1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. Src
  4. Src Inhibitors

Src Inhibitors

Lck

Fyn

Blk

Hck

Lyn

Yes

SRC-3

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Src Degraders & Inhibitors
Product Name Lck Fyn Blk Hck Lyn Yes SRC-3 Purity
PRT062607 Hydrochloride
Lck, IC50: 249 nM ([2])
            98.07%
GLPG3312
Lck, IC50: 385 nM
Fyn, IC50: 447 nM
Blk, IC50: 730 nM
Hck, IC50: 2511 nM
Lyn, IC50: 272 nM
Yes, IC50: 598 nM
  98.57%
Velzatinib
Lck, IC50: 141 nM
            99.47%
AZM475271
Lck, IC50: 0.03 μM
            99.89%
SB 220025
p56-Lck, IC50: 3.5 μM
            99.90%
PRT062607 acetate
Lck, IC50: 249 nM ([2])
            99.83%
RK-20448
Lck, IC50: 0.24 μM
Fyn, IC50: 2.03 μM
Blk, IC50: 0.37 μM
        99.38%
Lck-IN-2
Lck, IC50: 10.6 nM
           
Antifibrotic agent 1
Lck
Fyn
 
Hck
Lyn
Yes
 
BY13            
SRC-3, DC50: 0.031 μM
BMS-243117
Lck, IC50: 4 nM
Fyn, IC50: 32 nM
Blk, IC50: 84 nM