1. Signaling Pathways
  2. PI3K/Akt/mTOR
  3. mTOR
  4. mTOR Inhibitors

mTOR Inhibitors

mTOR

mTORC1

mTORC2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

mTOR Inhibitors, Activators & Modulators
Product Name mTOR mTORC1 mTORC2 Purity
Rapamycin  
mTOR, IC50: 0.1 nM (in HEK293 cells )
  99.94%
MHY1485  
mTORC1
mTORC2
99.93%
Everolimus  
mTOR, IC50: 5-6 nM
  99.85%
Torin 1
mTOR, IC50: 3 nM
mTORC1, IC50: 2-10 nM
mTORC2, IC50: 2-10 nM
99.28%
AZD-8055
mTOR, IC50: 0.8 nM
    99.60%
Sapanisertib
mTOR, IC50: 1 nM
    99.78%
Salidroside
mTOR
    99.90%
Temsirolimus  
mTOR, IC50: 1.76 μM
  99.56%
L-Leucine  
mTORC1
  99.79%
Dactolisib
mTOR, IC50: 20.7 nM
    99.94%
Torin 2
mTOR, IC50: 2.81 nM
mTOR, EC50: 0.25 nM (Cell Assay)
    99.65%
PI-103  
mTORC1, IC50: 20 nM
mTORC2, IC50: 83 nM
99.82%
Omipalisib  
mTORC1, Ki: 0.18 nM
mTORC2, Ki: 0.3 nM
99.94%
Dihydromyricetin  
mTORC1
mTORC2
99.73%
RMC-5552  
mTORC1
  99.94%
JR-AB2-011    
mTORC2, IC50: 0.36 μM
98.15%
Camonsertib
mTOR, IC50: 120 nM
    99.75%
RapaLink-1
mTOR
    99.92%
Torkinib
mTOR, IC50: 8 nM
mTORC1, IC50: 30 nM
mTORC2, IC50: 58 nM
99.03%
3BDO
mTOR
    99.93%
Aloe emodin    
mTORC2
98.32%
hSMG-1 inhibitor 11j
mTOR, IC50: 50 nM
    99.82%
Vistusertib
mTOR, IC50: 2.81 nM
    99.32%
Gedatolisib
mTOR, IC50: 1.6 nM
    99.68%
Paxalisib
mTOR, Ki: 70 nM
    99.51%
PF-04691502
mTOR, Ki: 16 nM
    99.91%
hSMG-1 inhibitor 11e
mTOR, IC50: 45 nM
    99.94%
KU-0063794  
mTORC1, IC50: 10 nM
mTORC2, IC50: 10 nM
99.67%
Samotolisib
mTOR, IC50: 165 nM
    99.27%
Apitolisib
mTOR, Ki: 17 nM
    99.29%
Bimiralisib
mTOR, IC50: 89 nM
    98.62%
CC-115
mTOR, IC50: 21 nM
    99.82%
BGT226
mTOR
    99.85%
Voxtalisib
mTOR, IC50: 157 nM
mTORC1, IC50: 160 nM
mTORC2, IC50: 910 nM
99.82%
OSI-027
mTOR, IC50: 4 nM
mTORC1, IC50: 22 nM
mTORC2, IC50: 65 nM
99.95%
Dactolisib Tosylate
mTOR, IC50: 20.7 nM
    99.87%
WYE-132
mTOR, IC50: 0.19 nM
    99.90%
Onatasertib
mTOR, IC50: 16 nM
    99.13%
PP121
mTOR, IC50: 10 nM
    99.51%
PKI-402
mTOR, IC50: 3 nM
    99.17%
GSK1059615
mTOR, IC50: 12 nM
    99.76%
mTOR inhibitor-3
mTOR, Ki: 1.5 nM
    99.79%
Ridaforolimus  
mTOR
  99.75%
VS-5584
mTOR, IC50: 37 nM
    98.71%
GNE-317
mTOR
    98.76%
CZ415
mTOR, pIC50: 8.07
    98.39%
ETP-46464
mTOR, IC50: 0.6 nM
    99.54%
(+)-Usnic acid  
mTORC1
mTORC2
99.63%
PI-103 Hydrochloride  
mTORC1, IC50: 20 nM
mTORC2, IC50: 83 nM
98.55%
BGT226 maleate
mTOR
    99.92%
PQR530
mTOR, Kd: 0.33 nM
    99.98%
Palomid 529  
TORC1
TORC2
99.37%
CC-115 hydrochloride
mTOR, IC50: 21 nM
    98.03%
PF-04979064
mTOR, Ki: 1.42 nM
    99.54%
GNE-493
mTOR, IC50: 30 nM
    99.81%
GDC-0349
mTOR, Ki: 3.8 nM
    98.02%
PQR620  
mTORC1
mTORC2
98.01%
WAY-600
mTOR, IC50: 9 nM
    99.86%
PI3K/mTOR Inhibitor-2
mTOR, IC50: 4.7 nM
    99.10%
Hederacolchiside A1
mTOR
    ≥99.0%
HDACs/mTOR Inhibitor 1
mTOR, IC50: 1.2 nM
    99.01%
PKI-179
mTOR, IC50: 0.42 nM
    ≥98.0%
NSC781406
mTOR, IC50: 5.4 nM
    99.97%
MT 63-78  
mTORC1
  98.00%
MTI-31
mTOR, Ki: 0.2 nM
mTOR, IC50: 39 nM (100 μM ATP)
    99.98%
XL388
mTOR, IC50: 9.9 nM
    99.74%
WYE-354
mTOR, IC50: 5 nM
    98.04%
mTOR inhibitor-8
mTOR
    98.14%
Rotundic acid
mTOR
    99.41%
GNE-477
mTOR, Ki: 21 nM
    98.75%
ETP-45658
mTOR, IC50: 152.0 nM
    98.97%
Zederone
mTOR
    99.61%
PI3K/mTOR Inhibitor-4
mTOR, IC50: 13.85 nM
   
