2. Others

Others

Others

Related Products

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There are a number of inhibitors, agonists, and antagonists which we cannot make precise classification because the research area is still unknown.

Others Related Products (60510):

Cat. No. Product Name CAS No. Purity Chemical Structure
  • HY-117460
    Indanorex 16112-96-2 98%
    Indanorex is a stimulant agent with appetite suppressant effects and antihyperglycemic effects.
    Indanorex
  • HY-117484
    Rubrosterone 19466-41-2 98%
    Rubrosterone is a metabolite of insect metamorphosing substances, that can be isolated from Achyranthes rubrofuca and A. fmaiei (Amaranthaceae).
    Rubrosterone
  • HY-117615
    Rhapontisterone 137476-71-2 98%
    Rhapontisterone is a natural product.
    Rhapontisterone
  • HY-117636
    (Rac)-L-659989 129314-27-8 98%
    (Rac)-L-659989 is the racemate of L-659989 (HY-121394). L-659989 s an orally active, extremely potent, selective and competitive platelet activating factor (PAF) receptor antagonist.
    (Rac)-L-659989
  • HY-117717
    (Rac)-SC-31391 144730-93-8 98%
    (Rac)-SC-31391, a prostaglandin analog, is a strong activator of the bladder muscle contractility that enhanced twitch responses elicited by field stimulation in the guinea pig detrusor muscle. (Rac)-SC-31391 contracts human bladder muscle through the activation of PGF2α receptors.
    (Rac)-SC-31391
  • HY-117740
    Heronamide C 1257083-94-5 98%
    Heronamide C is a polyketide macrolactam isolated from marine Streptomyces that has the activity of producing reversible non-cytotoxic effects on mammalian cell morphology.
    Heronamide C
  • HY-117901
    Sandoricin 133585-55-4 98%
    Sandoricin is a limonoid compound that can be extracted from the seeds of Sandoricum koetjape. Sandoricin exhibits strong antifeedant properties in larvae of Fall Armyworm (Spodoptera frugiperda) and European Corn Borer (Ostrinia nubilalis) fed on artificial diets. Sandoricin induces reduced growth rate and delayed pupation at lower doses, while higher doses cause massive mortality of larvae. Sandoricin is a potential field insecticide.
    Sandoricin
  • HY-117925
    Personalised postprandial-targeting 1529779-90-5 98%
    Personalised postprandial-targeting is a way to modulate water-heme interactions with activity against low-spin P450 complexes. Personalised postprandial-targeting is able to maintain the axial water ligands of CYP2C9 even in the presence of inhibitors. Personalised postprandial-targeting also allows the hydrogen atoms of the axial water ligands to be observed by EPR spectroscopy, providing insights into the enzyme active site.
    Personalised postprandial-targeting
  • HY-118009
    Azotochelin 23369-85-9 98%
    Azotochelin (ISD-I 207) is a biscatecholate siderophore found in the strain of Azotobacter vinelandii.
    Azotochelin
  • HY-118112
    4-N-Maleimidobenzoicacid-NHS 64191-06-6 98%
    4-N-Maleimidobenzoicacid-NHS is a PEG linker that finds utility in bioconjugation endeavors and protein labeling ventures. Specifically designed for selective reaction with thiol groups, the maleimide group establishes covalent linkages, thereby facilitating the coupling of proteins, peptides, or diverse molecules to thiol-bearing biomolecules. The NHS ester is able to react specifically and efficiently with primary amines (e.g. the side chain of lysine residues or aminosilane-coated surfaces) at neutral or slightly basic conditions to form a covalent bond.
    4-N-Maleimidobenzoicacid-NHS
  • HY-118115
    Pyrabactin 419538-69-5 98%
    Pyrabactin is a seed-selective abscisic acid (ABA) agonist that acts through Pyrabactin Resistance 1 (PYR1) and PYL1. Pyrabactin is used as a synthetic plant growth inhibitor.
