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Isoforms Recommended:	β adrenergic receptor

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β2 adrenoceptor

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Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-14301

Olodaterol 1 Publications Verification BI1744	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Olodaterol (BI1744) is a selective, long acting *β₂-adrenoceptor* (β₂-AR) agonist (EC₅₀=0.1 nM and pK_i= 9.14 for human β₂-adrenoceptor, respectively). Olodaterol can be used for chronic obstructive pulmonary disease (COPD) and pulmonary fibrosis ^[2] .

HY-14301A

Olodaterol hydrochloride 1 Publications Verification BI1744 hydrochloride	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Olodaterol (BI1744) hydrochloride is a selective, long acting *β₂-adrenoceptor* (β₂-AR) agonist (EC₅₀=0.1 nM and pK_i= 9.14 for human β₂-adrenoceptor, respectively). Olodaterol can be used for chronic obstructive pulmonary disease (COPD) and pulmonary fibrosis ^[2] .

HY-136435

Mapenterol hydrochloride	Adrenergic Receptor	Endocrinology
Mapenterol hydrochloride is a type of *β2-adrenoceptor* agonist .

HY-B0010

Formoterol fumarate 3 Publications Verification (±)Formoterol fumarate	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Formoterol fumarate (Formoterol) is a potent, selective and long-acting β2-adrenoceptor agonist.

HY-12980

Batefenterol GSK961081; TD-5959	Adrenergic Receptor mAChR	Inflammation/Immunology Endocrinology
Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and *β₂-adrenoceptor* agonist; displays high affinity for hM2, hM3 muscarinic and hβ₂-adrenoceptor with K_i values of 1.4, 1.3 and 3.7 nM, respectively.

HY-157502S

Buctopamine-d9	Adrenergic Receptor Isotope-Labeled Compounds	Metabolic Disease
Buctopamine-d9 is the deuterium labeled Buctopamine. Buctopamine is a β2 adrenoceptor agonist .

HY-135487

Sibenadet AR-C68397AA free base; AR-C68397XX	Dopamine Receptor Adrenergic Receptor	Neurological Disease
Sibenadet (AR-C68397AA free base) is a dual dopamine D₂/β₂-adrenoceptor agonist with selective β₂-adrenoceptor agonism. Sibenadet inhibits capsaicin-induced plasma protein extravasation in rat trachea. Sibenadet suppresses edema from sensory nerve fiber activation by activating β₂-adrenoceptor. Sibenadet is promising for research of chronic obstructive pulmonary disease (COPD) .

HY-U00206

D2343	Adrenergic Receptor	Endocrinology
D2343 is a *β2-adrenoceptor* agonist and also is an α1- adrenoceptor inhibitor.

HY-14301AR

Olodaterol (hydrochloride) (Standard)	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Olodaterol (hydrochloride) (Standard) is the analytical standard of Olodaterol (hydrochloride). This product is intended for research and analytical applications. Olodaterol (BI1744) hydrochloride is a selective, long acting *β₂-adrenoceptor* (β₂-AR) agonist (EC₅₀=0.1 nM and pK_i= 9.14 for human β₂-adrenoceptor, respectively). Olodaterol can be used for chronic obstructive pulmonary disease (COPD) and pulmonary fibrosis ^[2] .

HY-19942A

TD-5471 hydrochloride	Adrenergic Receptor	Metabolic Disease Endocrinology
TD-5471 hydrochloride is a potent and selective full agonist of the human *β₂-adrenoceptor*.

HY-12463

Carmoterol hydrochloride	Adrenergic Receptor	Inflammation/Immunology
Carmoterol hydrochloride is a highly potent, selective and long-acting *β2-adrenoceptor* agonist with the pEC₅₀ of 10.19. Carmoterol has 53 times higher affinity for the β2-adrenoceptors than for the β1-adrenoceptors. Carmoterol hydrochloride can be used for the research of asthma and chronic obstructive pulmonary disease (COPD) ^[2].

HY-19942

TD-5471	Adrenergic Receptor	Metabolic Disease Endocrinology
TD-5471 is a potent and selective full agonist of the human *β₂-adrenoceptor* .

