2. Apoptosis
  3. MDM-2/p53 Apoptosis Ferroptosis
  4. Eprenetapopt

Eprenetapopt (GMP) (APR-246(GMP)) is Eprenetapopt (HY-19980) in GMP grade. Eprenetapopt (APR-246) is a first-in-class, small molecule that restores wild-type p53 functions in TP53-mutant cells. Eprenetapopt triggers apoptosis in tumor cells. Eprenetapopt also targets the selenoprotein thioredoxin reductase 1 (TrxR1), a key regulator of cellular redox balance.

For research use only. We do not sell to patients.

Eprenetapopt Chemical Structure

Eprenetapopt Chemical Structure

CAS No. : 5291-32-7

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Eprenetapopt Related Antibodies

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Description

Eprenetapopt (GMP) (APR-246(GMP)) is Eprenetapopt (HY-19980) in GMP grade. Eprenetapopt (APR-246) is a first-in-class, small molecule that restores wild-type p53 functions in TP53-mutant cells. Eprenetapopt triggers apoptosis in tumor cells. Eprenetapopt also targets the selenoprotein thioredoxin reductase 1 (TrxR1), a key regulator of cellular redox balance[1][2][3].

Molecular Weight

199.25

Formula

C10H17NO3
CAS No.
SMILES

O=C1C(COC)(CO)N2CCC1CC2
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Room temperature in continental US; may vary elsewhere.
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Purity & Documentation
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Eprenetapopt Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Eprenetapopt (GMP)5291-32-7APR-246 (GMP)PRIMA-1Met (GMP)MDM-2/p53ApoptosisFerroptosisp53apoptosiswild-type p53TP53-mutantthioredoxin reductase 1 (TrxR1)Inhibitorinhibitorinhibit

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HY-19980G
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