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Results for "

peptidergic

" in MedChemExpress (MCE) Product Catalog:

7

Inhibitors & Agonists

5

Peptides

2

Natural
Products

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-P0249A
    Phe-Met-Arg-Phe amide trifluoroacetate

    		Potassium Channel Neurological Disease
    Phe-Met-Arg-Phe amide trifluoroacetate is an activator of K + current, with ED50 of 23 nM in the peptidergic caudodorsal neurons.
    Phe-Met-Arg-Phe amide trifluoroacetate
  • HY-135013
    Umbellulone

    		TRP Channel Neurological Disease
    Umbellulone is an active constituent of the leaves of Umbellularia californica. Umbellulone stimulates the TRPA1 channel in a subset of peptidergic, nociceptive neurons, activating the trigeminovascular system via this mechanism .
    Umbellulone
  • HY-105174
    BPC 157

    		JAK FAK Inflammation/Immunology
    BPC 157 is the 15-amino acide fragment of gastric peptide BPC. BPC 157 exhibits wound healing promoting and neuroprotective activity. BPC 157 maintains the integrity of the gastrointestinal mucosa without significant toxicity. BPC 157 acetate counteracts NSAIDs/insulin overdose/copper-induced toxicity. BPC 157 ameliorates specific (over)stimulated/damaged neurotransmitter systems-induced behavioral disorders through serotonergic and dopaminergic systems .
    BPC 157
  • HY-P0249
    Phe-Met-Arg-Phe, amide

    		Potassium Channel Neurological Disease
    Phe-Met-Arg-Phe, amide dose dependently (ED50=23 nM) activates a K + current in the peptidergic caudodorsal neurons.
    Phe-Met-Arg-Phe, amide
  • HY-P0249B
    Phe-Met-Arg-Phe, amide acetate

    		Potassium Channel Neurological Disease
    Phe-Met-Arg-Phe, amide acetate dose dependently (ED50=23 nM) activates a K + current in the peptidergic caudodorsal neurons .
    Phe-Met-Arg-Phe, amide acetate
  • HY-107095
    JNJ19567470

    R317573; CRA5626; TAI041

    		 CRFR Neurological Disease
    JNJ19567470 (R317573) is a selective, non-peptidergic CRF type 1 receptor (CRF1) antagonist. JNJ19567470 blocks NaLac-induced panic-like behaviour and cardiovascular responses. JNJ19567470 decreases regional glucose utilization in the amygdala, and attenuates anxiety responses .
    JNJ19567470
  • HY-168758
    Delta3,5-cholestadien-7-one

    		GABA Receptor Neurological Disease
    Delta3,5-cholestadien-7-one is an oxysterol and a negative allosteric modulator of GABAA receptors. Delta3,5-cholestadien-7-one reduces GABA-induced currents in HEK cells expressing α1β1γ2 or α4β3γ2 subunit-containing GABAA receptors with IC50 values of 1.5 and 1 µM, respectively. Delta3,5-cholestadien-7-one reduces GABA-induced depolarization of peptidergic and non-peptidergic nociceptors, C-LTMRs, and cold thermosensors in isolated mouse dorsal root ganglion (DRG) neurons .
    Delta3,5-cholestadien-7-one

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