2. GPCR/G Protein Neuronal Signaling Others
  3. Cholecystokinin Receptor Drug Isomer
  4. (rac)-CHEMBL333994

(rac)-CHEMBL333994 is the racemate of CHEMBL333994 (HY-U00363). CHEMBL333994 is a potent and orally active Cholecystokinin A receptor (CCK-A receptor) antagonist, with an IC50 of 0.67 nM. CHEMBL333994 selectively antagonizes peripheral CCK receptors. CHEMBL333994 increases CCK mRNA level. CHEMBL333994 can be used for research of chronic pancreatitis.

For research use only. We do not sell to patients.

(rac)-CHEMBL333994

(rac)-CHEMBL333994 Chemical Structure

CAS No. : 126149-42-6

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(rac)-CHEMBL333994 Related Antibodies

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Description

(rac)-CHEMBL333994 is the racemate of CHEMBL333994 (HY-U00363). CHEMBL333994 is a potent and orally active Cholecystokinin A receptor (CCK-A receptor) antagonist, with an IC50 of 0.67 nM. CHEMBL333994 selectively antagonizes peripheral CCK receptors. CHEMBL333994 increases CCK mRNA level. CHEMBL333994 can be used for research of chronic pancreatitis[1][2][3].

Molecular Weight

438.45

Formula

C26H19FN4O2
CAS No.
SMILES

O=C(C(N1)=CC2=C1C=CC=C2)NC3C(N4C5=C(CC4)C=CC=C5C(C6=CC=CC=C6F)=N3)=O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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(rac)-CHEMBL333994 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(rac)-CHEMBL333994126149-42-6(rac)-FK-480Cholecystokinin ReceptorDrug IsomerCCK ReceptorInhibitorinhibitorinhibit

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