HY-12463A

Carmoterol	Adrenergic Receptor	Inflammation/Immunology
Carmoterol is a highly potent, selective and long-acting *β2-adrenoceptor* agonist with the pEC₅₀ of 10.19. Carmoterol has 53 times higher affinity for the β2-adrenoceptors than for the β1-adrenoceptors ^[2]. Carmoterol can be used for the research of asthma and chronic obstructive pulmonary disease (COPD) ^[2].

HY-14300

Vilanterol 5 Publications Verification GW642444	Adrenergic Receptor	Inflammation/Immunology Endocrinology Cancer
Vilanterol (GW642444) is a long-acting *β₂-adrenoceptor* (β₂-AR) agonist with 24 h activity. The pEC₅₀s for β₂-AR,β₁-AR and β₃-AR is 10.37±0.05, 6.98±0.03 and 7.36±0.03, respectively.

HY-14300A

Vilanterol trifenatate 5 Publications Verification GW642444 trifenatate	Adrenergic Receptor	Inflammation/Immunology Endocrinology Cancer
Vilanterol trifenatate (GW642444 trifenatate) is a long-acting *β₂-adrenoceptor* (β₂-AR) agonist with inherent 24-hour activity. The pEC₅₀s for β₂-AR, β₁-AR and β₃-AR are 10.37, 6.98 and 7.36, respectively.

HY-136435S1

Mapenterol-d6 hydrochloride	Isotope-Labeled Compounds Adrenergic Receptor	Endocrinology
Mapenterol-d₆ (hydrochloride) is the deuterium labeled Mapenterol hydrochloride. Mapenterol hydrochloride is a type of β2-adrenoceptor agonist ^[2].

HY-119868

Butaxamine Butoxamin	Adrenergic Receptor	Metabolic Disease
Butaxamine (Butoxamin) is a potent, selective and orally active *β2-adrenoceptor* antagonist. Butaxamine shows antiosteoporotic activity .

HY-100704A

(Rac)-Procaterol hydrochloride	Adrenergic Receptor	Inflammation/Immunology
(Rac)-Procaterol hydrochloride is a selective, orally active agonist at *β2-adrenoceptor*. (Rac)-Procaterol hydrochloride is used as a bronchodilator ^[2].

HY-U00183

Epanolol Visacor; ICI141292	Adrenergic Receptor	Cardiovascular Disease Endocrinology
Epanolol (Visacor; ICI141292) is a potent *β-adrenoceptor* partial agonist with a greater affinity for β1- than β2-adrenoceptors.

HY-10998

Salmefamol AH 3923	Adrenergic Receptor	Inflammation/Immunology
Salmefamol (AH3923) is an orally active *β2-adrenoceptor* agonist. Salmefamol (AH3923) can be used in the study for asthma .

HY-159686

Aclidinium	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Aclidinium is a long-acting muscarinic antagonist and long-acting *β₂-adrenoceptor* (β₂-AR) agonist with bronchodilator activity. Aclidinium can reduce hyperinflation of the lungs and increase lung function and exercise endurance time. Aclidinium is used in research on chronic obstructive pulmonary disease (COPD) .

HY-B0010S

Formoterol-d6 (±)Formoterol-d₆	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology Endocrinology
Formoterol-d₆ is the deuterium labeled Formoterol. Formoterol ((±)Formoterol) is a potent, selective and long-acting β2-adrenoceptor agonist .

HY-124950A

(+)-Picumeterol (+)-GR114297A	Adrenergic Receptor	Metabolic Disease
(+)-Picumeterol is a configurations of Picumeterol (HY-124950). Picumeterol is a potent and selective *β₂-adrenoceptor* agonist with bronchodilator and anti-bronchoconstrictor effects .

HY-14300AS

Vilanterol-d4 trifenatate GW642444-d₄ trifenatate	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology Endocrinology
Vilanterol-d₄ (trifenatate) is deuterium labeled Vilanterol (trifenatate). Vilanterol trifenatate (GW642444 trifenatate) is a long-acting β2-adrenoceptor (β2-AR) agonist with inherent 24-hour activity. The pEC50s for β2-AR, β1-AR and β3-AR are 10.37, 6.98 and 7.36, respectively.

