2. Metabolic Enzyme/Protease
  3. Glutaminase
  4. TG-2-IN-5

TG-2-IN-5 (Compound CP4d) is a reversible TG2 inhibitor with a Ki of 1.0 μM for human TG2. TG-2-IN-5 can be used to study diseases associated with upregulation of TG2-mediated acyl transfer, such as fibrosis and cancer.

For research use only. We do not sell to patients.

TG-2-IN-5

TG-2-IN-5 Chemical Structure

CAS No. : 1082605-61-5

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TG-2-IN-5 Related Antibodies

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Description

TG-2-IN-5 (Compound CP4d) is a reversible TG2 inhibitor with a Ki of 1.0 μM for human TG2. TG-2-IN-5 can be used to study diseases associated with upregulation of TG2-mediated acyl transfer, such as fibrosis and cancer[1].

IC50 & Target

Ki: 1.0 μM for human TG2
Molecular Weight

379.33

Formula

C18H13N5O5
CAS No.
SMILES

O=C(C1=CN(CC2=CC=C([N+]([O-])=O)C=C2)N=N1)/C=C/C3=CC=C([N+]([O-])=O)C=C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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TG-2-IN-5 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

TG-2-IN-51082605-61-5GlutaminasefibrosiscancerInhibitorinhibitorinhibit

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TG-2-IN-5
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HY-176751
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