1. Signaling Pathways
  2. JAK/STAT Signaling
    Stem Cell/Wnt
  3. STAT
  4. STAT Inhibitors

STAT Inhibitors

STAT3

STAT5

STAT6

STAT1

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

STAT Degraders, Inducers, Inhibitors, Agonists & Activators
Product Name STAT3 STAT5 STAT6 STAT1 Purity
Stattic
STAT3
      99.58%
Cilengitide
STAT3 ([3])
      99.80%
Homoharringtonine
STAT3
      99.96%
AS1517499    
STAT6, IC50: 21 nM
  99.17%
STAT3-D11-PROTAC-VHL
STAT3
     
AG490
Stat-3
      99.86%
Artesunate
Stat-3
      99.89%
Niclosamide
STAT3, IC50: 0.25 μM (in HeLa cells)
      99.91%
GYY4137
Stat-3
      98.08%
Colivelin
STAT3
      99.27%
C188-9
STAT3, Kd: 4.7 nM
      99.84%
Ritlecitinib
STAT3
STAT5
STAT6
  99.80%
NSC 74859
STAT3, IC50: 86 μM
      98.35%
TPCA-1
STAT3
      99.66%
Astaxanthin
STAT3
      ≥98.0%
WP1066
STAT3
      99.77%
Scutellarin
STAT3
      99.04%
Cryptotanshinone
STAT3, IC50: 4.6 μM
      98.80%
Napabucasin
STAT3
      99.94%
Butyzamide
STAT3
STAT5
    99.62%
STAT5-IN-1  
STAT5β, IC50: 47 μM
    98.35%
Pimozide
STAT3
STAT5
    99.91%
SD-36
STAT3, Kd: 50 nM
      99.73%
Diosgenin
STAT3
      99.92%
Colivelin TFA
STAT3
      99.52%
AC-4-130  
STAT5
    99.93%
Saikosaponin D
STAT3
      98.76%
SH-4-54
STAT3, Kd: 300 nM
STAT5, Kd: 464 nM
    99.80%
Morusin
STAT3
      99.94%
AS2863619  
STAT5
    99.94%
Cucurbitacin I
STAT3
      99.44%
SI-109
STAT3, Ki: 9 nM
      99.91%
AK-1690    
STAT6, DC50: 1 nM
  99.91%
SC-43
p-STAT3
      99.01%
BP-1-102
STAT3, IC50: 6.8 μM
      99.52%
AK-2292  
STAT5, DC50: 0.10 μM
    99.73%
Alantolactone
STAT3
      99.94%
Erasin
STAT3, IC50: 9.7 μM
   
STAT1, IC50: 24 μM
YM-341619    
STAT6, IC50: 0.70 nM
  98.01%
Nifuroxazide
STAT3
      99.90%
1-Stearoyl-sn-glycero-3-phosphocholine
p-STAT3
      99.53%
AS1810722    
STAT6, IC50: 1.9 nM
  98.10%
NSC-370284
STAT3
STAT5
    99.27%
Peramivir
STAT3
      99.94%
STAT3-IN-1
Stat-3, IC50: 1.82 μM (in HT29 cells)
Stat-3, IC50: 2.14 μM (in MDA-MB 231 cells)
     
Brevilin A
STAT3, IC50: 10.6 μM
      99.86%
ML115
Stat-3, EC50: 2 nM
      99.89%
STAT6-IN-4    
STAT6, IC50: 0.34 μM
  99.77%
Atractylenolide II
p-STAT3
      99.94%
Flubendazole
STAT3
      99.05%
HJC0152
STAT3
      99.75%
CAY10594
p-STAT3
      98.64%
Stafia-1  
STAT5a, Ki: 10.9 μM
STAT5a, IC50: 22.2 μM
    99.39%
KT-333
STAT3
     
STAT3-IN-3
STAT3
      98.40%
STAT6-IN-5    
STAT6, IC50: 0.24 μM
  99.88%
Radotinib
STAT3
      99.19%
BD750  
STAT5
    99.02%
LLL12
p-STAT3
      99.45%
Broussonin E
STAT3
      98.11%
Stafib-1  
STAT5b, IC50: 154 nM
    ≥98.0%
HO-3867
STAT3
      99.67%
STAT3-IN-25
STAT3
      99.36%
Anti-Mouse IL-6 Antibody (MP5-20F3)
STAT3
      99.20%
Perindopril erbumine
STAT3
      99.98%
Picroside I    
STAT6
  99.48%
Perindopril
STAT3
      98.11%
Garcinone D
p-STAT3
      99.88%
IST5-002  
STAT5a, IC50: 1.5 μM
STAT5b, IC50: 3.5 μM
    99.83%
STX-0119
STAT3, IC50: 74 μM (STAT3 transcription)
     
