2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. iGluR
  4. EU 1622-240

EU 1622-240 is a biased positive allosteric modulator of GluN2B, GluN2C, and GluN2D, with EC50s of 0.57, 0.82, 1.1 μM respectively. EU 1622-240 has good physicochemical properties, in vitro stability, and permeability.

For research use only. We do not sell to patients.

EU 1622-240 Chemical Structure

EU 1622-240 Chemical Structure

CAS No. : 3057728-22-7

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EU 1622-240 Related Antibodies

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Description

EU 1622-240 is a biased positive allosteric modulator of GluN2B, GluN2C, and GluN2D, with EC50s of 0.57, 0.82, 1.1 μM respectively. EU 1622-240 has good physicochemical properties, in vitro stability, and permeability[1].

Molecular Weight

478.31

Formula

C20H14BrF2N3O2S
CAS No.
SMILES

C#CC1=C(C2=C(N=CN(C2=O)CC(N3CC(F)(C3)C)=O)S1)C4=CC=C(C(Br)=C4)F
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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EU 1622-240 Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

EU 1622-2403057728-22-7iGluRIonotropic glutamate receptorsGluN2BGluN2CGluN2DInhibitorinhibitorinhibit

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