2. Signaling Pathways
  3. GPCR/G Protein
  4. Chemerin Receptor
  5. ChemR23/CMKLR1 Isoform

ChemR23/CMKLR1

 

ChemR23/CMKLR1 Related Products (1):

Cat. No. Product Name Effect Purity
  • HY-174140
    CMKLR1 antagonist 3
    		Antagonist
    CMKLR1 antagonist 3 (Compound VU0514009) is a competitive chemokine-like receptor 1 (CMKLR1) antagonist (EC50=2 nM). CMKLR1 antagonist 3 prevents chemerin-9-induced arrestin recruitment and receptor internalization, significantly reducing Ca2+ flux response in HEK293 cells. CMKLR1 antagonist 3 is promising for research of inflammatory diseases and metabolic syndrome.