1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    PI3K/Akt/mTOR
  3. ATM/ATR
  4. ATM/ATR Inhibitors

ATM/ATR Inhibitors

ATM

ATR

TRRAP

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

ATM/ATR Inhibitors & Activators
Product Name ATM ATR TRRAP Purity
AZD-7648
ATM, IC50: 17.93 μM
    99.86%
Ceralasertib  
ATR, IC50: 1 nM
  99.76%
KU-55933
ATM, IC50: 12.9 nM
    99.92%
VE-821
ATM, Ki: 16 μM
ATR, Ki: 13 nM
  99.67%
Berzosertib
ATM, Ki: 34 nM
ATR, Ki: 0.2 nM
  99.70%
ATR/PARP1-IN-1
ATM, IC50: >5000 nM
ATR, IC50: 17.3 nM
 
AZD-7648 (GMP)
ATM, IC50: 17.93
   
Elimusertib  
ATR, IC50: 7 nM
  99.99%
KU-60019
ATM, IC50: 6.3 nM
    99.43%
AZD0156
ATM
    99.83%
AZD1390
ATM
    99.22%
Camonsertib
ATM, IC50: >30 μM
    99.75%
Gartisertib  
ATR, Ki: <150 pM
  99.77%
AZ20  
ATR, IC50: 5 nM
  99.40%
Lartesertib
ATM
    99.94%
Elimusertib hydrochloride  
ATR, IC50: 7 nM
  99.85%
CGK733
ATM
ATR
  99.83%
CP-466722
ATM, IC50: 4.1 μM
    99.74%
ETP-46464
ATM, IC50: 545 nM
ATR, IC50: 14 nM
  99.54%
Ro 90-7501
ATM
    99.10%
Garcinone C  
ATR
  99.66%
AD1058  
ATR, IC50: 1.6 nM
  98.11%
AZ32
ATM, IC50: 6.2 nM
ATM, IC50: 0.31 μM (in cell)
    99.94%
AZ31
ATM, IC50: 1.2 nM
ATM, IC50: 46 nM (in cell)
    98.13%
NU6027  
ATR
  99.04%
ATR kinase substrate peptide  
ATR, Ki: 6 nM
  99.17%
ATM Inhibitor-1
ATM, IC50: 0.7 nM
ATM, IC50: 2.8 nM (Cellular assay)
   
ATR-IN-14  
ATR
 
ATM Inhibitor-3
ATM, IC50: 0.71 nM
   
ATM Inhibitor-7
ATM, IC50: 1.0 nM
   
ATM Inhibitor-4
ATM, IC50: 0.32 nM
   
ICT10336  
ATR
 
ATM Inhibitor-11
ATM, IC50: 0.32 nM
   
Abd110  
ATR
 
ATR-IN-10  
ATR, IC50: 2.978 μM
 
ATR-IN-19  
ATR
 
ATR-IN-15
ATM, IC50: > 10000 nM
ATR, IC50: 8 nM
 
ATR-IN-21  
ATR, IC50: <1000 nM
 
ATR-IN-17  
ATR
 
ATM Inhibitor-2
ATM, IC50: <1 nM
   
ATR-IN-20
ATM, IC50: 100 nM
ATR, IC50: 3 nM
 
Antitumor agent-28
ATM
ATR
 
ATR-IN-29  
ATR, IC50: 1 nM
 
ATR-IN-13  
ATR, IC50: 2 nM
 
ATR-IN-18  
ATR, IC50: 0.69 nM
 
ATR-IN-16  
ATR
 
Trrap Mouse Pre-designed siRNA Set A    
TRRAP