2. Metabolic Enzyme/Protease
  3. Glutathione S-transferase
  4. GSTA4-IN-1

GSTA4-IN-1 (Compound 3a) is a potent and competitive inhibitor of glutathione S-transferase A4 (GSTA4), with an IC50 of 3.12 μM and a Ki of 2.38 μM. GSTA4-IN-1 is cytotoxic to colorectal cancer cells. GSTA4-IN-1 can be used for research on colorectal cancer.

For research use only. We do not sell to patients.

GSTA4-IN-1

GSTA4-IN-1 Chemical Structure

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GSTA4-IN-1 Related Antibodies

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Description

GSTA4-IN-1 (Compound 3a) is a potent and competitive inhibitor of glutathione S-transferase A4 (GSTA4), with an IC50 of 3.12 μM and a Ki of 2.38 μM. GSTA4-IN-1 is cytotoxic to colorectal cancer cells. GSTA4-IN-1 can be used for research on colorectal cancer[1].

Molecular Weight

550.00

Formula

C27H21ClFN5O3S
SMILES

O=C(NC1=CC=CC(F)=C1)NC2=NN=C(CC3=C(C)N(C(C4=CC=C(Cl)C=C4)=O)C5=C3C=C(OC)C=C5)S2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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GSTA4-IN-1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GSTA4-IN-1Glutathione S-transferaseGlutathione transferasesGSTsIndomethacin ureaThiadiazole ringGSTA4 inhibitionCytotoxicityMolecular dockingInhibitorinhibitorinhibit

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