FT-1518  
mTORC1
mTORC2
98.62%
HTH-01-091
mTOR, IC50: 632 nM
    98.64%
AZD3147  
mTORC1
mTORC2
99.93%
WYE-687
mTOR, IC50: 7 nM
    98.05%
PKI-179 hydrochloride
mTOR, IC50: 0.42 nM
    99.66%
CC214-2  
mTORC1
mTORC2
98.41%
GNE-490
mTOR, IC50: 750 nM
   
TML-6
mTOR
    99.01%
Pomiferin
mTOR, IC50: 6.2 μM
    98.98%
8-Aminoadenosine
mTOR
    99.94%
PI3K-IN-37
mTOR, IC50: 4 nM
    ≥99.0%
PI3K-IN-22
mTOR, IC50: 0.6 nM
    99.50%
SN32976
mTOR, IC50: 194 nM
    99.49%
WYE-687 dihydrochloride
mTOR, IC50: 7 nM
    ≥98.0%
Coronarin A  
mTORC1
  ≥98.0%
PI3K-IN-18
mTOR, IC50: 49 nM
    ≥99.0%
FD274
mTOR, IC50: 2.03 nM
    99.45%
PI3Kα/mTOR-IN-1
mTOR, Ki: 10.6 nM
    99.30%
HSP90/mTOR-IN-1
mTOR, IC50: 29 nM
   
PI3K/mTOR Inhibitor-1
mTOR, IC50: 186 nM
   
mTOR inhibitor-2
mTOR, IC50: 7 nM
   
PI3K/mTOR Inhibitor-9
mTOR, IC50: 38 nM (phospho-S6 cellular assay)
mTOR, IC50: 16 nM (Ser240/244 cellular assay)
   
ATM Inhibitor-3
mTOR
   
ATM Inhibitor-4
mTOR
   
mTOR/HDAC-IN-1
mTOR, IC50: 0.49 nM
   
PI3K/mTOR Inhibitor-3
mTOR
   
PI3Kα-IN-5
mTOR, IC50: 3.3 nM
   
PI3K/mTOR Inhibitor-12
mTOR, IC50: 3.12 nM
   
PI3K/mTOR Inhibitor-8
mTOR, IC50: 12 nM
   
ATR-IN-20
mTOR, IC50: 18 nM
   
Antifungal agent 106
mTOR, IC50: 0.8 μM
   
PI3K/mTOR Inhibitor-14
mTOR, IC50: 10.1 nM
   
mTOR/HDAC6-IN-1
mTOR, IC50: 133.7 nM
   
PI3K/mTOR-IN-17
mTOR, IC50: 0.21 μM
   
mTOR inhibitor-13
mTOR, IC50: 0.29 nM
   
mTOR inhibitor-17
mTOR, IC50: 0.68 nM
   
mTOR inhibitor-16
mTOR, IC50: 1.25 nM
   
mTOR inhibitor-10
mTOR, IC50: 0.7 nM