OSM-SMI-10B
p-STAT3
      99.70%
Ginkgolic acid C17:1
STAT3
      99.80%
GMB-475  
STAT5
    98.69%
Serplulimab
p-STAT3
      99.30%
Corylifol A
STAT3, IC50: 0.81 μM
      99.90%
Cenisertib  
STAT5
    99.86%
Garcinone C
Stat-3
      99.66%
Phellodendrine chloride
STAT3
      99.79%
Telocinobufagin
STAT3
      99.93%
Desmethoxyyangonin
STAT3
      99.46%
STAT5-IN-2  
STAT5, EC50: 9 μM (in K562 cells)
STAT5, EC50: 5 μM (in KU812 cells )
    99.08%
Reticuline
STAT3
      98.91%
Anti-Mouse CD276/B7-H3 Antibody (MJ18)
p-STAT3
     
Mogrol
STAT3
      99.76%
UNC1062    
STAT6
  98.92%
inS3-54A18
STAT3
      99.93%
Anti-Mouse NK1.1 Antibody (PK136)
p-STAT3
   
STAT1
Triacetylresveratrol
STAT3
      99.11%
Protosappanin A
STAT3
      99.95%
Olokizumab
Stat-3
     
STAT3-IN-12
STAT3
      99.87%
LL-K8-22      
STAT1
99.76%
Ochromycinone
STAT3
      98.29%
Tetramethylcurcumin
STAT3
      99.91%
YMU1
STAT3
      99.19%
Golotimod hydrochloride
STAT3
      99.79%
AK-068    
STAT6
  99.57%
HODHBt  
STAT5
    99.93%
AS2863619 free base  
STAT5
    99.87%
ASP3026
STAT3
      99.88%
HJC0416 hydrochloride
STAT3
      98.68%
STAT3-IN-15
STAT3
      98.99%
Balsalazide
STAT3
      99.20%
Anti-Mouse CD106/VCAM-1 Antibody (M/K-2.7)
p-STAT3
     
STAT3-IN-17
STAT3
      ≥98.0%
Patiromer
STAT3
STAT5
STAT6
 
SC99
STAT3
      98.90%
Equisetin
STAT3
      99.40%
SB02024      
STAT1
99.70%
PROTAC FLT-3 degrader 1  
STAT5
    99.74%
QL-1200186
STAT3
STAT5
 
STAT1
99.95%
Mulberrofuran G
STAT3
      99.84%
OK2
p-STAT3
     
Graveoline
p-STAT3
      99.96%
WB436B
STAT3
      99.93%
STAT1/3-IN-1
STAT3
   
STAT1
Zharp1-211      
STAT1
99.15%
Golotimod
STAT3
      98.04%
APTSTAT3-9R
STAT3
      98.82%
UC-514321
STAT3
STAT5
    ≥98.0%
1-(4-Chloro-3-(trifluoromethyl)phenyl)-3-(4-(4-cyanophenoxy)phenyl)urea
p-STAT3
      98.02%
Balsalazide sodium hydrate
STAT3
      99.61%
Eflepedocokin alfa
STAT3
      ≥99.0%
MNK8
STAT3
      99.76%
SD-1029
STAT3
     
Vanicoside B
STAT3
      99.82%
Iminostilbene
STAT3
      99.34%
Ac-GpYLPQTV-NH2 acetate
STAT3, IC50: 0.33 μM
      99.38%
Ritlecitinib tosylate
STAT3
STAT5
STAT6
  99.77%
Phellodendrine
STAT3
      99.60%
ENMD-1198
STAT3
      98.87%
Momordicine I
STAT3
     
SH5-07
STAT3, IC50: 3.9 μM
      ≥98.0%
Syk-IN-6
STAT3
STAT5
   
Pimozide-d4
STAT3
STAT5
    99.2%
Galiellalactone
STAT3, IC50: 250-500 nM
     
WB518
STAT3
p-STAT3
     
Fulipiftide
STAT3
     
Biflorin      
STAT1
99.54%
15(R)-Lipoxin A4    
STAT6
  98.3%
Stafia-1-dipivaloyloxymethyl ester  
STAT5a
   
