2. Membrane Transporter/Ion Channel
  3. OAT URAT1
  4. Epaminurad hydrochloride

Epaminurad hydrochloride  (Synonyms: UR-1102 hydrochloride; URC-102 hydrochloride)

Cat. No.: HY-111345A
Handling Instructions Technical Support

Epaminurad (UR-1102) hydrochloride is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad hydrochloride quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad hydrochloride is a uricosuric agent. Epaminurad hydrochloride can be used for gout and hyperuricemia research.

For research use only. We do not sell to patients.

Epaminurad hydrochloride

Epaminurad hydrochloride Chemical Structure

CAS No. : 1198153-46-6

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Epaminurad hydrochloride Related Antibodies

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Description

Epaminurad (UR-1102) hydrochloride is an orally active, potent and selective URAT1 (urate transporter 1) inhibitor, with a Ki of 0.057 μM. Epaminurad hydrochloride quite modestly inhibits OAT1 and OAT3 (organic anion transporter). Epaminurad hydrochloride is a uricosuric agent. Epaminurad hydrochloride can be used for gout and hyperuricemia research[1].

IC50 & Target

Ki: 0.057 ± 0.036 μM (URAT1), 2.4 ± 0.2 μM (OAT3), 7.2 ± 0.8 μM (OAT1)[1].
Clinical Trial
Molecular Weight

450.51

Formula

C14H11Br2ClN2O3
CAS No.
SMILES

O=C(N1C2=C(OCC1)C=CN=C2)C3=CC(Br)=C(C(Br)=C3)O.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Epaminurad hydrochloride Related Classifications

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Epaminurad1198153-46-6UR-1102URC-102UR1102UR 1102URC102URC 102OATURAT1Organic anion transporterUrate transporter 1SLC22A12HEK293 cellsUricosuricgouthyperuricemiap-aminohippuric acidurateInhibitorinhibitorinhibit

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