5-002  
STAT5a, IC50: 1.5 μM
STAT5b, IC50: 3.5 μM
    99.83%
Serplulimab
p-STAT3
      99.30%
Anti-Mouse CD276/B7-H3 Antibody (MJ18)
p-STAT3
     
Cenisertib  
STAT5
    99.86%
Desmethoxyyangonin
STAT3
      99.46%
STAT5-IN-2  
STAT5, EC50: 9 μM (in K562 cells)
STAT5, EC50: 5 μM (in KU812 cells )
    99.08%
Anti-Mouse NK1.1 Antibody (PK136)
p-STAT3
   
STAT1
Telocinobufagin
STAT3
      99.93%
Garcinone C
Stat-3
      99.66%
Reticuline
STAT3
      98.91%
Corylifol A
STAT3, IC50: 0.81 μM
      99.90%
STAT3-IN-12
STAT3
      99.87%
UNC1062    
STAT6
  98.92%
Olokizumab
Stat-3
      99.54%
Phellodendrine chloride
STAT3
      99.79%
Mogrol
STAT3
      99.76%
inS3-54A18
STAT3
      99.93%
LL-K8-22      
STAT1
99.76%
AK-068    
STAT6
  99.57%
Protosappanin A
STAT3
      99.95%
YMU1
STAT3
      99.19%
Ochromycinone
STAT3
      98.29%
HODHBt  
STAT5
    99.93%
Triacetylresveratrol
STAT3
      99.11%
Tetramethylcurcumin
STAT3
      99.91%
AS2863619 free base  
STAT5
    99.87%
Cyanidin 3,5-diglucoside chloride
STAT3
      99.37%
STAT3-IN-15
STAT3
      98.99%
Golotimod hydrochloride
STAT3
      99.79%
STAT1/3-IN-1
STAT3
   
STAT1
Balsalazide
STAT3
      99.20%
ASP3026
STAT3
      99.88%
HJC0416 hydrochloride
STAT3
      98.68%
Equisetin
STAT3
      99.40%
SB02024      
STAT1
99.70%
Anti-Mouse CD106/VCAM-1 Antibody (M/K-2.7)
p-STAT3
     
PROTAC FLT-3 degrader 1  
STAT5
    99.74%
Ac-GpYLPQTV-NH2 acetate
STAT3, IC50: 0.33 μM
      99.38%
STAT3-IN-17
STAT3
      98.0%
Patiromer
STAT3
STAT5
STAT6
 
SC99
STAT3
      98.90%
Balsalazide sodium hydrate
STAT3
      99.61%
QL-1200186
STAT3
STAT5
 
STAT1
99.95%
Mulberrofuran G
STAT3
      99.84%
Zharp1-211      
STAT1
99.15%
OK2
p-STAT3
     
Graveoline
p-STAT3
      99.96%
WB436B
STAT3
      99.93%
Ritlecitinib tosylate
STAT3
STAT5
STAT6
  99.77%
Golotimod
STAT3
      98.04%
STAT3-IN-48
p-STAT3
      98.02%
Eflepedocokin alfa
STAT3
      ≥99.0%
SH5-07
STAT3, IC50: 3.9 μM
      ≥98.0%
MNK8
STAT3
      99.76%
SD-1029
STAT3
     
Vanicoside B
STAT3
      99.82%
WB518
STAT3
p-STAT3
     
APTSTAT3-9R
STAT3
      98.82%
ENMD-1198
STAT3
      98.87%
UC-514321
STAT3
STAT5
    98.0%
Phellodendrine
STAT3
      99.60%
Iminostilbene
STAT3
      99.34%
Momordicine I
STAT3
     
SD-436
STAT3, IC50: 19 nM
STAT5, IC50: >10 μM
STAT6, IC50: >10 μM
STAT1, IC50: 270 nM
98.27%
Pimozide-d4
STAT3
STAT5
    99.2%
ER-464195-01
STAT3
     
GSK2618960  
STAT5
   
STAT3-D11-PROTAC-VHL
STAT3
     
Galiellalactone
STAT3, IC50: 250-500 nM
     
Biflorin      
STAT1
99.54%
15(R)-Lipoxin A4    
STAT6
  98.3%
Stafia-1-dipivaloyloxymethyl ester  
STAT5a
   
Eupalinolide K
STAT3
      99.20%
Niclosamide monohydrate
STAT3, IC50: 0.25 μM (in HeLa cells)
     