HY-14304

Zinterol MJ 9184	Adrenergic Receptor	Cardiovascular Disease
Zinterol (MJ 9184) is a potent and selective *β2-adrenoceptor* agonist . Zinterol increases I_Ca in a concentration-dependent manner with an EC₅₀ of 2.2 nM ^[2].

HY-117024

Abediterol napadisylate AZD0548 napadisylate; LAS100977 napadisylate	Adrenergic Receptor	Inflammation/Immunology
Abediterol napadisylate is an inhaled long-acting *β2-adrenoceptor* agonist (LABA) and can be used for the research of asthma and chronic obstructive pulmonary disease (COPD) .

HY-101822

Naminterol	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Naminterol is a phenethanolamine derivative, is a β₂ adrenoceptor agonist with bronchodilatory properties. Naminterol is used for treatment of asthma.

HY-14302

Salmeterol Maximum Cited Publications 7 Publications Verification GR33343X	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Salmeterol (GR33343X) is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively .

HY-111144

Abediterol AZD0548; LAS100977	Adrenergic Receptor	Inflammation/Immunology
Abediterol (LAS100977) is an inhaled long-acting *β2-adrenoceptor* agonist (LABA) and can be used for the research of asthma and chronic obstructive pulmonary disease (COPD) .

HY-137909

Formoterol O-β-D-glucuronide	Adrenergic Receptor	Inflammation/Immunology
Formoterol O-β-D-glucuronide is a metabolite of Formoterol (HY-B0010). Formoterol is a potent, selective and long-acting β2-adrenoceptor agonist .

HY-101355A

CGP 20712 dihydrochloride	Adrenergic Receptor	Neurological Disease Endocrinology
CGP 20712 dihydrochloride is a highly selective *β1-adrenoceptor* antagonist with an IC₅₀ of 0.7 nM. CGP 20712 dihydrochloride exhibits ~10,000-fold selectivity over β2-adrenoceptors .

HY-14300S2

Vilanterol-d12 GW642444-d₁₂	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology Endocrinology Cancer
Vilanterol-d₁₂ (GW642444-d₁₂) is deuterium labeled Vilanterol. Vilanterol (GW642444) is a long-acting *β₂-adrenoceptor* (β₂-AR) agonist with 24 h activity. The pEC₅₀s for β₂-AR,β₁-AR and β₃-AR is 10.37±0.05, 6.98±0.03 and 7.36±0.03, respectively.

HY-17453

Salmeterol xinafoate Maximum Cited Publications 7 Publications Verification GR 33343X xinafoate	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Salmeterol (GR 33343X) xinafoate is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively .

HY-107327

Carazolol (±)-Carazolol; DL-Carazolol; Suacron	Adrenergic Receptor	Cardiovascular Disease
Carazolol is a **β₁/β₂ adrenoceptor antagonist of high potency used in the research of hypertension. Carazolol is also a potent, selective β₃-adrenoceptor** agonist .

HY-101355B

CGP 20712 A CGP 20712 mesylate	Adrenergic Receptor	Cardiovascular Disease
CGP 20712 A (CGP 20712 mesylate) is a highly selective *β1-adrenoceptor* antagonist with an IC₅₀ of 0.7 nM. CGP 20712 A exhibits ~10,000-fold selectivity over β2-adrenoceptors .

HY-135119

Salmeterol-d3	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Salmeterol-d₃ is a deuterium labeled Salmeterol. Salmeterol is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively .

HY-135490

Reproterol	Adrenergic Receptor Phosphodiesterase (PDE)	Inflammation/Immunology
Reproterol is a dual acting *β2-adrenoceptor* agonist and PDE inhibitor. The theophylline constituent of Reproterol inhibits phosphodiesterase activity induced by adenylyl cyclase. Reproterol has the potential for asthma research ^[2].

HY-14302S1

Salmeterol-d5 GR33343X-d₅	Isotope-Labeled Compounds Adrenergic Receptor	Endocrinology
Salmeterol-d5 is a deuterated labeled Salmeterol . Salmeterol (GR33343X) is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively ^[2].

