2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. RS-127445 hydrochloride (Standard)

RS-127445 hydrochloride (Standard) 

Cat. No.: HY-15419R Purity: ≥98%
Handling Instructions Technical Support

RS-127445 (hydrochloride) (Standard) is the analytical standard of RS-127445 (hydrochloride). This product is intended for research and analytical applications. RS-127445 hydrochloride is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 hydrochloride shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites.

For research use only. We do not sell to patients.

RS-127445 hydrochloride (Standard) Chemical Structure

RS-127445 hydrochloride (Standard) Chemical Structure

CAS No. : 199864-86-3

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Description

RS-127445 (hydrochloride) (Standard) is the analytical standard of RS-127445 (hydrochloride). This product is intended for research and analytical applications. RS-127445 hydrochloride is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. RS-127445 hydrochloride shows 1000 fold selectivity for this receptor as compared to numerous other receptor and ion channel binding sites.

Molecular Weight

317.79

Formula

C17H17ClFN3
CAS No.
SMILES

NC1=NC(C(C)C)=CC(C2=C3C=CC=CC3=C(F)C=C2)=N1.[H]Cl
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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RS-127445 hydrochloride (Standard) Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

RS-127445 hydrochloride (Standard)199864-86-35-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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