2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. Amauromine

Amauromine is a peripheral selective cannabinoid receptor type 1 (CB1) receptor antagonist with Ki and Kb values of 178 nM and 66.6 nM, respectively.

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Amauromine

Amauromine Chemical Structure

CAS No. : 88360-87-6

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Based on 1 publication(s) in Google Scholar

Amauromine Related Antibodies

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Description

Amauromine is a peripheral selective cannabinoid receptor type 1 (CB1) receptor antagonist with Ki and Kb values of 178 nM and 66.6 nM, respectively[1].

IC50 & Target

CB1

178 nM (Ki)

CB1

66.6 nM (Kb)

Molecular Weight

508.65

Formula

C32H36N4O2
CAS No.
SMILES

C=CC(C)([C@]12[C@](NC3=CC=CC=C23)([H])N4[C@@](C(N5[C@](C[C@]6(C(C)(C)C=C)[C@@]5([H])NC7=CC=CC=C67)([H])C4=O)=O)([H])C1)C
Structure Classification
Initial Source

Auxarthron reticulatum
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Amauromine Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Amauromine88360-87-6Cannabinoid ReceptorAuxarthron reticulatumamaurominecannabinoid receptorsCB1CB2natural productsInhibitorinhibitorinhibit

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