HY-W517264

Carazolol hydrochloride BM 51052 hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Carazolol (BM 51052) hydrochloride is a highly potent antagonist of **β₁/β₂ adrenoceptor. Carazolol hydrochloride is also a potent, selective β₃-adrenoceptor** agonist. Carazolol hydrochloride can be used in the research of hypertension .

HY-148527

LAS190792 AZD8999	Adrenergic Receptor mAChR	Others
LAS190792 (AZD8999) is a potent muscarinic antagonist and *β2-adrenoceptor* agonist with pIC₅₀ 8.9, 8.8, 8.8, 9.2, 8.2, 7.5, 9.1, 5.6 for M1, M2, M3, M4, M5, β1, β2, β3, respectively. LAS190792 can be used as a bronchodilator .

HY-17453S

Salmeterol-d3 xinafoate GR 33343X-d₃ xinafoate	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology Endocrinology
Salmeterol-d₃ (xinafoate) is the deuterium labeled Salmeterol xinafoate. Salmeterol (GR 33343X) xinafoate is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively .

HY-17453S1

Salmeterol-13C6 xinafoate GR 33343X-¹³C₆ xinafoate	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology Endocrinology
Salmeterol- ¹³C₆ (xinafoate) is the ¹³C₆ labeled Salmeterol (xinafoate). Salmeterol (GR 33343X) xinafoate is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively.

HY-B0976

Fenoterol Th-1165; Phenoterol	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Fenoterol (Th-1165), a sympathomimetic agent, is a selective and orally active *β2-adrenoceptor* agonist. Fenoterol is an effective bronchodilator and can be used for bronchospasm associated with asthma, bronchitis and other obstructive airway diseases research ^[2].

HY-14304A

Zinterol hydrochloride 1 Publications Verification MJ 9184 hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Zinterol hydrochloride (MJ 9184 hydrochloride) is a potent and selective *β2-adrenoceptor* agonist . Zinterol hydrochloride increases I_Ca in a concentration-dependent manner with an EC₅₀ of 2.2 nM ^[2]. Zinterol hydrochloride induces ventricular arrhythmias in conscious heart failure rabbits .

HY-B0010B

Formoterol-1 (±)Formoterol	Adrenergic Receptor	Inflammation/Immunology
Formoterol ((±)Formoterol) is an orally active β2-selective agonist. Formoterol potently relaxes the peripheral airways through stimulating the beta 2-adrenoceptors selectively as is the case in the central airways and that it significantly inhibits IgE-mediated slow reactive substance of anaphylaxis (SRS-A) release through beta-adrenoceptor stimulation .

HY-50291

HOKU-81 4-Hydroxytulobuterol	Adrenergic Receptor	Cardiovascular Disease Endocrinology
HOKU-81 (4-Hydroxytulobuterol) is one of the metabolites of Tulobuterol (HY-B1810). HOKU-81 is a potent and selective *β2-adrenoceptor* stimulant. HOKU-81 has bronchodilating effect ^[2].

HY-17453R

Salmeterol (xinafoate) (Standard)	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Salmeterol (xinafoate) (Standard) is the analytical standard of Salmeterol (xinafoate). This product is intended for research and analytical applications. Salmeterol (GR 33343X) xinafoate is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively .

HY-157796

β2AR agonist 4	Adrenergic Receptor	Metabolic Disease
β2AR agonist 4 (compound A19) is a potent and selective β2-Adrenoceptor agonist with an EC₅₀ of 3.7 pM. β2AR agonist 4 suppresses the inflammatory cytokines and leukocytes upregulation and improves lung function in COPD rat model .

HY-107327R

Carazolol (Standard)	Adrenergic Receptor	Cardiovascular Disease
Carazolol (Standard) is the analytical standard of Carazolol. This product is intended for research and analytical applications. Carazolol is a **β₁/β₂ adrenoceptor antagonist of high potency used in the research of hypertension. Carazolol is also a potent, selective β₃-adrenoceptor** agonist .

