2. GPCR/G Protein
  3. P2Y Receptor
  4. MRS4608

MRS4608 (Compound 17) is a selective P2Y14 receptor antagonist with IC50 values of 20 (hP2Y14R) and 21.4 nM (mP2Y14R). MRS4608 has anti-inflammatory activity and can reduce the infiltration of eosinophils. MRS4608 can be used for the researches of inflammation and immunology, such as asthma.

For research use only. We do not sell to patients.

MRS4608

MRS4608 Chemical Structure

CAS No. : 2370976-04-6

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MRS4608 Related Antibodies

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Description

MRS4608 (Compound 17) is a selective P2Y14 receptor antagonist with IC50 values of 20 (hP2Y14R) and 21.4 nM (mP2Y14R). MRS4608 has anti-inflammatory activity and can reduce the infiltration of eosinophils. MRS4608 can be used for the researches of inflammation and immunology, such as asthma[1].

IC50 & Target[1]

hP2Y14R

20 nM (IC50)

mP2Y14R

21.4 nM (IC50)

Molecular Weight

501.54

Formula

C31H26F3NO2
CAS No.
SMILES

O=C(C1=CC2=C(C(C3=CC=C(C45CCN(CC5)CC4)C=C3)=C1)C=CC(C6=CC=C(C(F)(F)F)C=C6)=C2)O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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MRS4608 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MRS46082370976-04-6MRS 4608MRS-4608P2Y ReceptorInhibitorinhibitorinhibit

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