1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    Metabolic Enzyme/Protease
  3. HSP
  4. HSP Inhibitors

HSP Inhibitors

HSP40

HSP70

HSP90

HSP105

HSF1

HSP

HSPA5

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

HSP Pre-designed Sets, Inducers, Inhibitors, Antagonists & Activators
Product Name HSP40 HSP70 HSP90 HSP105 HSF1 HSP HSPA5 Purity
Tamoxifen    
HSP90
        99.96%
Polyinosinic-polycytidylic acid  
HSP70
          99.40%
Tanespimycin    
HSP90, IC50: 5 nM
        99.01%
VER-155008  
HSP70, IC50: 0.5 μM
HSC70, IC50: 2.6 μM
Grp78, IC50: 2.6 μM
          99.91%
Tamoxifen Citrate    
HSP90
        99.88%
Geldanamycin    
HSP90, Kd: 1.2 μM
        99.78%
Ganetespib    
HSP90
        99.94%
Gamitrinib TPP hexafluorophosphate    
HSP90
        99.68%
Luminespib    
HSP90α, IC50: 7.8 nM
HSP90β, IC50: 21 nM
GRP94, IC50: 535 nM
        99.81%
Rocaglamide        
HSF1, IC50: 50 nM
    99.34%
Novobiocin sodium    
HSP90
        99.12%
Pifithrin-μ  
HSP70
          99.66%
Onalespib    
HSP90, Kd: 0.71 nM
        99.92%
Pimitespib    
HSP90α, Ki: 34.7 nM
HSP90β, Ki: 21.3 nM
        99.15%
Apoptozole  
HSP70, Kd: 0.14 μM
HSC70, Kd: 0.21 μM
          99.42%
Tamoxifen (Standard)    
HSP90
       
HSF1A        
HSF1
    99.94%
KRIBB11        
HSF1, IC50: 1.2 μM
    99.69%
Poly (I:C):Kanamycin (1:1)  
HSP70
         
Col003
HSP47, IC50: 1.8 μM
            99.87%
MKT-077  
HSP70
          98.05%
Alvespimycin hydrochloride    
HSP90, EC50: 62 nM
GRP94, EC50: 65 nM
        98.80%
Arimoclomol maleate          
HSP
  99.96%
BIIB021    
HSP90, Ki: 1.7 nM
HSP90, EC50: 38 nM
        99.19%
ML346  
HSP70, EC50: 4.6 μM (HeLa cells)
          98.25%
Zelavespib    
HSP90, IC50: 51 nM (MDA-MB-468 cells)
        99.93%
Alvespimycin    
HSP90, EC50: 62 nM
GRP94, EC50: 65 nM
        99.24%
Novobiocin    
HSP90
       
Teprenone          
HSP
  99.58%
NXP800        
HSF1
    99.86%
PU-WS13    
GRP94, EC50: 0.22 μM
HSP90α, EC50: 27.3 μM
HSP90β, EC50: 41.8 μM
        99.88%
NVP-HSP990    
HSP90α, IC50: 0.6 nM
HSP90β, IC50: 0.8 nM
GRP94, IC50: 8.5 nM
        99.49%
Grp94 Inhibitor-1    
GRP94, IC50: 2 nM
        98.72%
SNX-2112  
TRAP-1, IC50: 862 nM
HSP90α, IC50: 30 nM
HSP90β, IC50: 30 nM
GRP94, IC50: 4275 nM
        99.49%
AMP-PCP disodium    
HSP90, Kd: 3.8 μM
        99.29%
Retaspimycin Hydrochloride    
HSP90, EC50: 119 nM
GRP94, EC50: 119 nM
       
XL888    
HSP90, IC50: 24 nM
        99.41%
Radicicol    
HSP90, IC50: 1 μM
        99.96%
KNK437
HSP40
HSP70
 
HSP105
      99.04%
Glutamic acid sodium salt            
HSPA5
99.23%
TRC051384  
HSP70
          99.79%
Smurf1-IN-A01    
HSP90β
        99.81%
CCT018159    
human Hsp90β, IC50: 3.2 μM
yeast Hsp90, IC50: 6.6 μM
        99.94%
CCT251236  
HSP72, IC50: 19 nM (SK-OV-3 cells)
          98.82%
Dihydroberberine    
HSP90
        98.44%
VER-82576    
HSP90β, IC50: 58 nM
GRP94, IC50: 4.1 μM
        98.76%
KW-2478    
HSP90α, IC50: 3.8 nM
        99.53%
HM03            
HSPA5
99.51%
Eupalinolide A        
HSF1
    99.92%
Solanesol  
HSP70
          ≥98.0%
Debio 0932    
HSP90α, IC50: 100 nM
HSP90β, IC50: 103 nM
        99.97%
PROTAC HSP90 degrader BP3    
HSP90
        99.54%
NMS-E973    
HSP90α, DC50: 10 nM
        99.61%
VER-49009    
HSP90, IC50: 25 nM
        99.45%
Chetomin    
HSP90
        ≥99.0%
Geldanamycin-FITC    
HSP90
        98.43%
Cucurbitacin D    
HSP90
        99.91%
JG-231  
HSP70
          98.47%
Ethoxyquin    
HSP90
        98.76%
VER-50589    
HSP90, IC50: 21 nM
        99.76%
Icapamespib    
HSP90
        99.60%
MAL3-101  
HSP70
          98.22%
AT-533    
HSP90
        98.38%
Zelavespib hydrochloride    
HSP90, IC50: 51 nM (MDA-MB-468 cells)
        98.80%
GRP78-IN-3            
HSPA5, IC50: 0.59 μM
99.88%
NCT-58    
HSP90
        99.63%
Ursolic acid acetate    
HSP90
        ≥98.0%
Arimoclomol citrate          
HSP
  99.76%
YK5  
HSP70
HSP90
        99.66%
3-Phenyltoxoflavin    
HSP90, Kd: 585 nM
        99.76%
HSP70-IN-1  
HSP70
          98.07%
Rosolutamide        
HSF1
    99.03%
Bimoclomol          
HSP
  99.29%
DN401    
HSP90, IC50: 698 nM
        ≥99.0%
CH5138303    
HSP90α, Kd: 0.52 nM
        99.05%
Tamoxifen-d5    
HSP90
        99.99%
2-Methoxyhydroquinone    
HSP90
        99.57%
YZ129    
HSP90
        99.85%
HS-27    
HSP90
        98.48%
Arimoclomol          
HSP
  99.74%
Icapamespib hydrochloride    
HSP90
        98.67%
SW02  
TRAP1 ATPase, EC50: 150 ± 21 μM
          98.30%
Conglobatin    
HSP90
       