HY-101355AR

CGP 20712 dihydrochloride (Standard)	Adrenergic Receptor Reference Standards	Neurological Disease Endocrinology
CGP 20712 (dihydrochloride) (Standard) is the analytical standard of CGP 20712 (dihydrochloride). This product is intended for research and analytical applications. CGP 20712 dihydrochloride is a highly selective β1-adrenoceptor antagonist with an IC50 of 0.7 nM. CGP 20712 dihydrochloride exhibits ~10,000-fold selectivity over β2-adrenoceptors .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-136409R

N-Decanoyl-L-homoserine lactone (Standard)	Microorganisms Source classification	Bacterial Reactive Oxygen Species
Formoterol (hemifumarate hydrate) (Standard) is the analytical standard of Formoterol (hemifumarate hydrate). This product is intended for research and analytical applications. Formoterol hemifumarate hydrate is a selective, long-acting beta 2-adrenoceptor agonist. Formoterol is a bronchodilator used for the research of the asthma and chronic obstructive pulmonary disease (COPD). Formoterol hemifumarate hydrate induces mitochondrial biogenesis and promotes cognitive recovery after traumatic brain injury ^[2] .

HY-N8268R

Nordeoxycholic acid (Standard)	Animals Source classification	Drug Metabolite
Reproterol (hydrochloride) (Standard) is the analytical standard of Reproterol (hydrochloride). This product is intended for research and analytical applications. Reproterol hydrochloride is a dual-acting beta2-adrenoceptor agonist and phosphodiesterase inhibitor. Reproterol hydrochloride is more potent than albuterol and feterol in stimulating cAMP production in human monocytes, demonstrating its potential in enhancing airway function. Furthermore, Reproterol significantly inhibited the production of LTB4, indicating its anti-inflammatory properties. Reproterol hydrochloride may have inhibitory effects in respiratory diseases such as asthma and COPD .

Cat. No.	Compare	Product Name	Species	Source

HY-P702206

	ADRB2 Protein, Human (Cell-Free, His, SUMO) Beta-2 adrenergic receptor; Beta-2 adrenoreceptor; Beta-2 adrenoceptor	Human	E. coli Cell-free
	ADRB2 protein is an important member of the β-adrenergic receptor family and mediates catecholamine-induced adenylyl cyclase activation through G protein action. It has 30 times greater affinity for epinephrine and plays a crucial role in cellular responses to sympathetic nervous system stimulation. ADRB2 Protein, Human (Cell-Free, His, SUMO) is the recombinant human-derived ADRB2 protein, expressed by E. coli Cell-free , with N-6*His, N-SUMO labeled tag and G16R, E27Q mutation.

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Cat. No.	Product Name	Chemical Structure

HY-135119

Salmeterol-d3
Salmeterol-d₃ is a deuterium labeled Salmeterol. Salmeterol is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively .

HY-107327S

Carazolol-d7
Carazolol-d₇ is the deuterium labeled Carazolol (HY-107327). Carazolol is a highly potent antagonist of **β₁/β₂ adrenoceptor. Carazolol is also a potent, selective β₃-adrenoceptor** agonist. Carazolol can be used in the research of hypertension .

HY-157502S

Buctopamine-d9
Buctopamine-d9 is the deuterium labeled Buctopamine. Buctopamine is a β2 adrenoceptor agonist .

HY-136435S1

Mapenterol-d6 hydrochloride
Mapenterol-d₆ (hydrochloride) is the deuterium labeled Mapenterol hydrochloride. Mapenterol hydrochloride is a type of β2-adrenoceptor agonist ^[2].

HY-B0010S

Formoterol-d6
Formoterol-d₆ is the deuterium labeled Formoterol. Formoterol ((±)Formoterol) is a potent, selective and long-acting β2-adrenoceptor agonist .

HY-14300AS

Vilanterol-d4 trifenatate
Vilanterol-d₄ (trifenatate) is deuterium labeled Vilanterol (trifenatate). Vilanterol trifenatate (GW642444 trifenatate) is a long-acting β2-adrenoceptor (β2-AR) agonist with inherent 24-hour activity. The pEC50s for β2-AR, β1-AR and β3-AR are 10.37, 6.98 and 7.36, respectively.

