1. Academic Validation
  2. Rapavir, a novel inhibitor of sodium taurocholate cotransporting polypeptide, potently blocks hepatitis B virus entry

Rapavir, a novel inhibitor of sodium taurocholate cotransporting polypeptide, potently blocks hepatitis B virus entry

  • Signal Transduct Target Ther. 2025 Apr 23;10(1):130. doi: 10.1038/s41392-025-02214-x.
Jia He # 1 Haibo Yu # 2 Kunling Song # 1 Ailong Huang 3 Yongjun Dang 4 Juan Chen 5 6 Zufeng Guo 7
Affiliations

Affiliations

  • 1 Basic Medicine Research and Innovation Center for Novel Target and Therapeutic Intervention (Ministry of Education), College of Pharmacy & Department of Breast and Thyroid Surgery of the Second Affiliated Hospital, Chongqing Medical University, Chongqing, China.
  • 2 Institute for Viral Hepatitis, Key Laboratory of Molecular Biology for Infectious Diseases (Ministry of Education), Department of Infectious Diseases, The Second Affiliated Hospital, Chongqing Medical University, Chongqing, China.
  • 3 Institute for Viral Hepatitis, Key Laboratory of Molecular Biology for Infectious Diseases (Ministry of Education), Department of Infectious Diseases, The Second Affiliated Hospital, Chongqing Medical University, Chongqing, China. ahuang@cqmu.edu.cn.
  • 4 Basic Medicine Research and Innovation Center for Novel Target and Therapeutic Intervention (Ministry of Education), College of Pharmacy & Department of Breast and Thyroid Surgery of the Second Affiliated Hospital, Chongqing Medical University, Chongqing, China. yjdang@cqmu.edu.cn.
  • 5 Institute for Viral Hepatitis, Key Laboratory of Molecular Biology for Infectious Diseases (Ministry of Education), Department of Infectious Diseases, The Second Affiliated Hospital, Chongqing Medical University, Chongqing, China. chenjuan2014@cqmu.edu.cn.
  • 6 College of Biomedical Engineering, Chongqing Medical University, Chongqing, China. chenjuan2014@cqmu.edu.cn.
  • 7 Basic Medicine Research and Innovation Center for Novel Target and Therapeutic Intervention (Ministry of Education), College of Pharmacy & Department of Breast and Thyroid Surgery of the Second Affiliated Hospital, Chongqing Medical University, Chongqing, China. zfguo@cqmu.edu.cn.
  • # Contributed equally.
Figures
Products
  • Cat. No.
    Product Name
    Description
    Target
    Research Area
  • HY-172835
    NTCP Inhibitor
    HBV