2. GPCR/G Protein
  3. P2Y Receptor
  4. P2Y1 antagonist 2

P2Y1 antagonist 2 (Compound 19) is a P2Y1 receptor antagonist (IC50: 0.49 μM). P2Y1 antagonist 2 has significant antiplatelet aggregation activity and exerts its effects by inhibiting P2Y1 receptor. P2Y1 antagonist 2 can upregulate nuclear Nrf2 protein levels, exhibit neuroprotective effects, and resist oxidative stress damage. P2Y1 antagonist 2 can effectively reduce cerebral infarction area and improve neurobehavioral function, and can be used in the study of ischemic stroke.

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P2Y1 antagonist 2 Chemical Structure

P2Y1 antagonist 2 Chemical Structure

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P2Y1 antagonist 2 Related Antibodies

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Description

P2Y1 antagonist 2 (Compound 19) is a P2Y1 receptor antagonist (IC50: 0.49 μM). P2Y1 antagonist 2 has significant antiplatelet aggregation activity and exerts its effects by inhibiting P2Y1 receptor. P2Y1 antagonist 2 can upregulate nuclear Nrf2 protein levels, exhibit neuroprotective effects, and resist oxidative stress damage. P2Y1 antagonist 2 can effectively reduce cerebral infarction area and improve neurobehavioral function, and can be used in the study of ischemic stroke[1].

Molecular Weight

391.35

Formula

C16H11F2N5O3S
SMILES

NC1=NC(CON2C(C(O)=O)=C(N=C2C3=CC(C#N)=CC=C3)C(F)F)=CS1
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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P2Y1 antagonist 2 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

P2Y1 antagonist 2P2Y ReceptorP2Y1MACOHT22 cellsPGE1SD ratsDPPHInhibitorinhibitorinhibit

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P2Y1 antagonist 2
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HY-174126
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