HY-14300S2

Vilanterol-d12
Vilanterol-d₁₂ (GW642444-d₁₂) is deuterium labeled Vilanterol. Vilanterol (GW642444) is a long-acting *β₂-adrenoceptor* (β₂-AR) agonist with 24 h activity. The pEC₅₀s for β₂-AR,β₁-AR and β₃-AR is 10.37±0.05, 6.98±0.03 and 7.36±0.03, respectively.

HY-14302S1

Salmeterol-d5
Salmeterol-d5 is a deuterated labeled Salmeterol . Salmeterol (GR33343X) is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively ^[2].

HY-17453S

Salmeterol-d3 xinafoate
Salmeterol-d₃ (xinafoate) is the deuterium labeled Salmeterol xinafoate. Salmeterol (GR 33343X) xinafoate is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC₅₀s of 9.6, 6.1, and 5.9, respectively .

HY-17453S1

Salmeterol-13C6 xinafoate
Salmeterol- ¹³C₆ (xinafoate) is the ¹³C₆ labeled Salmeterol (xinafoate). Salmeterol (GR 33343X) xinafoate is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively.

HY-107327S1

Carazolol-d7 hydrochloride
Carazolol-d₇ (hydrochloride) is the deuterium labeled Carazolol hydrochloride (HY-W517264). Carazolol hydrochloride is a highly potent antagonist of **β₁/β₂ adrenoceptor. Carazolol hydrochloride is also a potent, selective β₃-adrenoceptor** agonist. Carazolol hydrochloride can be used in the research of hypertension .

HY-W777156

Carazolol-d6 hydrochloride
Carazolol-d₆ (hydrochloride) is deuterium labeled Carazolol hydrochloride (HY-W517264). Carazolol hydrochloride is a highly potent antagonist of **β₁/β₂ adrenoceptor. Carazolol hydrochloride is also a potent, selective β₃-adrenoceptor** agonist. Carazolol hydrochloride can be used in the research of hypertension .

HY-15746S1

(rac)-Dobutamine-d6 hydrochloride

(rac)-Dobutamine-d₆ (hydrochloride) is a labelled racemic Dobutamine hydrochloride. Dobutamine hydrochloride is a synthetic catecholamine that acts on α1-AR, β1-AR, β2-AR (α-1, β-1 andβ-2 adrenoceptors). Dobutamine hydrochloride is a selective β1-AR agonist, relatively weak activity at α1-AR and β2-AR. Dobutamine hydrochloride can increase cardiac output and correct hypoperfusion ^[2] .

HY-15746S

(rac)-Dobutamine-d4 hydrochloride

(rac)-Dobutamine-d₄ (hydrochloride) is a labelled racemic Dobutamine hydrochloride. Dobutamine hydrochloride is a synthetic catecholamine that acts on α1-AR, β1-AR, β2-AR (α-1, β-1 andβ-2 adrenoceptors). Dobutamine hydrochloride is a selective β1-AR agonist, relatively weak activity at α1-AR and β2-AR. Dobutamine hydrochloride can increase cardiac output and correct hypoperfusion ^[2] .

HY-B1810S

Tulobuterol-d9 hydrochloride
Tulobuterol-d₉ (hydrochloride) is the deuterium labeled Tulobuterol. Tulobuterol (C-78 free base) is a long-acting β2-adrenoceptor agonist, which reduces the frequency of exacerbations of chronic obstructive pulmonary disease and bronchial asthma. Tulobuterol is also a sympathomimetic agent used as a transdermal patch, and increases normal diaphragm muscle strength .

HY-B0976AS

Fenoterol-d6 hydrobromide
Fenoterol-d₆ (hydrobromide) (Th-1165a-d₆) is the deuterium labeled Fenoterol hydrobromide. Fenoterol hydrobromide (Th-1165a), a sympathomimetic agent, is a selective and orally active β2-adrenoceptor agonist. Fenoterol hydrobromide is an effective bronchodilator and can be used for bronchospasm associated with asthma, bronchitis and other obstructive airway diseases research ^[2].

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