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  3. Drug Derivative
  4. CGP 29030A

CGP 29030A is an orally effective and specific analgesic agent. CGP 29030A inhibits nociceptive spinal cord neurons without affecting normal sensory functions. CGP 29030A also inhibits gamma motor neurons, which may be beneficial for treating pain disorders that occur concurrently due to increased motor activity (such as cramp, spasm).

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CGP 29030A

CGP 29030A Chemical Structure

CAS No. : 113240-27-0

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Description

CGP 29030A is an orally effective and specific analgesic agent. CGP 29030A inhibits nociceptive spinal cord neurons without affecting normal sensory functions. CGP 29030A also inhibits gamma motor neurons, which may be beneficial for treating pain disorders that occur concurrently due to increased motor activity (such as cramp, spasm)[1].

In Vivo

CGP 29030A (≥ 10 mg/kg, p.o.) rapidly inhibits nociceptive dorsal horn neurons in the rat and significantly inhibits the activity of γ-motor neurons in gastrocnemius-soleus muscle[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

425.35

Formula

C21H26Cl2N2O3
CAS No.
SMILES

O=C(N1CCN(CC1)CCC2=CC=C(C=C2)Cl)C3=CC(OC)=CC(OC)=C3.Cl
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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CGP 29030A Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CGP 29030A113240-27-0Drug DerivativeDrug derivativepiperazine derivativedorsal horn neuronsgamma-motoneuronsnociceptivehigh-threshold mechanosensitive receptorsinhibitory actionanalgesic actionsupraspinal CNSInhibitorinhibitorinhibit

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