2. PROTAC Metabolic Enzyme/Protease Cell Cycle/DNA Damage
  3. PROTACs PDI
  4. PROTAC PDIA1 degrader 1

PROTAC PDIA1 degrader 1 (Compound H4) is a PDIA1 PROTAC degrader with a DC50 of 29.71 μM. PROTAC PDIA1 degrader 1 has potent anticancer activity and significantly inhibits cancer cell proliferation. Pink: PDIA1 ligand (HY-100433); Blue: CRBN ligase ligand (HY-10984); Black: linker (HY-W015088)

For research use only. We do not sell to patients.

PROTAC PDIA1 degrader 1

PROTAC PDIA1 degrader 1 Chemical Structure

CAS No. : 3024292-21-2

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PROTAC PDIA1 degrader 1 Related Antibodies

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Description

PROTAC PDIA1 degrader 1 (Compound H4) is a PDIA1 PROTAC degrader with a DC50 of 29.71 μM. PROTAC PDIA1 degrader 1 has potent anticancer activity and significantly inhibits cancer cell proliferation[1]. Pink: PDIA1 ligand (HY-100433); Blue: CRBN ligase ligand (HY-10984); Black: linker (HY-W015088)

Molecular Weight

832.88

Formula

C40H44N6O12S
CAS No.
SMILES

COC1=C(N(C(C#C)=O)C(C(NCC(NCCOCCOCCOCCNC2=C(C(N(C3C(NC(CC3)=O)=O)C4=O)=O)C4=CC=C2)=O)=O)C5=CC=CS5)C=CC(OC)=C1
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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PROTAC PDIA1 degrader 1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PROTAC PDIA1 degrader 13024292-21-2PROTACsPDIProtein Disulfide IsomerasesPROTACDegradationPDIA1AnticancerA431 cellsMCF-7 cellsInhibitorinhibitorinhibit

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PROTAC PDIA1 degrader 1
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