Eupalinolide K
STAT3
      99.20%
Niclosamide monohydrate
STAT3, IC50: 0.25 μM (in HeLa cells)
     
SD-1008
STAT3
      99.10%
KT-333 ammonium
STAT3
      99.48%
Ritlecitinib (malonate)
STAT3
STAT5
STAT6
 
STAT3-IN-8
STAT3
     
KT-333 diammonium
STAT3
     
YSY01A
Stat-3
     
c-Met-IN-24
STAT3, IC50: 4.7 μM
     
STAT3-IN-37
STAT3
     
STAT3 HiBiT degrader 1
STAT3
     
STAT3-IN-38
STAT3, Kd: 45.33 μM
     
STAT3-IN-29
STAT3
     
VEGFR-2/STAT-3-IN-1
STAT3, IC50: 5.63 nM
     
8α-Tigloyloxyhirsutinolide 13-O-acetate
STAT3
     
KB-0118
STAT3
     
G721-0282
p-STAT3
     
WR-S-462
STAT3, Kd: 58 nM
     
JAK1/STAT3-IN-1
STAT3
     
FLT3-IN-28  
STAT5
   
SD-436
STAT3, IC50: 19 nM
STAT5, IC50: >10 μM
STAT6, IC50: >10 μM
STAT1, IC50: 270 nM
STAT6-IN-7    
STAT6
 
STAT3/AKT-IN-1
Stat-3
     
ROCK2-IN-7
Stat-3
     
Anti-inflammatory agent 92
STAT3
     
STAT3-IN-41
STAT3
     
Golotimod TFA
STAT3
     
HJC0416
STAT3
     
HJC0123
STAT3
     
JAK2-IN-13
STAT3
STAT5
   
PROTAC JAK2 degrader-1
p-STAT3
STAT5
   
HAT-SIL-TG-1&AT
STAT3
STAT5
   
STAT3/NF-κB-IN-1
STAT3, IC50: 5.86 μM
     
GSK2618960  
STAT5
   
7-epi-Isogarcinol
STAT3
     
STAT3-IN-44
STAT3
     
Cernuumolide J
Stat-3
     
Atractylenolide II (Standard)
p-STAT3
     
Antitumor agent-73
STAT3
     
STAT3-IN-5
p-STAT3, EC50: 170 nM
     
K882
Stat-3
     
STAT3-IN-32
STAT3
     
Hsp110-STAT3 PPI-IN-2
STAT3
     
STAT3-IN-43
STAT3, IC50: 40.7 μM
     
SD-91
STAT3, Ki: 5.5 nM
STAT3, Kd: 28 nM
     
VS1150  
STAT5
   
FLT3-IN-32 hydrochloride  
STAT5
   
Ac-GpYLPQTV-NH2
STAT3, IC50: 0.33 μM
     
Z169667518
STAT3
     
STAT3/CAIX-IN-1
STAT3, Kd: 60.03 μM
     
STAT3-IN-9
STAT3
     
PROTAC STAT3 degrader-2
STAT3, ID50: 3.54 μM
     
Ascochlorin
STAT3
     
Tyk2-IN-22-d3  
STAT5
   
Betavulgarin
p-STAT3
     
1-Stearoyl-sn-glycero-3-phosphocholine-d35
p-STAT3
     
PROTAC c-Met degrader-5
p-STAT3
     
NW16
STAT3, Kd: 11.0 μM
     
MRC-G-001
STAT3
     
CDK6/9-IN-2
STAT3
     
pro-FTY
p-STAT3
     
Furowanin A
STAT3
     
IMC-EB10  
STAT5
   
Antitumor agent-195
STAT3, IC50: 0.52 μM
     
STAT-3/c-Src-IN-1
STAT3, IC50: 0.844 μM
     
STAT3-IN-10
STAT3, IC50: 5.18 μM
     
Balsalazide disodium
STAT3
     
GYY4137 (GMP)
Stat-3
     
CHMFL-48  
STAT5
   
DETD-35
Stat-3
     
STAT3-IN-39
STAT3
     
TM-233
Stat-3
     
BP-1-108  
STAT5, Ki: 8.3 μM
   
PMMB-187
Stat-3, IC50: 1.81 μM