2. Signaling Pathways
  3. GPCR/G Protein
    Neuronal Signaling
  4. Neurokinin Receptor
  5. Neurokinin Receptor Isoform
  6. Neurokinin Receptor Antagonist

Neurokinin Receptor Antagonist

Neurokinin Receptor Antagonists (85):

Cat. No. Product Name Effect Purity
  • HY-P2603
    Bz-Dab(NBD)-AwFpP-Nle-NH2
    		Antagonist
    Bz-Dab(NBD)-AwFpP-Nle-NH2 (Compound 5B) is a potent fluorescent antagonist of NK2 receptor, with a pKi of 8.87 nM (Ex=340 nm, Em=505 nm).
  • HY-P2436
    L-659837
    		Antagonist
    L-659837 is a NK2 receptor antagonist, and can antagonize GR 64349 (HY-P1278)-induced contraction. L-659837 can be used for study of urinary bladder disorders.
  • HY-118356
    WIN 62,577
    		Antagonist
    WIN 62,577 is a rat-specific, but non-human, NK1 receptor antagonist. WIN 62,577 interacts with M1-M4 mAChRs and is an allosteric enhancer of acetylcholine affinity targeting the M3 receptor.
  • HY-U00392
    Tachykinin angatonist 1
    		Antagonist
    Tachykinin angatonist 1 is a neurokinin receptor antagonist extracted from patent US5968923, compound example 32.
  • HY-U00320
    Neurokinin antagonist 1
    		Antagonist
    Neurokinin antagonist 1 is a Neurokinin antagonist extracted from patent WO1998045262A1.