2. PROTAC Epigenetics
  3. Target Protein Ligand-Linker Conjugates Epigenetic Reader Domain
  4. CPI-203-PEG1-C3-O-COOH

CPI-203-PEG1-C3-O-COOH is a conjugate of the BRD4 ligand (HY-78695) and the linker (HY-42427). CPI-203-PEG1-C3-O-COOH can be used for synthesizing PROTAC BRD4 degrader ARV-771 (HY-100972).

For research use only. We do not sell to patients.

CPI-203-PEG1-C3-O-COOH

CPI-203-PEG1-C3-O-COOH Chemical Structure

CAS No. : 1997304-12-7

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CPI-203-PEG1-C3-O-COOH Related Antibodies

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Description

CPI-203-PEG1-C3-O-COOH is a conjugate of the BRD4 ligand (HY-78695) and the linker (HY-42427). CPI-203-PEG1-C3-O-COOH can be used for synthesizing PROTAC BRD4 degrader ARV-771 (HY-100972)[1].

Molecular Weight

560.06

Formula

C26H30ClN5O5S
CAS No.
SMILES

CC1=C(C)C(C(C2=CC=C(Cl)C=C2)=N[C@@H](CC(NCCOCCCOCC(O)=O)=O)C3=NN=C(C)N34)=C4S1
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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CPI-203-PEG1-C3-O-COOH Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CPI-203-PEG1-C3-O-COOH1997304-12-7Target Protein Ligand-Linker ConjugatesEpigenetic Reader DomainBRD4CancerInhibitorinhibitorinhibit

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CPI-203-PEG1-C3-O-COOH
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HY-42429
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