2. Signaling Pathways
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  4. Drug Derivative

Drug Derivative

Drug derivative

Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.

Drug Derivative Related Products (1529):

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-147251
    SRI 6409-94
    		99.25%
    SRI 6409-94 is an orally active Ro 13-6298 analogue that is teratogenic. SRI 6409-94 serves as a molecular tool to study the effect of the three-dimensional configuration of retinol on teratogenic activity.
    SRI 6409-94
  • HY-W011180
    Vitamin A Propionate
    Vitamin A Propionate is an ester compound of vitamin A. In nutritional studies of foals, different doses have different effects on growth, serum biochemistry and hematological indicators. Too high or too low doses will produce adverse effects and are related to the vitamin A concentration in plasma, liver and kidneys.
    Vitamin A Propionate
  • HY-Y0123
    DL-Tyrosine
    		≥98.0%
    DL-Tyrosine is an aromatic nonessential amino acid synthesized from the essential amino acid phenylalanine. DL-Tyrosine is a precursor for several important neurotransmitters (epinephrine, norepinephrine, dopamine).
    DL-Tyrosine
  • HY-W140465
    L-Homotyrosine
    L-Homotyrosine is a tyrosine derivative that can be used for solid-phase peptide synthesis.
    L-Homotyrosine
  • HY-148586
    β-Estradiol 17-hemisuccinate
    		98.83%
    β-Estradiol 17-hemisuccinate is a synthetic derivative of estradiol (HY-B0141).
    β-Estradiol 17-hemisuccinate
  • HY-122365R
    Inositol nicotinate (Standard)
    Inositol nicotinate (Standard) is the analytical standard of Inositol nicotinate. This product is intended for research and analytical applications. Inositol nicotinate, with vasodilatory effect, is used in the study of Peripheral arterial disease (PAD).
    Inositol nicotinate (Standard)
  • HY-Y0004
    2-Pyridinemethanol
    		99.98%
    2-Pyridinemethanol is a pyridylalcohol, with hypoglycemic activity.
    2-Pyridinemethanol
  • HY-B0917
    Bromindione
    		98.11%
    Bromindione is a potent and long-acting, Inandione-derived, oral anticoagulant compound.
    Bromindione
  • HY-N8531
    4α-Methylcholesterol
    		99.90%
    4α-Methylcholesterol is a Cholesterol derivative. 4α-Methylcholesterol can oxidize 3-hydroxy steroid, with the apparent Km of 12.6 μM.
    4α-Methylcholesterol
  • HY-400882
    Tosylate-DPA-714
    Tosylate-DPA-714 (compound 2) is a DPA-714 (HY-122607) tosylate analog. Tosylate-DPA-714 is a precursor for 18F-DPA-714. DPA-714 is a translocator protein (TSPO)-specific ligand.
    Tosylate-DPA-714
  • HY-W004288
    Methyl myristate
    		99.70%
    Methyl myristate is a saturated fatty acid methyl ester obtained from the esterification of myristic acid. Methyl myristate shows a high melanin induction in B16F10 melanoma.
    Methyl myristate
  • HY-W004286
    Methyl laurate
    		99.78%
    Methyl laurate, a 12-carbon saturated fatty acid, is an esterified version of lauric acid.
    Methyl laurate
  • HY-W087207
    Loxoprofen L-menthol ester
    		99.73%
    Loxoprofen L-menthol ester is a degradation product Loxoprofen sodium (HY-B0578A). Loxoprofen sodium is a non-steroidal, orally active anti-inflammatory agent with analgesic and anti-pyretic properties.
    Loxoprofen L-menthol ester
  • HY-W587486R
    N-Acetyltaurine (Standard)
    N-Acetyltaurine (Standard) is the analytical standard of N-Acetyltaurine. This product is intended for research and analytical applications. N-Acetyltaurine is a sulfonate that can serve as a carbon source or a nitrogen source, and an energy source for microbial growth (such as the NAT strain). Additionally, N-Acetyltaurine is also a substrate for the amidase enzyme, porcine kidney N-acetyl-β-alanine deacetylase [EC 3.5.1.21][1].
    N-Acetyltaurine (Standard)
  • HY-128856
    P7C3-OMe
    		98.26%
    P7C3-OMe is a pro-neurogenic compound, has therapeutic benefits in neuropsychiatric and/or neurodegenerative disease. The R-enantiomer of P7C3-OMe is far more active than the S-enantiomer.
    P7C3-OMe
  • HY-W050088
    Isoxepac
    		99.92%
    Isoxepac (HP 549) is an orally active non-steroidal anti-inflammatory agent. Isoxepac can inhibit Carrageenan (HY-125474) paw oedema, adjuvant-induced polyarthritis, and prostaglandin synthesis. Isoxepac (200 mg) has an analgesic effect after meniscectomy with a low incidence of side effects. Isoxepac can be used in the research of inflammatory (rheumatoid arthritis) and pain-related diseases.
    Isoxepac
  • HY-76779
    4-(Chloromethyl)-7-hydroxycoumarin
    		98.01%
    4-(Chloromethyl)-7-hydroxycoumarin (compound 4) is a hydroxycoumarin derivative with potent antioxidant effect and high hydroxyl radical-scavenging property. 4-(Chloromethyl)-7-hydroxycoumarin contains a methyl group and a chlorine group in the heterocyclic ring. A series of coumarins incorporating hydroxy-, chloro- and/or chloromethyl-moieties has been investigated as potent inhibitors of the zinc enzyme carbonic anhydrase, expecially tumor-associated isoforms CA IX and XII.
    4-(Chloromethyl)-7-hydroxycoumarin
  • HY-12692
    DO3A tert-Butyl ester
    		98.0%
    DOTA tert-Butyl ester is a cyclic tosamide benzyl derivative.
    DO3A tert-Butyl ester
  • HY-139453
    LP-184
    		99.37%
    LP-184 (compound 6), an acylfulvene analog, inhibits tumor growth. LP-184 has potent anti-cancer activity in the ovarian, colon, prostate and pancreatic cell lines. (patent WO2007019308A2).
    LP-184
  • HY-105270A
    Tallimustine hydrochloride
    		98.23%
    Tallimustine hydrochloride, a distamycin-A derivative, is an anticancer agent.
    Tallimustine hydrochloride