SD-1008
STAT3
      99.10%
KT-333 ammonium
STAT3
      99.48%
Ritlecitinib (malonate)
STAT3
STAT5
STAT6
 
STAT3-IN-8
STAT3
     
KT-333 diammonium
STAT3
     
YSY01A
Stat-3
     
c-Met-IN-24
STAT3, IC50: 4.7 μM
     
STAT3-IN-37
STAT3
     
PROTAC STAT6 degrader-1    
STAT6, DC50: <1 nM
 
STAT3 HiBiT degrader 1
STAT3
     
STAT3-IN-38
STAT3, Kd: 45.33 μM
     
STAT3-IN-29
STAT3
     
VEGFR-2/STAT-3-IN-1
STAT3, IC50: 5.63 nM
     
8α-Tigloyloxyhirsutinolide 13-O-acetate
STAT3
     
KB-0118
STAT3
     
G721-0282
p-STAT3
     
WR-S-462
STAT3, Kd: 58 nM
     
JAK1/STAT3-IN-1
STAT3
     
FLT3-IN-28  
STAT5
   
CHI3L1-IN-4
p-STAT3
     
STAT6-IN-7    
STAT6
 
STAT3/AKT-IN-1
Stat-3
     
ROCK2-IN-7
Stat-3
     
Anti-inflammatory agent 92
STAT3
     
STAT3-IN-41
STAT3
     
(trans)-STAT6 modulator-5    
STAT6
 
Golotimod TFA
STAT3
     
HJC0416
STAT3
     
HJC0123
STAT3
     
JAK2-IN-13
STAT3
STAT5
   
STAT3-IN-46
STAT3, Kd: 323.3 nM
     
PROTAC JAK2 degrader-1
p-STAT3
STAT5
   
HAT-SIL-TG-1&AT
STAT3
STAT5
   
STAT3/NF-κB-IN-1
STAT3, IC50: 5.86 μM
     
SD-2301
STAT3
     
STAT3-IN-47
STAT3
     
STAT6-IN-8    
STAT6
 
7-epi-Isogarcinol
STAT3
     
STAT6-IN-9    
STAT6, EC50: 4 nM
 
STAT3-IN-44
STAT3
     
Cernuumolide J
Stat-3
     
Atractylenolide II (Standard)
p-STAT3
     
Antitumor agent-73
STAT3
     
STAT3-IN-5
p-STAT3, EC50: 170 nM
     
K882
Stat-3
     
STAT3-IN-32
STAT3
     
Hsp110-STAT3 PPI-IN-2
STAT3
     
STAT3-IN-43
STAT3, IC50: 40.7 μM
     
SD-91
STAT3, Ki: 5.5 nM
STAT3, Kd: 28 nM
     
VS1150  
STAT5
   
FLT3-IN-32 hydrochloride  
STAT5
   
Ac-GpYLPQTV-NH2
STAT3, IC50: 0.33 μM
     
Z169667518
STAT3
     
STAT3/CAIX-IN-1
STAT3, Kd: 60.03 μM
     
STAT3-IN-9
STAT3
     
PROTAC STAT3 degrader-2
STAT3, ID50: 3.54 μM
     
Ascochlorin
STAT3
     
NSC 850745
Stat-3, IC50: 670 nM
     
Tyk2-IN-22-d3  
STAT5
   
Betavulgarin
p-STAT3
     
1-Stearoyl-sn-glycero-3-phosphocholine-d35
p-STAT3
     
PROTAC c-Met degrader-5
p-STAT3
     
NW16
STAT3, Kd: 11.0 μM
     
MRC-G-001
STAT3
     
CDK6/9-IN-2
STAT3
     
pro-FTY
p-STAT3
     
JAK2-IN-14  
STAT5
   
Cyanidin 3,5-diglucoside chloride (Standard)
STAT3
     
Furowanin A
STAT3
     
IMC-EB10  
STAT5
   
Antitumor agent-195
STAT3, IC50: 0.52 μM
     
ALOX5 stabilizer-1
STAT3
     
STAT-3/c-Src-IN-1
STAT3, IC50: 0.844 μM
     
STAT3-IN-10
STAT3, IC50: 5.18 μM
     
Balsalazide disodium
STAT3
     
GYY4137 (GMP)
Stat-3
     
CHMFL-48  
STAT5
   
DETD-35
Stat-3
     
STAT3-IN-39
STAT3
     
TM-233
Stat-3
     
BP-1-108  
STAT5, Ki: 8.3 μM
   
PMMB-187
Stat-3, IC50: 1.81 μM