    Pyrabactin
  • HY-118124
    2-Iodoestradiol 24381-12-2 98%
    2-Iodoestradiol is a potent human sex hormone binding globulin (SHBG) ligand with a remarkably high affinity for SHBG. 2-Iodoestradiol exhibits competition for the same binding site as dihydrotestosterone in binding to human SHBG. The binding affinity constant of 2-Iodoestradiol at physiological pH and 37 degrees Celsius is 2.4 x 10(9) M-1, exceeding that for SHBG. 2-Iodoestradiol has been shown to bind to serum albumin, but with lower affinity. The radioisotope 125I-derivative of 2-Iodoestradiol has been used to study the binding properties of human SHBG, demonstrating its potential application in biological research.
    2-Iodoestradiol
  • HY-118136
    CGP 28392 89289-93-0 98%
    CGP 28392 is an activator for calcium channel, and reactivates the oxygen evolution in calcium-deficient photosystem II (PS II) particles.
    CGP 28392
  • HY-118156
    L-699333 155238-60-1 98%
    L-699333 is a 5-lipoxygenase (5-LO) inhibitor belonging to the thieno[2,3,4-cd]indole class. This compound has a 2-ethoxybutyric acid side chain and is a potent inhibitor of the biosynthesis of 5-HPETE and LTB4 produced from human 5-LO, with ICm values of 22 nM, 7 nM, and 3.8 pM for human neutrophils and whole blood, respectively. L-699333 has shown anti-inflammatory and antiasthmatic effects in a variety of animal models, including rat pleurisy models, antigen-induced wheezing models, and awake macaque and sheep asthma models. Its inhibition of 5-LO is highly selective, with higher ICm values or stronger competitive inhibition in FLAP binding assays compared to inhibition of human 15-LO, porcine 12-LO, and ram epididymal cyclooxygenase. The racemic enantiomer 14g of L-699333 is the most potent enantiomer to date, with inhibitory effects similar to those of the known MK-0591, which has been shown in clinical trials to inhibit the biochemical effects of LTB4 biosynthesis in vitro and LTE4 excretion in urine.
    L-699333
  • HY-118161
    1-Adamantylaspartate 115545-59-0 98%
    1-Adamantylaspartate is a newly developed β-β-1-imidopropionic acid used to synthesize the C-terminal octapeptide of the β subunit of human chorionic gonadotropin (hCG) and the hexadecapeptide of the α subunit of the insulin receptor (30-55) by conventional solution methods and solid phase methods, aiming to inhibit the formation of asparagine during the synthesis of asparagyl peptides. Studies have shown that β-β-1-imidopropionic acid is an effective protector of the β-carboxyl function of aspartic acid residues.
    1-Adamantylaspartate
  • HY-118217
    Cyclanilide 113136-77-9 99.91%
    Cyclanilide (RPA90946) serves as a plant growth regulator that is applied to cotton during various growth stages.
    Cyclanilide
  • HY-118226
    5,6,7,8-Tetrahydro-2-naphthoic acid 1131-63-1 98.53%
    5,6,7,8-Tetrahydro-2-naphthoic acid is a synthetic intermediate useful for pharmaceutical synthesis.
    5,6,7,8-Tetrahydro-2-naphthoic acid
  • HY-118234
    (Rac)-PD 138312 107334-06-5 98%
    (Rac)-PD 138312 is the racemate of PD 138312. PD 138312 is a potent and orally active antibacterial agent against Gram-positive bacteria.
    (Rac)-PD 138312
  • HY-118265
    N-Acetylglutaminylglutamine amide 123199-99-5 98%
    N-Acetylglutaminylglutamine amide is a dipeptide previously reported only in osmotically stressed Rhizobium meliloti and Pseudomonas fluorescens.
    N-Acetylglutaminylglutamine amide
  • HY-118325
    Epibatidine dihydrochloride 166374-43-2 98%
    Epibatidine dihydrochloride serves as a powerful agonist for nicotinic receptors.
    Epibatidine dihydrochloride