2. Signaling Pathways
  3. Others
  4. Drug Derivative

Drug Derivative

Drug derivative

Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.

Drug Derivative Related Products (1652):

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-158595
    15(R),19(R)-Hydroxy prostaglandin F2α
    15(R),19(R)-Hydroxy prostaglandin F2α (15(R),19(R)-Hydroxy PGF2α) is an analog of 19(R)-Hydroxy-prostaglandin F2α. 19(R)-Hydroxy-prostaglandin F2α (HY-N7857) is an ω-1 hydroxylase metabolite of PGF2α found in human semen.
    15(R),19(R)-Hydroxy prostaglandin F2α
  • HY-120700
    L-682,679
    L-682,679 is an active compound.
    L-682,679
  • HY-169479
    Betulinic glycine amide
    Betulinic glycine amide (compound 5a) is a pentacyclic triterpenoid and derivative of Betulinic acid (HY-10529). Betulinic glycine amide has been used as a precursor in the synthesis of betulinic acid derivatives with anticancer and antiviral activity.
    Betulinic glycine amide
  • HY-117486
    RU 56187
    RU 56187 is an active compound.
    RU 56187
  • HY-117412
    KCG 1
    KCG 1 is a potent and selective anti-tumor agent that displays anti-prollferative and cytotoxic effects on epithelial tumoral cells.
    KCG 1
  • HY-113526
    AR-12463
    AR-12463 is a derivative of Trapidil (HY-B1016). AR-12463 inhibits the conversion of [14C]acetate to cholesterol. AR-12463 significantly reduces the elevation of total cholesterol in rabbit serum and prevents cholesterol incorporation into tissues. AR-12463 can be used to study atherosclerosis.
    AR-12463
  • HY-127069
    Methiomeprazine
    Methiomeprazine is an active compound.
    Methiomeprazine
  • HY-115774
    5-HT4R agonist-1
    5-HT4R agonist-1 is an active compound.
    5-HT4R agonist-1
  • HY-103432
    DPP4-In
    DPP4-In is an active compound.
    DPP4-In
  • HY-113942
    Cycloate
    Cycloate is an active compound.
    Cycloate
  • HY-122712
    CB-002
    CB-002 is an active molecule that can be used for the study of advanced malignant solid neoplasm.
    CB-002
  • HY-105270
    Tallimustine
    Tallimustine (FCE 24517), a distamycin-A derivative, is an anticancer agent.
    Tallimustine
  • HY-106469
    Taltrimide
    Taltrimide (MY-117), a lipophilic derivative of Taurine (HY-B0351), strongly inhibits the sodium-independent binding of Taurine to synaptic membranes of brain, the effects on the binding of GABA being less pronounced. Taltrimide exhibits definitive anticonvulsive effects in experimental epilepsy models.
    Taltrimide
  • HY-108409
    Progesterone carboxylic acid
    Progesterone carboxylic acid (Testosterone-17β-carboxylic acid) is an androstenedione analogue. Progesterone carboxylic acid can conjugate with 20-mer peptide nucleic acid (PNA) and the conjugate has superior binding capacity on complementary DNA. Progesterone carboxylic acid can be used for cancers and type 2 diabetes (T2D) research.
    Progesterone carboxylic acid
  • HY-139068
    Ibuprofen arginine
    Ibuprofen arginine is an orally active L-arginine of Ibuprofen (HY-78131). With rapid absorption and high bioavailability, Ibuprofen arginine can effectively relieve a variety of acute pain, and has little damage to gastric mucosa and is well tolerated. Ibuprofen arginine can be used in research for pain relief.
    Ibuprofen arginine
  • HY-19300A
    PNU-142731A
    PNU-142731A is an active compound.
    PNU-142731A
  • HY-117439
    (R)-Norverapamil
    (R)-Norverapamil is an active compound.
    (R)-Norverapamil
  • HY-124168
    PF-244
    PF-244 is an active compound.
    PF-244
  • HY-171977
    UTKO1
    UTKO1 (Compound 2) is a derivate of Moverastin.UTKO1 has optical activity and significant inhibitory activity against tumor cell migration by abrogating the binding of 14-3-3ζ/Tiam1. UTKO1 can be used for cancers like esophageal cancer and epidermoid carcinoma research.
    UTKO1
  • HY-113812
    ZK110841
    ZK110841 is an active compound.
    ZK110841