1. Signaling Pathways
  2. NF-κB
  3. NF-κB
  4. NF-κB Inhibitors

NF-κB Inhibitors

NF-κB

NF-κB1/p50

RelA/p65

RelB

c-Rel

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

NF-κB Degraders, Inhibitors, Agonists, Activators & Modulators
Product Name NF-κB NF-κB1/p50 RelA/p65 RelB c-Rel Purity
Phorbol 12-myristate 13-acetate
NF-κB
        99.80%
BAY 11-7082
NF-κB
        99.98%
JSH-23
NF-κB, IC50: 7.1 μM (in RAW 264.7 cells)
        99.92%
Shikonin
NF-κB
        99.80%
Baicalin
NF-κB
        98.92%
5-Aminosalicylic Acid    
p65
    99.97%
Sulfasalazine    
RelA
    99.04%
Dihydroartemisinin    
RelA
    99.03%
Pyrrolidinedithiocarbamate ammonium
NF-κB
        ≥98.0%
Parthenolide
NF-κB
        99.91%
TNF-α (31-45), human
NF-κB
        99.66%
SC75741    
p65, IC50: 200 nM
    99.51%
Andrographolide  
p50
      99.74%
Betulinic acid
NF-κB
        99.06%
BAY 11-7085
NF-κB
        99.99%
Ginsenoside Rg1    
p65
    99.91%
20(S)-Ginsenoside Rg3    
p65
    99.65%
NF-κΒ activator 1
NF-κB, EC50: 0.9 μM
        99.59%
CBL0137 hydrochloride
NF-κB, IC50: 0.47 μM
        99.72%
Withaferin A
NFκB
        99.92%
Ginsenoside Rb1    
p65
    99.28%
Diprovocim
NF-κB
        98.82%
Nafamostat mesylate
I-kappaBalpha
        99.85%
QNZ
NF-κB, IC50: 11 nM (in human Jurkat cells transfected with pNFκB-Luc)
        99.50%
Lidocaine
NF-κB
        99.96%
Fibrinogen (Bovine)  
p50
p65
 
c-Rel
(-)-DHMEQ    
RelA
RelB
  99.81%
Indole-3-carbinol
NF-κB
        98.87%
SN50
NF-κB
        99.66%
Berbamine
NF-κB
        99.59%
Maslinic acid    
p65
    ≥98.0%
Caffeic acid phenethyl ester
NF-κB
        99.85%
Saikosaponin D
NF-κB
        98.76%
Mangiferin  
p50
p65
    99.79%
Astragalin    
p65
    99.94%
MnTBAP chloride
NFκB
        ≥98.0%
α-Lipoic Acid
NF-κB
        99.86%
Forsythoside B
NF-κB
        99.99%
Astilbin
NF-κB
        99.97%
Morusin    
p65
    99.94%
18α-Glycyrrhetinic acid
NF-κB
        99.87%
Isovitexin
NF-κB
        99.77%
Muscone
NF-κB
        ≥98.0%
Vanillic acid    
p65
    99.75%
Tomatidine    
p65
    ≥98.0%
Neferine    
p65
    99.92%
Neochlorogenic acid    
p65
    99.77%
Ginsenoside Re
NF-κB
        99.22%
Sinomenine hydrochloride
NF-κB
        99.89%
Stachydrine    
p65
    ≥98.0%
DCZ0415
NF-κB
        99.81%
Guaiacol
NF-κB
        99.95%
Rhoifolin
NF-κB
        99.25%
Nimbolide
NF-κB
        99.79%
Lidocaine hydrochloride
NF-κB
        99.84%
(±)-Naringenin
NF-κB
        98.88%
Berbamine dihydrochloride
NF-κB
       
Ginsenoside Rd
NF-κB, IC50: 12.05 μM (in HepG2 cells)
        99.88%
NF-κΒ activator 2
NF-κB, EC50: 1.58 μM
        99.76%
EUK-134
NF-κB
        98.27%
Okanin    
p65
    99.98%
Stachydrine hydrochloride    
p65
    ≥98.0%
Peiminine    
p65
    99.94%
Peimine
NFκB
        99.43%
Ginsenoside Rg5    
p65
    99.87%
Schisantherin A    
p65
    99.87%
(R)-Sulforaphane
NF-κB
        99.48%
Chymostatin
NF-κB
        ≥99.0%
Homoplantaginin    
p65
    99.90%
Ethyl Caffeate
NF-κB
        99.34%
Sarsasapogenin
NF-κB
        99.91%
Licochalcone D    
p65
    99.81%
Sciadopitysin
NF-κB
        ≥99.0%
Lidocaine (Standard)
NF-κB
        99.85%
Cafestol
NF-κB
        99.91%
Engeletin
NF-κB
        99.88%
Cynaropicrin
NF-κB
        99.79%
Ophiopogonin D
NF-κB
        99.80%
CHPG sodium salt
NF-κB
        99.25%
Oxaprozin
NF-κB
        99.94%
Ginsenoside Rg2
NF-κB
        98.11%
Tectochrysin  
p50
p65
    99.88%
Yangonin    
RelA
    99.79%
NF-κB/MAPK-IN-1
NF-κB
        98.71%
Hesperidin methylchalcone
NF-κB
        ≥98.0%
IT-901
NF-κB, IC50: 0.1 μM
     
c-Rel, IC50: 3 μM
99.32%
11-​Keto-​beta-​boswellic acid
NF-κB
        99.96%
Dendrophenol
NF-κB
        99.93%
Laquinimod
NF-κB
        99.46%
CDDO-dhTFEA
NF-κB
        99.71%
Tomatidine hydrochloride    
p65
    99.58%
Deoxyelephantopin
NF-κB
        99.87%
Triacetylresveratrol
NF-κB
        99.11%
Ginsenoside Rb3
NF-κB, IC50: 8.2 μM (in 293T cell lines)
        99.47%
4-O-Methyl honokiol
NF-κB
        98.18%
Myrcene
NF-κB
       