Gedunin    
HSP90
        ≥98.0%
Gamitrinib TPP    
HSP90
       
AP-4-139B  
HSP70, IC50: 180 nM
          98.87%
Aminohexylgeldanamycin    
HSP90
        99.56%
SNX-5422 mesylate    
HSP90, Kd: 41 nM
       
CH5015765    
HSP90
        98.01%
Zelavespib formic    
HSP90, IC50: 51 nM
       
HSP90/mTOR-IN-1    
HSP90, IC50: 69 nM
       
Onalespib lactate    
HSP90, Kd: 0.71 nM
       
Cemdomespib    
HSP90
       
Shepherdin (79-87)    
HSP90
       
Gamendazole    
HSP90AB1
        99.44%
BX-2819    
HSP90, IC50: 41 nM
       
EZH2/HSP90-IN-29    
HSP90, IC50: 60.1 nM
       
A8 peptide  
HSP72
         
Macbecin    
HSP90, IC50: 2 μM
HSP90, Kd: 0.24 μM
       
EV206  
HSP70
         
HSP90/LSD1-IN-1    
HSP90
       
HSP90-IN-20    
HSP90, IC50: ≤10 μM
       
Colletofragarone A2    
HSP90
       
A17 peptide  
HSP70
         
HSP90α-IN-1    
HSP90α, IC50: 111 nM
       
HEMTAC WEE1 degrader-1    
HSP90, IC50: 16.76 nM
       
Aminohexylgeldanamycin hydrochloride    
HSP90
       
YM-08  
HSP70
         
DMT003096  
HSP70
         
Hsp90-IN-40    
HSP90
       
Hsp90-IN-15    
HSP90
       
Antiproliferative agent-72    
HSP90, Kd: 11 nM
       
Hsp90-IN-38    
HSP90, Kd: 68 nM
       
HSP70-IN-6  
HSP70
         
HSP90-IN-33    
HSP90α, EC50: ≥200 μM
HSP90β, EC50: 7.3 μM
       
HSP90-IN-13    
HSP90, IC50: 25.07 nM
       
Tasiamide B    
HSP90
       
KU-177    
HSP90
       
HSP90-IN-9    
HSP90
       
Antitumor agent-174    
HSP90
       
MAO A/HSP90-IN-2    
HSP90, IC50: 0.016 μM
       
HDAC/HSP90-IN-3    
HSP90, IC50: 0.83 μM (fungal Hsp90)
HSP90, IC50: 19.52 μM (human Hsp90)
       
17-AEP-GA    
HSP90
       
GRP78-IN-1  
Grp78
         
HDAC6/HSP90-IN-1    
HSP90, IC50: 46.8 nM
       
HDAC6/HSP90-IN-3    
HSP90, IC50: 0.88 μM
       
Grp94 Inhibitor-2    
GRP94, Kd: 0.48 nM
HSP90α, Kd: 0.65 nM
       
HSP70/SIRT2-IN-1  
HSP70
         
17-GMB-APA-GA    
HSP90
       
HSP90-IN-14    
HSP90β, Kd: 0.26 ± 0.0 μM
       
YM-1 tosylate  
HSP70, IC50: 3.2 μM
         
DDO-6691    
HSP90
       
AMP-PCP    
HSP90, Kd: 3.8 μM
       
PU24FCl    
HSP90
       
Solanesol (Standard)  
HSP70
         
MPC-0767    
HSP90
       
Hsp90-IN-42    
HSP90, IC50: 15.65 nM
       
MAO A/HSP90-IN-1    
HSP90, IC50: 0.019 μM
       
HSP90-IN-29    
HSP90, IC50: 30 nM
       
HSP90-IN-35    
HSP90, IC50: 0.05-0.5 μM
       
CYP51/Hsp90-IN-1    
HSP90
       
Retaspimycin    
HSP90, EC50: 119 nM
GRP94, EC50: 119 nM