Naringin Dihydrochalcone
NF-κB
        99.53%
L6H21
NF-κB
        99.19%
Cornuside
NF-κB
        99.99%
CHPG
NF-κB
        99.51%
Aconine
NF-κB
        99.78%
Isoliquiritin apioside
NF-κB
        99.87%
Anti-Mouse NK1.1 Antibody (PK136)
NF-κB
       
Reticuline
NF-κB
        98.91%
Sanggenon C
NF-κB
        98.46%
Armepavine    
p65
    99.53%
Lidocaine hydrochloride hydrate
NF-κB
        99.90%
Sauchinone
I-kappaBalpha
 
p65
    99.88%
SM-7368
NF-κB
        99.77%
Anti-Mouse RANKL/CD254 Antibody (IK22/5)
NF-κB
       
Obtusifolin
NF-κB
        99.91%
AT-533
NF-κB
        98.38%
Barlerin
NF-κB
        99.82%
2,5-Dihydroxyacetophenone
NF-κB
        99.89%
Inulicin
NF-κB
        99.94%
Tenuigenin
NF-κB
        99.24%
JAK-IN-23
NF-κB, IC50: 150.7 nM
        98.90%
(R)-(-)-Ibuprofen
NF-κB
        99.96%
Regaloside A    
p65
    99.64%
14-Deoxy-11,12-didehydroandrographolide
NF-κB
        98.63%
Ergolide
NF-κB
        99.75%
Cyclo(his-pro) TFA
NF-κB
        99.13%
Chelidonic acid
NF-κB
        99.91%
Polygalasaponin F
NF-κB
        99.85%
α-Lipoic Acid sodium
NF-κB
        99.92%
Erdosteine
NF-κB
        99.54%
Aurantiamide
NF-κB
        98.09%
Penehyclidine hydrochloride
NF-κB
        99.2%
Methylthiouracil
NF-κB
        ≥98.0%
Ginsenoside Rg6
NF-κB, IC50: 29.34 μM (in HepG2 cell)
NF-κB, IC50: 25.12 μM (in SK-Hep1 cell)
        99.13%
Ginsenoside Rk3
NF-κB, IC50: 14.24 μM (in HepG2 cells)
NF-κB, IC50: 15.32 μM (in SK-Hep1 cell)
        99.79%
Enniatin B1
NF-κB
        99.34%
Fosfenopril
NF-κB
        99.85%
Adelmidrol
NF-κB
        ≥98.0%
8-Deoxygartanin    
p65, IC50: 11.3 μM
    99.24%
Rubiadin-1-methyl ether    
p65
    98.57%
CID-2858522
NF-κB, IC50: 70 nM
        99.78%
Flaconitine
NF-κB
        99.77%
Anti-inflammatory agent 35
I-kappaBalpha
NF-κB
 
p65
    99.77%
DPLG3  
p50
p65
    99.18%
TML-6
NF-κB
        99.01%
Phellodendrine
NF-κB
        99.60%
α-Lipoic Acid (Standard)
NF-κB
        99.90%
TNF-α (31-45), human TFA
NF-κB
       
Echinulin
NF-κB
        98.63%
Nafamostat
I-kappaBalpha
       
Coelonin
NF-κB
        ≥98.0%
Salicortin
NF-κB
       
R-HP210
NF-κB
        98.21%
Cyclo(his-pro)
NF-κB
        98.76%
Sanggenon A
NF-κB
       
Anemarsaponin B    
p65
   
Ginsenoside Rb1 (Standard)    
p65
   
Nafamostat hydrochloride
I-kappaBalpha
       
WAY-204688
NF-κB
        99.89%
Laquinimod sodium
NF-κB
       
Penehyclidine
NF-κB
       
Mumefural
NF-κB
       
IMD-biphenylC
NF-κB
       
NF-κB-IN-3
NF-κB, IC50: 0.70 μM
       
JP-163-16    
p65
   
Verproside
NF-κB
       
Ginsenoside Rb3 (Standard)
NF-κB
       
G721-0282
NF-κB
       
MMH-165-26    
p65
   
NF-κB degrader 1  
p50
     
Ginsenoside Rd (Standard)
NF-κB
       
Eudebeiolide B
NF-κB
       
Ginsenoside Re (Standard)
NF-κB
       
Oxaprozin potassium
NF-κB
       
IMD-catechol
NF-κB
       
Sootepin D
NF-κB
       
NF-κB-IN-14
NF-κB
       
PROTAC STING degrader-4
NF-κB
       
Lucidone
NF-κB
p50
p65
   
IMD-biphenylB
NF-κB
       
Aurothiomalate disodium
NF-κB
       
Anti-inflammatory agent 20
NF-κB
       
Coronalolic acid
NF-κB
       
Ginsenoside Rg2 (Standard)
NF-κB
       
MR2938
NF-κB
       
Xanthine oxidase-IN-6
NF-κB
       
20(S)-Ginsenoside Rg3 (Standard)    
p65
   
NLRP3-IN-32    
p65
   
Mesalamine impurity P
NF-κB
       
Triphala
NF-κB
       
Ginsenoside Rg1 (Standard)    
p65
   
MOR-106
NF-κB
       
Cudraflavone B
NF-κB
       
DHMEQ racemate
NF-κB
       
NF-κB-IN-13
NF-κB
       
Icariside F2
NF-κB, IC50: 16.25 μM